Target Details
| UniProt AC | P06493 |
|---|---|
| Gene Symbol | CDK1 |
| Protein Name | Cyclin-dependent kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,900
- Clinical molecules 608
- Avg pChEMBL 7.06
KEGG Pathways (8)
Active Molecules (1,900)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MRPGRAKIAJJGMM
|
7.6 | IC50 | 11 | — | |
MVJMMLFMPWITEJ
|
7.6 | Ki | 110 | — | |
OVJIHFBAXJKTRF
|
7.6 | IC50 | 2 | — | |
RXGQFYCBXVUJTL
|
7.6 | IC50 | 4 | — | |
UTBSBSOBZHXMHI
|
7.6 | pIC50 | 15 | Yes | |
WFNUAOKMXUQUHV
|
7.6 | IC50 | 3 | — | |
WLTRIWCDHOZNRP
|
7.6 | IC50 | 14 | — | |
WYEXOAKSTKXOBU
|
7.6 | IC50 | 3 | — | |
XFWUTMHVDGPWLH
|
7.6 | Ki | 75 | — | |
FUZBMVCWAVMNGW
|
7.6 | pIC50 | 2 | Yes | |
IYNDTACKOAXKBJ
|
7.6 | IC50 | 17 | — | |
XPLSUUKNUUIIKH
|
7.6 | pIC50 | 2 | Yes | |
CGKJOISVQXEPSG
|
7.6 | Ki | 9 | — | |
GWODBBFDCZIKBY
|
7.6 | IC50 | 2 | — | |
MCFCYLCLAYXQIZ
|
7.6 | Ki | 9 | — | |
PYEYLKGWDVDOAS
|
7.6 | pIC50 | 9 | Yes | |
SOHOEERULHWXJB
|
7.6 | IC50 | 5 | — | |
VIIIAPSCTBJJNE
|
7.6 | pIC50 | 4 | Yes | |
AMHWMCSHBYIXCE
|
7.6 | IC50 | 3 | — | |
CXDXSBLYPKFPLO
|
7.6 | IC50 | 3 | — | |
DLNVXQGIVOPKFV
|
7.6 | IC50 | 3 | — | |
HEFHQIBQGOCQAF
|
7.6 | pIC50 | 11 | Yes | |
KMHNZVWSMBCPMT
|
7.6 | IC50 | 8 | — | |
MROGTPNQSHMKIG
|
7.6 | pIC50 | 2 | Yes | |
VASFNXBXECJRSY
|
7.6 | IC50 | 15 | — | |
HGAFXPHIIHJZEB
|
7.5 | pIC50 | 2 | Yes | |
MGYDUQVCVWCQMO
|
7.5 | Ki | 6 | — | |
PSWIPMICOQJHRP
|
7.5 | IC50 | 3 | — | |
YREVWYJUWQLUFX
|
7.5 | IC50 | 2 | Yes | |
LOYSCNBYDPTSAA
|
7.5 | IC50 | 10 | — | |
OPVFXMUETZOYIY
|
7.5 | IC50 | 2 | — | |
QSDYIYAFRFRSKH
|
7.5 | IC50 | 2 | — | |
IHBOEHLUIBMBMY
|
7.5 | pIC50 | 7 | Yes | |
BIIVYFLTOXDAOV
|
7.5 | IC50 | 3 | — | |
BIIVYFLTOXDAOV
|
7.5 | pIC50 | 82 | Yes | |
DVTLAQZTCJXBPC
|
7.5 | pIC50 | 2 | Yes | |
SJIUAJVZBGNRFY
|
7.5 | IC50 | 3 | — | |
TUSYHQBFGFIWOG
|
7.5 | pIC50 | 5 | Yes | |
WIXXUCKYLZMMCZ
|
7.5 | IC50 | 3 | — | |
CEZKUHAOXFVYTL
|
7.5 | IC50 | 2 | — | |
CIBIVMWDVTYWNT
|
7.5 | IC50 | 2 | Yes | |
LDNQAJNFIYSIHK
|
7.5 | pIC50 | 3 | Yes | |
TYSWNLQZLBRNSE
|
7.5 | IC50 | 15 | — | |
UFDKTUULSMNAME
|
7.5 | IC50 | 2 | Yes | |
UOXBVHRCZIPJEI
|
7.5 | IC50 | 4 | — | |
AOBLBPWPSKBHSI
|
7.5 | Ki | 55 | — | |
BIIVYFLTOXDAOV
|
7.5 | Ki | 31 | — | |
BSDJIQDLIJZWHF
|
7.5 | pIC50 | 8 | Yes | |
CLEGDJQQHUTCOW
|
7.5 | Ki | 43 | — | |
JXSGQHRSUUOSAF
|
7.5 | pIC50 | 3 | Yes |