Target Details
| UniProt AC | P06493 |
|---|---|
| Gene Symbol | CDK1 |
| Protein Name | Cyclin-dependent kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,900
- Clinical molecules 608
- Avg pChEMBL 7.06
KEGG Pathways (8)
Active Molecules (1,900)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FKAJEPVSQITQLJ
|
7.7 | IC50 | 15 | — | |
FLEAYYMORDPWAJ
|
7.7 | Ki | 90 | — | |
FMUUGBFOPCVEBP
|
7.7 | IC50 | 7 | — | |
GCYXEGSPUDSZJY
|
7.7 | Ki | 82 | — | |
JFSGUSJACVSEKX
|
7.7 | pIC50 | 7 | Yes | |
NDUNPMAPBHPTHE
|
7.7 | pIC50 | 8 | Yes | |
NLUPJKQOKWBWFC
|
7.7 | Ki | 69 | — | |
SSMMYRQDZBSVCY
|
7.7 | pIC50 | 7 | Yes | |
TVOSCVSFFYTFBC
|
7.7 | IC50 | 2 | Yes | |
VBDQMJNIWDFAKI
|
7.7 | pIC50 | 8 | Yes | |
WNMRVXGHICLEOM
|
7.7 | pIC50 | 3 | Yes | |
AAYPLLWGPJQWCC
|
7.7 | pIC50 | 15 | Yes | |
AHFARWUGWOGTLO
|
7.7 | IC50 | 3 | — | |
LNPGEMWHMALOTH
|
7.7 | pIC50 | 2 | Yes | |
MBKBRIBQHFBRHO
|
7.7 | IC50 | 3 | — | |
QENSBTHLGFPXQZ
|
7.7 | IC50 | 3 | — | |
UVNWLDYNLOHPKC
|
7.7 | IC50 | 5 | — | |
SUMQWZPREGGMNQ
|
7.7 | IC50 | 6 | — | |
WSYHYLUWICJSJV
|
7.7 | IC50 | 8 | — | |
ATBAETXFFCOZOY
|
7.7 | IC50 | 39 | — | |
ATBAETXFFCOZOY
|
7.7 | IC50 | 10 | — | |
CPGPEVNIOCXOPN
|
7.7 | IC50 | 3 | — | |
KHGITEBUGKISDS
|
7.7 | pIC50 | 4 | Yes | |
MKCHHXTWUNRKMA
|
7.7 | IC50 | 3 | — | |
OARXLGLBMAHALM
|
7.7 | IC50 | 12 | Yes | |
ONVJWTCYZZHCFH
|
7.7 | pIC50 | 2 | Yes | |
DLFSESWOWKXVMD
|
7.7 | pIC50 | 3 | Yes | |
GGRVRRFOVWKWMD
|
7.6 | IC50 | 11 | — | |
IOCPGDFUHJLQTO
|
7.6 | IC50 | 2 | Yes | |
MRAOFFFVZQWILN
|
7.6 | pIC50 | 3 | Yes | |
OTPNDVKVEAIXTI
|
7.6 | Ki | 4 | — | |
QSGKPYRFWJINEH
|
7.6 | IC50 | 12 | — | |
UBDAMLJKQGPQFB
|
7.6 | pIC50 | 2 | Yes | |
UVKIWKFJDSCWJY
|
7.6 | IC50 | 3 | — | |
XFWNXRYYGPIPLI
|
7.6 | pIC50 | 6 | Yes | |
ACNJMIYZGUUYIE
|
7.6 | pIC50 | 3 | Yes | |
AGIIDJZSMZSLJN
|
7.6 | pIC50 | 9 | Yes | |
CDKIUTDNGTUHKC
|
7.6 | IC50 | 3 | — | |
CKIFWVSQRJHDKI
|
7.6 | Ki | 9 | — | |
GTQSNWXKTIFPBY
|
7.6 | IC50 | 5 | — | |
KYRQRRGDKAIFMA
|
7.6 | IC50 | 7 | — | |
LBVIZFWUIQSZHP
|
7.6 | IC50 | 10 | — | |
MSGWNYXBVMCUNQ
|
7.6 | IC50 | 3 | — | |
NKRSLISCOPHPJT
|
7.6 | IC50 | 3 | — | |
QYLYUTQSYHCBOD
|
7.6 | IC50 | 13 | — | |
SZDPBHAPNGSXHF
|
7.6 | pIC50 | 4 | Yes | |
WMUSBRFXXCFZTI
|
7.6 | pIC50 | 2 | Yes | |
DXXJDEVFDVVIGG
|
7.6 | IC50 | 2 | — | |
HOPYTUITHBXQSC
|
7.6 | pIC50 | 5 | Yes | |
MKJQNJOYGXZGII
|
7.6 | pIC50 | 4 | Yes |