Target Details
| UniProt AC | P06493 |
|---|---|
| Gene Symbol | CDK1 |
| Protein Name | Cyclin-dependent kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,900
- Clinical molecules 608
- Avg pChEMBL 7.06
KEGG Pathways (8)
Active Molecules (1,900)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WFRNKIOQSRRDQF
|
7.8 | IC50 | 3 | — | |
YZUCJGXJSJSVQK
|
7.8 | IC50 | 2 | Yes | |
DASFSPDIWCMVRW
|
7.8 | Ki | 21 | — | |
HNMARRTVPIAGPR
|
7.8 | IC50 | 3 | — | |
JWOJZWRKDLDOEO
|
7.8 | IC50 | 3 | — | |
KKKIPUHVQOUJTL
|
7.8 | IC50 | 2 | — | |
MEKQZIRNPYPHGO
|
7.8 | pIC50 | 3 | Yes | |
RBWPUACOPXHFHA
|
7.8 | pIC50 | 2 | Yes | |
VWVYILCFSYNJHF
|
7.8 | Ki | 49 | — | |
WJRRGYBTGDJBFX
|
7.8 | IC50 | 16 | Yes | |
XEXXLSSPQTWUID
|
7.8 | IC50 | 3 | — | |
IJIGRXABGQBDBA
|
7.8 | Ki | 10 | — | |
ZTEGEMFKBZMGOF
|
7.8 | IC50 | 9 | — | |
BNXUVHSQMZRHIA
|
7.8 | pIC50 | 3 | Yes | |
NSGQRIPFMLCLFH
|
7.8 | pIC50 | 8 | Yes | |
PAEDTQQTYBULPN
|
7.8 | IC50 | 4 | — | |
DIXITDIZTSWFDW
|
7.8 | pIC50 | 4 | Yes | |
DULGHLDQYKRXTJ
|
7.8 | IC50 | 3 | — | |
JNLCGKQCDLVQAH
|
7.8 | IC50 | 2 | — | |
ZWVNPBSQSAHHNR
|
7.8 | IC50 | 11 | Yes | |
HFMGTBLBSYZDFW
|
7.8 | pIC50 | 8 | Yes | |
SYQYDDZJODBESY
|
7.8 | pIC50 | 3 | Yes | |
IIJWYFPAKYPUIM
|
7.8 | IC50 | 8 | — | |
ASUFRYKYWHJUIO
|
7.7 | Ki | 9 | — | |
GNHNRVSQWNAGHC
|
7.7 | pIC50 | 7 | Yes | |
HXZXJLLRGFULES
|
7.7 | Ki | 9 | — | |
IOKHECWXZNKBBH
|
7.7 | pIC50 | 2 | Yes | |
QUDNAUWPTMNNHI
|
7.7 | IC50 | 8 | Yes | |
UYSFMAROJRGQCA
|
7.7 | pIC50 | 3 | Yes | |
WWAYNSNYYIIADR
|
7.7 | IC50 | 2 | — | |
XKDKTKPNGXUGSV
|
7.7 | pIC50 | 3 | Yes | |
YARIHEYYGBAEDE
|
7.7 | Ki | 10 | — | |
ANWMSXOBKGKAOJ
|
7.7 | Ki | 6 | — | |
BIOJVWLNPPOUGW
|
7.7 | IC50 | 3 | — | |
DAKPITMJALLHHF
|
7.7 | pIC50 | 2 | Yes | |
DINLHKGZVRGQQO
|
7.7 | IC50 | 3 | — | |
DMGXKGMPNXDFPN
|
7.7 | IC50 | 2 | — | |
HCSOUJXRCJMNFB
|
7.7 | pIC50 | 8 | Yes | |
IZIPWCFRXVNDNX
|
7.7 | pIC50 | 4 | Yes | |
JBHXXYIRQFVFOU
|
7.7 | pIC50 | 3 | Yes | |
ORZSTHMXZBZWIN
|
7.7 | pIC50 | 3 | Yes | |
SJEPMZVFPSMGMK
|
7.7 | IC50 | 2 | — | |
VAFGRMAYAKICTQ
|
7.7 | IC50 | 3 | — | |
WVRPZYQKQWOMIH
|
7.7 | Ki | 8 | — | |
ZOLPUEOXQAILTM
|
7.7 | Ki | 9 | — | |
ZTKKJFAJTKWNOE
|
7.7 | IC50 | 2 | Yes | |
AWSQADBSXFTFKL
|
7.7 | IC50 | 5 | — | |
BHNRAKLQOOFPBU
|
7.7 | pIC50 | 4 | Yes | |
FDEXXQUKUXAVRQ
|
7.7 | IC50 | 2 | Yes | |
FKAJEPVSQITQLJ
|
7.7 | IC50 | 15 | — |