Target Details
| UniProt AC | P06493 |
|---|---|
| Gene Symbol | CDK1 |
| Protein Name | Cyclin-dependent kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,900
- Clinical molecules 608
- Avg pChEMBL 7.06
KEGG Pathways (8)
Active Molecules (1,900)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LSGWJMLNFPIPPC
|
8.0 | IC50 | 4 | Yes | |
PHZDWQYTFQOSSZ
|
8.0 | IC50 | 15 | — | |
RPSMUTSVMKSFIZ
|
8.0 | pIC50 | 4 | Yes | |
ZGJLAVYYTJNBMN
|
8.0 | pIC50 | 4 | Yes | |
BAOWDLOLYGOWOE
|
8.0 | IC50 | 4 | — | |
ATRHQBQEZHPYKB
|
7.9 | IC50 | 2 | — | |
BPSQKVIOXGCIIK
|
7.9 | IC50 | 2 | — | |
FYYYMEMZRSXLIX
|
7.9 | IC50 | 4 | — | |
GEQMDKKVXALFFX
|
7.9 | Ki | 9 | — | |
GJHVXBPCYTULDM
|
7.9 | pIC50 | 4 | Yes | |
JYIASQGROAISCJ
|
7.9 | IC50 | 4 | — | |
KDLIWXJGIZBHKK
|
7.9 | IC50 | 3 | — | |
KGEGZSPPABUDIC
|
7.9 | pIC50 | 4 | Yes | |
QAQKNZRNOQBKRE
|
7.9 | IC50 | 2 | — | |
SGOFFNQMBSXTRU
|
7.9 | Ki | 9 | — | |
SOTHNRIRXPUQEZ
|
7.9 | pIC50 | 5 | Yes | |
YDTIWHFPTISVND
|
7.9 | IC50 | 4 | — | |
YZVFJIYEYQIHIP
|
7.9 | IC50 | 15 | — | |
FETXAWXOSWHGHF
|
7.9 | pIC50 | 9 | Yes | |
SSIDJRGNBKXDGV
|
7.9 | IC50 | 8 | — | |
GAASHZGNZTYOCB
|
7.9 | IC50 | 6 | — | |
QVUJFGWIMPTAEH
|
7.9 | pIC50 | 2 | Yes | |
WSNJGDJRGNRVDV
|
7.9 | pIC50 | 3 | Yes | |
AHIMCOQTGQUIII
|
7.9 | IC50 | 3 | — | |
GDXJAAIAGCCGJP
|
7.9 | IC50 | 4 | — | |
KHLSGMMGWBAAOY
|
7.9 | IC50 | 11 | Yes | |
LPPPFWQCXCFAAN
|
7.9 | IC50 | 3 | — | |
MDIDMHALYFMVFV
|
7.9 | pIC50 | 5 | Yes | |
NTRCIHPFGKPYRR
|
7.9 | IC50 | 2 | — | |
SLTWTVOINKYHIE
|
7.9 | pIC50 | 3 | Yes | |
XEXXLSSPQTWUID
|
7.9 | IC50 | 3 | — | |
XSTAWOGBOKIKIE
|
7.9 | pIC50 | 2 | Yes | |
AHZUHDSHQGQZRW
|
7.8 | IC50 | 4 | Yes | |
DOXLZSAKRJWFJV
|
7.8 | pIC50 | 2 | Yes | |
GEICEYBJACBCSI
|
7.8 | IC50 | 3 | — | |
GFXMFSCCEVADLF
|
7.8 | pIC50 | 11 | Yes | |
JMHQUQCLIVNTHT
|
7.8 | IC50 | 24 | — | |
RWSCYFXGWJPUQX
|
7.8 | IC50 | 15 | — | |
RYQTYXLOEDUZBQ
|
7.8 | IC50 | 3 | — | |
BDMNMAWBZWPSJC
|
7.8 | pIC50 | 9 | Yes | |
MVLOBPPFCUCBHT
|
7.8 | IC50 | 9 | — | |
BUGPWXMPCMTLIX
|
7.8 | pIC50 | 7 | Yes | |
NWIPTENCWQPQTO
|
7.8 | pIC50 | 4 | Yes | |
HSEUQWUJSFQRHV
|
7.8 | pIC50 | 2 | Yes | |
IFRYUGXGLYZVSY
|
7.8 | IC50 | 3 | — | |
JWOJZWRKDLDOEO
|
7.8 | IC50 | 3 | — | |
LHOZDNGAEMLEKU
|
7.8 | pIC50 | 2 | Yes | |
OLUKILHGKRVDCT
|
7.8 | pIC50 | 44 | Yes | |
QWDLZMUWYCLKFF
|
7.8 | IC50 | 10 | — | |
UXGASSHBBXBLJM
|
7.8 | IC50 | 2 | — |