Target Details
| UniProt AC | P06493 |
|---|---|
| Gene Symbol | CDK1 |
| Protein Name | Cyclin-dependent kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,900
- Clinical molecules 608
- Avg pChEMBL 7.06
KEGG Pathways (8)
Active Molecules (1,900)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NDQPEKJCVSIVHE
|
8.1 | IC50 | 4 | — | |
ABEGFBRZNZWQBS
|
8.1 | pIC50 | 5 | Yes | |
ASEKFENKLHTYMI
|
8.1 | pIC50 | 3 | Yes | |
IEWLQUDDCQIINQ
|
8.1 | IC50 | 3 | — | |
VMXUAXSUFHWVMR
|
8.1 | IC50 | 3 | Yes | |
DJXMWMFZMCZDNH
|
8.1 | IC50 | 6 | — | |
UQABTPYYEALKPO
|
8.1 | pIC50 | 2 | Yes | |
HYBCPKCAHCAFSQ
|
8.1 | pIC50 | 3 | Yes | |
NSKFUKOVLGRMFV
|
8.1 | IC50 | 6 | — | |
RVKNONNXSNALJV
|
8.1 | IC50 | 21 | — | |
UTGUSPCINACJKQ
|
8.1 | pIC50 | 3 | Yes | |
AEMJGAHADFWBRW
|
8.1 | pIC50 | 2 | Yes | |
AJJOCYLKITUOSA
|
8.1 | pIC50 | 2 | Yes | |
DJXMWMFZMCZDNH
|
8.1 | IC50 | 6 | — | |
FTQYGMLRLRXBPT
|
8.1 | pIC50 | 2 | Yes | |
GKJRCQIJVHMRJB
|
8.1 | IC50 | 3 | — | |
GOWOIXBMOFKIQJ
|
8.1 | IC50 | 4 | Yes | |
JLMIHNJHBAEFKC
|
8.1 | IC50 | 6 | — | |
LLLCCJOBPGNPTB
|
8.1 | IC50 | 4 | — | |
TWRINNPUKAHNGL
|
8.1 | pIC50 | 2 | Yes | |
UPQKBKLECVIXJR
|
8.1 | IC50 | 12 | — | |
VXBAJLGYBMTJCY
|
8.1 | IC50 | 34 | Yes | |
PVLOKYREDKFWTF
|
8.0 | pIC50 | 2 | Yes | |
VPHNNRKBCWFFKK
|
8.0 | pIC50 | 4 | Yes | |
FDWQSLRDIBRKEI
|
8.0 | pIC50 | 9 | Yes | |
GCYXEGSPUDSZJY
|
8.0 | pIC50 | 17 | Yes | |
CGBFAYLLULJFBW
|
8.0 | Ki | 8 | — | |
CKQXWWXJHFTWJZ
|
8.0 | IC50 | 6 | — | |
CXGFHBJFQBWPBO
|
8.0 | pIC50 | 4 | Yes | |
KZDYTAXBOFTVGN
|
8.0 | IC50 | 3 | — | |
NDEXUOWTGYUVGA
|
8.0 | Ki | 12 | — | |
OMCNPZUKTXGTFK
|
8.0 | pIC50 | 2 | Yes | |
QXAJGNKSKVWFIR
|
8.0 | IC50 | 4 | Yes | |
SBFPHSVZEXSHTL
|
8.0 | Ki | 62 | — | |
SEPHEVMRHYRRLS
|
8.0 | IC50 | 2 | — | |
SOXXWGSPFAGLBY
|
8.0 | pIC50 | 3 | Yes | |
SYCRYYILCMOTOI
|
8.0 | IC50 | 3 | — | |
SZYCBCZXRQISJY
|
8.0 | pIC50 | 3 | Yes | |
XJQPUMGIUIXVMH
|
8.0 | IC50 | 3 | — | |
XOXWOPNBJDVSJP
|
8.0 | Ki | 8 | — | |
ZWRDUCSPTGMSHB
|
8.0 | IC50 | 3 | — | |
NBWQLTANUJBFJB
|
8.0 | pIC50 | 2 | Yes | |
QPKLKELWAIIBCT
|
8.0 | pIC50 | 2 | Yes | |
AEZMHSFAAKOLNC
|
8.0 | pIC50 | 2 | Yes | |
BTIHMVBBUGXLCJ
|
8.0 | pIC50 | 21 | Yes | |
CXDXSBLYPKFPLO
|
8.0 | IC50 | 3 | — | |
DJXFMECMJJONCX
|
8.0 | pIC50 | 3 | Yes | |
JJQNDXCUJRPPDT
|
8.0 | IC50 | 2 | — | |
KAAFPSZABFPQAX
|
8.0 | IC50 | 2 | — | |
LOQNAQWIGMNXII
|
8.0 | pIC50 | 9 | Yes |