Target Details
| UniProt AC | P06493 |
|---|---|
| Gene Symbol | CDK1 |
| Protein Name | Cyclin-dependent kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,900
- Clinical molecules 608
- Avg pChEMBL 7.06
KEGG Pathways (8)
Active Molecules (1,900)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GKJRCQIJVHMRJB
|
8.2 | IC50 | 3 | — | |
IHOIRURKGWDCHK
|
8.2 | pIC50 | 2 | Yes | |
KLYOKJDELSPRDU
|
8.2 | pIC50 | 2 | Yes | |
QKVCYCAAFKGTNA
|
8.2 | IC50 | 3 | Yes | |
DZKMAWNYSJECKX
|
8.2 | IC50 | 12 | — | |
GXDMNAKMJVMWKQ
|
8.2 | pIC50 | 5 | Yes | |
JGBCHSGVRWYCES
|
8.2 | pIC50 | 2 | Yes | |
AANVTLVNTUEXNM
|
8.2 | pIC50 | 3 | Yes | |
BACSZMCLZIDTIO
|
8.2 | pIC50 | 2 | Yes | |
BUVUGYVWVBFUMI
|
8.2 | Ki | 11 | — | |
DIASEXMEBNQQHZ
|
8.2 | IC50 | 13 | — | |
FZLZLIAOYSKHJC
|
8.2 | Ki | 11 | — | |
HVMRLFSFHWCUCG
|
8.2 | IC50 | 3 | Yes | |
KDKUVYLMPJIGKA
|
8.2 | pIC50 | 91 | Yes | |
KOLSEKSFVMGHDV
|
8.2 | IC50 | 12 | — | |
KRKQVGZXTNLQSV
|
8.2 | IC50 | 9 | Yes | |
OOKAYBMMWNSBPA
|
8.2 | Ki | 9 | — | |
OTPFZAVDWPCJLJ
|
8.2 | Ki | 9 | — | |
QJOLFMLQXIPTTF
|
8.2 | IC50 | 3 | — | |
QZTBLEFQOCINTB
|
8.2 | pIC50 | 3 | Yes | |
SCFMWQIQBVZOQR
|
8.2 | IC50 | 14 | Yes | |
ZKDXRFMOHZVXSG
|
8.2 | pIC50 | 13 | Yes | |
ADMFLILDQJSEIK
|
8.2 | Ki | 72 | — | |
MDJCUXFFMNEBHG
|
8.2 | Ki | 13 | — | |
AAVOJGZMGDAVNM
|
8.2 | IC50 | 6 | — | |
SFGWUTHNZVSATD
|
8.2 | pIC50 | 11 | Yes | |
AIEHUMVISDRBPD
|
8.2 | pIC50 | 2 | Yes | |
BQLLLVDIZXOQJD
|
8.2 | Ki | 8 | — | |
CBARNMHMGRVVLO
|
8.2 | IC50 | 11 | — | |
GFMLSFXYFKGRNS
|
8.2 | pIC50 | 2 | Yes | |
GTVPOLSIJWJJNY
|
8.2 | pIC50 | 2 | Yes | |
IFRYUGXGLYZVSY
|
8.2 | IC50 | 3 | — | |
KGHAUONMJSXUDW
|
8.2 | pIC50 | 2 | Yes | |
KJHOORCYJSBANN
|
8.2 | IC50 | 15 | — | |
LNYKHAPIJVILRZ
|
8.2 | pIC50 | 7 | Yes | |
OPLHNOVRWYFVGR
|
8.2 | IC50 | 2 | — | |
PARUULGUCQEWNM
|
8.2 | pIC50 | 3 | Yes | |
PRXRQGZKWMOFLL
|
8.2 | IC50 | 11 | Yes | |
UELYDGOOJPRWGF
|
8.2 | IC50 | 4 | — | |
UELYDGOOJPRWGF
|
8.2 | IC50 | 5 | — | |
UELYDGOOJPRWGF
|
8.2 | IC50 | 13 | — | |
UELYDGOOJPRWGF
|
8.2 | IC50 | 9 | — | |
WFNUAOKMXUQUHV
|
8.2 | IC50 | 3 | — | |
ZKEDVROWQXMVGQ
|
8.2 | IC50 | 3 | — | |
DVMBLTDKHALLLH
|
8.1 | pIC50 | 6 | Yes | |
OWXORKPNCHJYOF
|
8.1 | pIC50 | 17 | Yes | |
CICSYFWWWTXRPT
|
8.1 | IC50 | 3 | — | |
GQTPCOMZBGFWLQ
|
8.1 | pIC50 | 11 | Yes | |
JXJHPQHLHQTQQI
|
8.1 | IC50 | 15 | — | |
NWJBWUFQUJNFKY
|
8.1 | pIC50 | 2 | Yes |