Target Details
| UniProt AC | P06493 |
|---|---|
| Gene Symbol | CDK1 |
| Protein Name | Cyclin-dependent kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,900
- Clinical molecules 608
- Avg pChEMBL 7.06
KEGG Pathways (8)
Active Molecules (1,900)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKSZLNNOFSGOKW
|
8.4 | Ki | 118 | — | |
KEBMLXBFCRPVRB
|
8.4 | IC50 | 4 | — | |
PMXCMJLOPOFPBT
|
8.4 | pIC50 | 17 | Yes | |
RVSKJUNTDGBSSS
|
8.4 | Ki | 25 | — | |
SPRSVKHLNRKLHA
|
8.4 | IC50 | 5 | — | |
SRJYCUWWNQFSQR
|
8.4 | pIC50 | 3 | Yes | |
VEMUNZLIOXAWMA
|
8.4 | IC50 | 3 | — | |
XIRBBABZYUQIMH
|
8.4 | pIC50 | 2 | Yes | |
WQZVTNFUNLTGDW
|
8.4 | Ki | 4 | — | |
MNROLFUOLVMVKW
|
8.4 | pIC50 | 2 | Yes | |
DXKGSLMPGXZMRN
|
8.3 | IC50 | 4 | — | |
ISZYBQYCHOZPBF
|
8.3 | pIC50 | 11 | Yes | |
OEHDHLJQYLJHHS
|
8.3 | pIC50 | 2 | Yes | |
VAOAJUWPEYBTAB
|
8.3 | pIC50 | 9 | Yes | |
IDNJKMAZNUUVIO
|
8.3 | IC50 | 9 | — | |
IGWUXPFABXHPLJ
|
8.3 | pIC50 | 2 | Yes | |
LFWPDIWWAQIGSW
|
8.3 | pIC50 | 2 | Yes | |
KQWTXAWKBUUOMU
|
8.3 | pIC50 | 20 | Yes | |
JDXDUTOQTGQWJD
|
8.3 | pIC50 | 3 | Yes | |
LMIPCDJYZXYYLQ
|
8.3 | IC50 | 5 | — | |
NBSJZWFDNFWQDN
|
8.3 | IC50 | 29 | — | |
NFTJDXGFOUFNKG
|
8.3 | IC50 | 16 | — | |
AXAQVNRYNMCZCK
|
8.3 | Ki | 10 | Yes | |
BCBUOCNTMGMTQK
|
8.3 | pIC50 | 3 | Yes | |
BKCOGSHTNWTZNI
|
8.3 | IC50 | 15 | — | |
CQVJGFKTRSGJHB
|
8.3 | Ki | 11 | — | |
CQWBHMMWZICZRH
|
8.3 | IC50 | 10 | — | |
JQLOWVFMFQYNIP
|
8.3 | IC50 | 3 | — | |
JYXVTNQLJPOFBP
|
8.3 | pIC50 | 3 | Yes | |
KAAFPSZABFPQAX
|
8.3 | IC50 | 3 | — | |
KJSJBGZSEZVHMS
|
8.3 | IC50 | 2 | — | |
OZOLFJMARMOUPD
|
8.3 | pIC50 | 3 | Yes | |
QFUXJZMXUXQIIB
|
8.3 | IC50 | 2 | — | |
RIEBONGMTZXFMR
|
8.3 | pIC50 | 3 | Yes | |
SPTNJNJCNRTHDY
|
8.3 | pIC50 | 3 | Yes | |
TVARIYLSKVWCHN
|
8.3 | Ki | 11 | — | |
UDFDIIVNIYWXDM
|
8.3 | Ki | 74 | — | |
VUIXUTVIIOVVHV
|
8.3 | IC50 | 3 | — | |
WCCYEJYTLNWYCC
|
8.3 | IC50 | 9 | — | |
WWUPNOVYRXPGJZ
|
8.3 | IC50 | 5 | — | |
WXFGSMZOKBRNIJ
|
8.3 | IC50 | 3 | — | |
WXPDCELKHNMODS
|
8.3 | pIC50 | 3 | Yes | |
XJQPUMGIUIXVMH
|
8.3 | IC50 | 3 | — | |
ZLCBGFVBDKXPBZ
|
8.3 | IC50 | 2 | — | |
ZSNHIQTXGFQNBW
|
8.3 | IC50 | 3 | — | |
ZUCAWWSJZRVUAX
|
8.3 | Ki | 11 | — | |
AEFFENQISAXIKE
|
8.3 | IC50 | 9 | — | |
KCVMRCBFSCVBTH
|
8.3 | pIC50 | 3 | Yes | |
MPJITOINOMJIJI
|
8.3 | pIC50 | 11 | Yes | |
ATIIMPVWPLDRSW
|
8.2 | pIC50 | 2 | Yes |