Target Details
| UniProt AC | P06493 |
|---|---|
| Gene Symbol | CDK1 |
| Protein Name | Cyclin-dependent kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,900
- Clinical molecules 608
- Avg pChEMBL 7.06
KEGG Pathways (8)
Active Molecules (1,900)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FUPOZFLWFNCROX
|
8.7 | pIC50 | 2 | Yes | |
QPQPCKPZCWKFDE
|
8.7 | IC50 | 4 | — | |
DQBASRYERZQRJJ
|
8.7 | IC50 | 15 | — | |
VCPXSBULBDYRLT
|
8.7 | pIC50 | 4 | Yes | |
MEKASOQEXYKAKM
|
8.6 | IC50 | 4 | — | |
GNODSQUZRSUVER
|
8.6 | IC50 | 3 | — | |
HKSZLNNOFSGOKW
|
8.6 | IC50 | 408 | — | |
WLIGHAXZSXWZCO
|
8.6 | IC50 | 3 | — | |
ZFHAOTRAAVCTPZ
|
8.6 | pIC50 | 2 | Yes | |
OLFNLUGZKOQDEV
|
8.6 | IC50 | 9 | — | |
GXAMBYHREJMOKQ
|
8.6 | pIC50 | 11 | Yes | |
UPLMSKBPWUAWBT
|
8.6 | IC50 | 4 | — | |
DUEBWXVTFJJWCJ
|
8.6 | pIC50 | 11 | Yes | |
FOLRMJVSUYSNKR
|
8.6 | IC50 | 5 | — | |
LTYGAJVXAFJKSY
|
8.6 | pIC50 | 2 | Yes | |
LTYGAJVXAFJKSY
|
8.6 | pIC50 | 3 | Yes | |
BDRDBXXWQDFXEC
|
8.5 | pIC50 | 5 | Yes | |
BEXPELAOVIOQHQ
|
8.5 | pIC50 | 3 | Yes | |
BHQZGGSZRHDQFZ
|
8.5 | pIC50 | 13 | Yes | |
BRBJCJHJBAMBPR
|
8.5 | IC50 | 12 | — | |
BYUAPXZEZUYLJI
|
8.5 | IC50 | 4 | — | |
CNSXYUZUUPJMQL
|
8.5 | pIC50 | 2 | Yes | |
DMCVVJAYVRAPRW
|
8.5 | Ki | 5 | — | |
FGLDVWQEBUVALV
|
8.5 | IC50 | 3 | — | |
FOTACNUKABBYFV
|
8.5 | pIC50 | 3 | Yes | |
KAAFPSZABFPQAX
|
8.5 | IC50 | 5 | — | |
KCKWQKDFLCMFNR
|
8.5 | IC50 | 4 | — | |
KJSJBGZSEZVHMS
|
8.5 | IC50 | 2 | — | |
OKVAXHZNBTZJCB
|
8.5 | IC50 | 3 | — | |
PIMQWRZWLQKKBJ
|
8.5 | IC50 | 4 | — | |
PIMQWRZWLQKKBJ
|
8.5 | IC50 | 36 | — | |
QURBHJPQZDAPGP
|
8.5 | IC50 | 3 | — | |
SZKRTTIHILIRKD
|
8.5 | pIC50 | 3 | Yes | |
VBYCLUNCQJLFHE
|
8.5 | IC50 | 4 | Yes | |
XDAVVOMFBOEFCG
|
8.5 | IC50 | 4 | — | |
XERLASHNAPKEEL
|
8.5 | pIC50 | 7 | Yes | |
YGZQAQIWZFMADC
|
8.5 | IC50 | 12 | — | |
AAOLDQJTTACKSD
|
8.5 | pIC50 | 4 | Yes | |
FVCARQMVVSNDMM
|
8.5 | IC50 | 4 | — | |
QDICJHBKGMJCQZ
|
8.5 | IC50 | 4 | — | |
REWUWHLCHRZZTC
|
8.5 | IC50 | 4 | — | |
ZJDFSKSBQBPOSK
|
8.5 | IC50 | 24 | Yes | |
TXWFROAATAZXFK
|
8.5 | pIC50 | 2 | Yes | |
AFMQUOLJZIETKV
|
8.4 | pIC50 | 2 | Yes | |
IAPISFUJUUDVNW
|
8.4 | IC50 | 15 | — | |
JBOXDNIWQACYPW
|
8.4 | IC50 | 4 | — | |
AXAGUGNJIAGPOV
|
8.4 | pIC50 | 4 | Yes | |
CDKRFBBXZQUTDX
|
8.4 | Ki | 9 | — | |
GAIOPWBQKZMUNO
|
8.4 | Ki | 13 | — | |
GJVPWZGJUOVEBA
|
8.4 | IC50 | 3 | — |