Target Details
| UniProt AC | P06493 |
|---|---|
| Gene Symbol | CDK1 |
| Protein Name | Cyclin-dependent kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,900
- Clinical molecules 608
- Avg pChEMBL 7.06
KEGG Pathways (8)
Active Molecules (1,900)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UBLFSMURWWWWMH
|
9.6 | IC50 | 7 | — | |
GULUZCYKKDJDGN
|
9.6 | IC50 | 3 | — | |
QFLOEOVVFKHAFI
|
9.5 | pIC50 | 2 | Yes | |
CDZRXVMQLQSKPO
|
9.5 | Ki | 3 | — | |
HKSZLNNOFSGOKW
|
9.4 | pIC50 | 49 | Yes | |
QNUFZYZRLJGZJL
|
9.4 | IC50 | 10 | — | |
FPHITTVVVWKENE
|
9.3 | Ki | 9 | — | |
YYFFSHNCRZXJNQ
|
9.3 | pIC50 | 2 | Yes | |
ARIOBGGRZJITQX
|
9.2 | IC50 | 24 | — | |
SCMJNQHUUQLKRS
|
9.2 | IC50 | 5 | — | |
UCSGBFLLOMEVMS
|
9.2 | IC50 | 4 | — | |
KRKHEOQTCZTRNA
|
9.2 | IC50 | 2 | — | |
URLYPAWCHVXIAA
|
9.2 | IC50 | 4 | Yes | |
BKMFUDJYEMHEKH
|
9.1 | IC50 | 2 | — | |
WNOFAMMMUOEJEM
|
9.1 | pIC50 | 3 | Yes | |
UEYQVGAFBVFHAU
|
9.0 | IC50 | 3 | Yes | |
AMOZPNFTPZCWKP
|
9.0 | pIC50 | 2 | Yes | |
BWONSNVPSAEXDY
|
9.0 | Ki | 9 | — | |
FGQLPUTYZYTKLO
|
9.0 | IC50 | 2 | — | |
PAXKGQZKOJPPEG
|
9.0 | IC50 | 5 | Yes | |
RWVYOYMRKMXRCK
|
9.0 | pIC50 | 2 | Yes | |
SEKBBOWCTFTKRL
|
9.0 | pIC50 | 2 | Yes | |
VWQIQPRBMMSYCE
|
9.0 | IC50 | 6 | — | |
XJKMKRYBCWBZML
|
9.0 | IC50 | 4 | — | |
DPAOHEUWPLGQDY
|
9.0 | IC50 | 4 | Yes | |
IRBHAVXRXYJMRS
|
9.0 | pIC50 | 2 | Yes | |
GNKARCUXNWYAPQ
|
8.9 | IC50 | 5 | — | |
DMXIHKQKBYZIHM
|
8.8 | IC50 | 5 | Yes | |
BXMBIVXDTXURDF
|
8.8 | Ki | 9 | — | |
XVXBWZZWJTYKPA
|
8.8 | pIC50 | 2 | Yes | |
WISHLJZJMNBRMX
|
8.8 | IC50 | 9 | — | |
HAIHTRCFSLFERU
|
8.7 | pIC50 | 3 | Yes | |
UQHPGIWKYQJUIE
|
8.7 | IC50 | 7 | — | |
NQCDYPGJGMFSFB
|
8.7 | IC50 | 4 | — | |
VNLUDQKOXAUGAO
|
8.7 | pIC50 | 2 | Yes | |
ADMFLILDQJSEIK
|
8.7 | IC50 | 4 | — | |
BACSZMCLZIDTIO
|
8.7 | pIC50 | 2 | Yes | |
BXQSENVZNNEEBV
|
8.7 | pIC50 | 5 | Yes | |
GAFYDJGFHJBXQQ
|
8.7 | Ki | 9 | — | |
GNODSQUZRSUVER
|
8.7 | IC50 | 3 | — | |
JRNJNYBQQYBCLE
|
8.7 | Ki | 40 | Yes | |
NTSDIJMNXYJJNG
|
8.7 | pIC50 | 2 | Yes | |
QTAXCQYCXMOZAD
|
8.7 | pIC50 | 2 | Yes | |
UHCNAXAEICMASJ
|
8.7 | IC50 | 5 | — | |
VXBMLLKHEDZLSY
|
8.7 | pIC50 | 4 | Yes | |
WLPVKLZUKCPKQL
|
8.7 | pIC50 | 2 | Yes | |
XCJRUIHXLFTUNW
|
8.7 | IC50 | 3 | — | |
XLSYZSRXVVCHLS
|
8.7 | IC50 | 48 | — | |
YLRRTJLWOJHWFB
|
8.7 | pIC50 | 2 | Yes | |
ZJJZCHNTRMUXMT
|
8.7 | pIC50 | 2 | Yes |