Target Details
| UniProt AC | P06401 |
|---|---|
| Gene Symbol | PGR |
| Protein Name | Progesterone receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00104 (Hormone_recep) PF02161 (Prog_receptor) PF00105 (zf-C4) |
Summary
- Multi-target molecules 617
- Clinical molecules 33
- Avg pChEMBL 7.21
KEGG Pathways (5)
Associated Diseases (1)
Active Molecules (617)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PLYZMJXXOPVZLJ
|
6.6 | IC50 | 2 | — | |
XCCRMYVOJIFMED
|
6.6 | Ki | 3 | — | |
XCZSJKKONDGKDF
|
6.6 | IC50 | 2 | — | |
AKMUGEXFTSZYPE
|
6.6 | Ki | 2 | — | |
HQVKFEYATUGVGI
|
6.6 | IC50 | 2 | — | |
JKPOACVGQYPLBU
|
6.6 | IC50 | 3 | — | |
JTNNQTQMGYMRGO
|
6.6 | IC50 | 3 | — | |
ZREYWBOITVVPOZ
|
6.6 | IC50 | 3 | — | |
HBWBMLKOCYUNSK
|
6.6 | Kd | 3 | — | |
KPKCYUMBFMYREG
|
6.6 | Ki | 3 | — | |
MIAURGNSNSBTNK
|
6.6 | Ki | 4 | — | |
UBRFDZVHGGUVEL
|
6.6 | IC50 | 2 | — | |
UUIWYLMDKKQBJQ
|
6.6 | IC50 | 3 | — | |
KNEYKCUMUCBZNB
|
6.6 | IC50 | 3 | — | |
GQEDWCRZISUBTM
|
6.6 | Ki | 2 | — | |
HINCRROTVFUICG
|
6.6 | IC50 | 3 | — | |
NRQQDFFSJPVQFQ
|
6.6 | IC50 | 2 | — | |
QGCIAWJCSRYRFH
|
6.6 | Ki | 2 | — | |
BEOADSCNJSAOSW
|
6.6 | Ki | 2 | — | |
KXRGUCHKDGYOHL
|
6.6 | IC50 | 2 | — | |
OFPJLMJVJSEKIP
|
6.6 | IC50 | 3 | — | |
QAJXXFBIGIATMT
|
6.6 | IC50 | 2 | — | |
ARAFJNZXJVLHDR
|
6.5 | IC50 | 3 | — | |
QHIXHFRNTAVAPK
|
6.5 | IC50 | 2 | — | |
QKTUOSGGPMYODZ
|
6.5 | Ki | 2 | — | |
XFVHCXVBLVMUSO
|
6.5 | IC50 | 2 | — | |
CFDUSNZVLMAHPE
|
6.5 | IC50 | 3 | — | |
QWKSNMYGEFJJIU
|
6.5 | Ki | 2 | — | |
BUUOLGKPFRELSS
|
6.5 | IC50 | 3 | — | |
QMISUBCKEDZHDT
|
6.5 | IC50 | 3 | — | |
BBQPRPRCQIFLIO
|
6.5 | IC50 | 2 | — | |
OWJRNHUDJKJKDG
|
6.5 | IC50 | 2 | — | |
PDXCFTVMFXAKMC
|
6.5 | IC50 | 2 | — | |
RVDUZNHKCJRYQY
|
6.5 | Ki | 2 | — | |
HQFHTXSVKRXPKT
|
6.5 | Ki | 2 | — | |
MIAURGNSNSBTNK
|
6.5 | Ki | 4 | — | |
RRWMFEXUNNLRMV
|
6.5 | IC50 | 2 | — | |
UGJGTPGLSLQCPP
|
6.5 | IC50 | 3 | — | |
VWFKACUYWYZVSW
|
6.5 | IC50 | 3 | — | |
JJBGOTRJBHAAQW
|
6.5 | IC50 | 2 | — | |
LCTXHPZYTFNYEN
|
6.5 | IC50 | 2 | — | |
WISJIBWIQKICSR
|
6.5 | Ki | 2 | — | |
XVYWAUINFAXEKA
|
6.5 | IC50 | 3 | — | |
YUMWHZCQHQAPAQ
|
6.5 | IC50 | 3 | — | |
CAEHKTJNVMDKLN
|
6.5 | IC50 | 2 | — | |
GAKWAQHHESGFAA
|
6.5 | IC50 | 3 | — | |
LPNILISJTWTRLC
|
6.5 | IC50 | 3 | — | |
SMYUZCJLGBMSME
|
6.5 | IC50 | 3 | — | |
UHRXKJFPPKYYEC
|
6.5 | Ki | 2 | — | |
VKNDUDKNPQIQIQ
|
6.5 | Ki | 3 | — |