Target Details
| UniProt AC | P06401 |
|---|---|
| Gene Symbol | PGR |
| Protein Name | Progesterone receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00104 (Hormone_recep) PF02161 (Prog_receptor) PF00105 (zf-C4) |
Summary
- Multi-target molecules 617
- Clinical molecules 33
- Avg pChEMBL 7.21
KEGG Pathways (5)
Associated Diseases (1)
Active Molecules (617)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QYEYUIJWYCBKBG
|
6.8 | Ki | 2 | — | |
FOSHWESRGNRMBT
|
6.8 | Ki | 2 | — | |
PYHAWYQXRVXAHX
|
6.8 | Ki | 4 | — | |
USLSTEHVCOVPEK
|
6.8 | IC50 | 3 | — | |
YXFRGFFRCABTFT
|
6.8 | IC50 | 2 | — | |
DORQSUNHACTGLQ
|
6.8 | IC50 | 3 | — | |
FMZKGKLLLCYGJW
|
6.8 | Ki | 3 | — | |
RRWMFEXUNNLRMV
|
6.8 | IC50 | 2 | — | |
UWRFZHBVLLTGSN
|
6.8 | IC50 | 2 | — | |
VGCGSAUUQCQDAY
|
6.8 | IC50 | 3 | — | |
AECUUHUGTSTYSJ
|
6.8 | IC50 | 2 | — | |
HQGRCFOENHIIQG
|
6.8 | IC50 | 2 | — | |
KSBBSPJEGUHNTP
|
6.8 | IC50 | 3 | — | |
WFQCSOVOMJIJSZ
|
6.8 | IC50 | 2 | — | |
XAEBVWFWHJQFCD
|
6.8 | IC50 | 2 | — | |
BLPNJKOYOIDEJJ
|
6.8 | IC50 | 2 | — | |
XCVIXZRNZRDCKE
|
6.8 | Kd | 4 | — | |
BVSCKUSMKCQTFI
|
6.7 | IC50 | 2 | — | |
QUJQBNBSMHJFAG
|
6.7 | IC50 | 2 | — | |
SEVGDNHYESBDRZ
|
6.7 | IC50 | 2 | — | |
CRODFMXMGHZTCT
|
6.7 | Ki | 2 | — | |
HYZGNFIJTUJTBY
|
6.7 | Ki | 2 | — | |
ULOAOMMDFZMTER
|
6.7 | IC50 | 3 | — | |
UZNBZDTUBTWOBU
|
6.7 | Ki | 4 | — | |
DQMJJYWWVJPLDX
|
6.7 | Ki | 2 | — | |
FVNZFSAGJPHSHT
|
6.7 | IC50 | 2 | — | |
HXJXFIBSBUSEJX
|
6.7 | IC50 | 2 | — | |
MQIWXSYBYIIVPE
|
6.7 | IC50 | 3 | — | |
QFWHAFOCMOQSHC
|
6.7 | IC50 | 3 | — | |
RNQOQGINTAOCKX
|
6.7 | IC50 | 3 | — | |
RWLAOUIUIWXAOY
|
6.7 | Ki | 2 | — | |
WDXRGPWQVHZTQJ
|
6.7 | Ki | 5 | — | |
ZANAAVXGSNLYBQ
|
6.7 | IC50 | 2 | — | |
HINCRROTVFUICG
|
6.7 | IC50 | 3 | — | |
MGDHDHQGYPSORD
|
6.7 | IC50 | 3 | — | |
OKMFMKSZIXQMRJ
|
6.7 | IC50 | 2 | — | |
SFFRJYDGTHMNDH
|
6.7 | IC50 | 3 | — | |
ZEOIRIKFAKERSP
|
6.7 | IC50 | 2 | — | |
FEKIYUBTGQLEBI
|
6.7 | Ki | 3 | — | |
GDJKXOLGMVNOGF
|
6.7 | Ki | 3 | — | |
NHOGRLKDZYGUSJ
|
6.7 | IC50 | 2 | — | |
NNTHLQVZGURUAX
|
6.7 | IC50 | 3 | — | |
WDXRGPWQVHZTQJ
|
6.7 | Ki | 5 | — | |
KAFURNBTIHQXCB
|
6.6 | Ki | 2 | — | |
PEEQAQFTZGENDO
|
6.6 | Ki | 2 | — | |
SWMIPBWORQVDRL
|
6.6 | IC50 | 2 | — | |
VQXYALIFGGOXRU
|
6.6 | Ki | 2 | — | |
CRLRDHCTZNQLSN
|
6.6 | Ki | 2 | — | |
DYJWFOYAGMZBFA
|
6.6 | IC50 | 2 | — | |
JRZWVYSKNVMDLP
|
6.6 | IC50 | 3 | — |