Target Details
| UniProt AC | P06401 |
|---|---|
| Gene Symbol | PGR |
| Protein Name | Progesterone receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00104 (Hormone_recep) PF02161 (Prog_receptor) PF00105 (zf-C4) |
Summary
- Multi-target molecules 617
- Clinical molecules 33
- Avg pChEMBL 7.21
KEGG Pathways (5)
Associated Diseases (1)
Active Molecules (617)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YFCOZFVKDGNSQY
|
7.1 | IC50 | 2 | — | |
UBDHJEXXHMTARH
|
7.1 | Kd | 4 | — | |
ZJHROHSTVJKUKT
|
7.1 | IC50 | 2 | — | |
HQCVWNZJFCYZOD
|
7.1 | Ki | 2 | — | |
DAYFWNQOWUPASA
|
7.1 | IC50 | 2 | — | |
DBWRTNRVJFYFDM
|
7.1 | IC50 | 2 | — | |
UTPNUAIWPWLJEC
|
7.1 | Ki | 4 | — | |
YGYIVBNMBYBQGZ
|
7.1 | IC50 | 3 | — | |
QLZJETYFHQVNRB
|
7.1 | IC50 | 2 | — | |
VQMSYLLYQOARPD
|
7.0 | IC50 | 3 | — | |
OYHQTRCZCQLKPX
|
7.0 | IC50 | 2 | — | |
BQZKKRYIQPCEKF
|
7.0 | Ki | 2 | — | |
MXEOXTXWJGNBGH
|
7.0 | IC50 | 2 | — | |
BJNAVMMYORPBLT
|
7.0 | IC50 | 2 | — | |
BQDLKNZJOSLJEM
|
7.0 | Ki | 2 | — | |
QWPDENUMNMUTHR
|
7.0 | IC50 | 2 | — | |
RUBRWONSGNOQIS
|
7.0 | IC50 | 2 | — | |
RVMQWZWBBBUEFH
|
7.0 | Ki | 2 | — | |
XDAWAGMTCJTDDV
|
7.0 | IC50 | 2 | — | |
YSJVBSSZEGNKMZ
|
7.0 | IC50 | 2 | — | |
HEVNCDKNAJNJPY
|
7.0 | Ki | 2 | — | |
MEWQFKSUHJZGCA
|
7.0 | Ki | 4 | — | |
FFJPGJNSRNWRSX
|
7.0 | IC50 | 2 | — | |
LCTFQUGGLDHXTH
|
7.0 | IC50 | 3 | — | |
QOSRQKJZZAEYCI
|
7.0 | IC50 | 2 | — | |
VKVZOFDGLCTSKW
|
7.0 | Ki | 2 | — | |
VTRALRXIBUAIMP
|
7.0 | IC50 | 2 | — | |
XFFATDFCPKLQRT
|
7.0 | Ki | 2 | — | |
MATZYFFMBFOOKH
|
7.0 | Ki | 2 | — | |
QGNJUOXZTPPCOF
|
7.0 | IC50 | 3 | — | |
UOYTXPZOHZGXMV
|
7.0 | IC50 | 2 | — | |
YOVQILQTFYDVHU
|
7.0 | IC50 | 2 | — | |
OJVZKFXAMCVCKM
|
6.9 | IC50 | 2 | — | |
RITZPFDVXSENFR
|
6.9 | IC50 | 2 | — | |
FZORYLRILGENBG
|
6.9 | Ki | 3 | — | |
JXCHEAFROKFUTG
|
6.9 | IC50 | 2 | — | |
HGHRCZOIYJBGPL
|
6.9 | IC50 | 2 | — | |
HGHRCZOIYJBGPL
|
6.9 | IC50 | 3 | — | |
NKANXQFJJICGDU
|
6.9 | IC50 | 35 | Yes | |
USLUSBGRSPWYFF
|
6.9 | IC50 | 3 | — | |
YROYMPDJQKBNTG
|
6.9 | IC50 | 3 | — | |
UUGJKSUOOIUEHL
|
6.9 | Ki | 2 | — | |
FYCXKGHEYHXTOX
|
6.9 | IC50 | 2 | — | |
DHMLTYBVPKCCCQ
|
6.9 | IC50 | 2 | — | |
AAJNWJFLYOFHIB
|
6.8 | IC50 | 3 | — | |
CFZKPYJJGYQRFD
|
6.8 | IC50 | 2 | — | |
CUNSDNZRZMUTPA
|
6.8 | Ki | 2 | — | |
SUBXROOMJNLXRP
|
6.8 | IC50 | 2 | — | |
FDXWONUERKJVPB
|
6.8 | Ki | 2 | — | |
USMFOMVHIKQVEN
|
6.8 | IC50 | 3 | — |