Target Details
| UniProt AC | P06401 |
|---|---|
| Gene Symbol | PGR |
| Protein Name | Progesterone receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00104 (Hormone_recep) PF02161 (Prog_receptor) PF00105 (zf-C4) |
Summary
- Multi-target molecules 617
- Clinical molecules 33
- Avg pChEMBL 7.21
KEGG Pathways (5)
Associated Diseases (1)
Active Molecules (617)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WSGANSMSRKUENH
|
7.3 | IC50 | 2 | — | |
LFLARVMSGCQYSZ
|
7.3 | IC50 | 2 | — | |
PZTMIXXVWUCYIR
|
7.3 | IC50 | 2 | — | |
DKFBPHVUBSXDJB
|
7.3 | IC50 | 3 | — | |
UKLYTFISJSJGSO
|
7.3 | IC50 | 2 | — | |
REOPBPDUXSVBMY
|
7.3 | IC50 | 2 | — | |
SGJHGBRSGXOPCU
|
7.3 | Ki | 2 | — | |
WLZJZUASQWXOGD
|
7.3 | IC50 | 2 | — | |
GAUXDXUKQPFNPK
|
7.3 | IC50 | 6 | Yes | |
OIANLDXMUCMGOG
|
7.3 | IC50 | 2 | — | |
XXYLLIHARBRABR
|
7.3 | Ki | 2 | — | |
KZGODNLSXIAMIQ
|
7.3 | IC50 | 2 | — | |
UFSVWJLQUADLKJ
|
7.3 | IC50 | 2 | — | |
LPVOSIGKKGTQCK
|
7.3 | Ki | 2 | — | |
MXEOXTXWJGNBGH
|
7.3 | IC50 | 2 | — | |
PCJNAMBTUJABGN
|
7.3 | Ki | 2 | — | |
QOSRQKJZZAEYCI
|
7.3 | IC50 | 2 | — | |
ZSMCHXGGQCKXMY
|
7.3 | Ki | 5 | Yes | |
HQCVWNZJFCYZOD
|
7.3 | Ki | 2 | — | |
HLRQXZBFIYYNOH
|
7.3 | Ki | 3 | — | |
NNEWMMFHUDIZPO
|
7.3 | IC50 | 3 | — | |
CCARZUVDBLMOLN
|
7.2 | Ki | 2 | — | |
GCKMJAVBEKTJOI
|
7.2 | IC50 | 2 | — | |
XFFATDFCPKLQRT
|
7.2 | Ki | 2 | — | |
CAVTYMQSFAIXRJ
|
7.2 | Ki | 4 | — | |
MUYIYYIMQMHGRZ
|
7.2 | Ki | 2 | — | |
CTRKFGYVXQHNDJ
|
7.2 | IC50 | 2 | — | |
ZUOVTFWGFULART
|
7.2 | IC50 | 2 | — | |
NZDONLCAMPFJHQ
|
7.2 | IC50 | 2 | — | |
QLCLQHCJXWSVTF
|
7.2 | IC50 | 3 | — | |
UXGUYYJUKZKENF
|
7.2 | Ki | 2 | — | |
XDFUKFMDLRMNOJ
|
7.2 | IC50 | 2 | — | |
MFAGIEMFDDDLMT
|
7.2 | Ki | 3 | — | |
PBRBWYQRHGSGKO
|
7.2 | IC50 | 2 | — | |
UHIOHBCVVQJMBM
|
7.2 | Ki | 2 | — | |
DFZYMRBKXQWSTE
|
7.2 | IC50 | 3 | — | |
PDCRQOSNBYFZJI
|
7.2 | Ki | 2 | — | |
SIMVLEKLLFIFBJ
|
7.2 | IC50 | 2 | — | |
IEVTWPPTWHIEGU
|
7.1 | Ki | 2 | — | |
KXMVPYRKURWIPA
|
7.1 | Ki | 4 | — | |
MPEPSOPXQDGEHP
|
7.1 | IC50 | 2 | — | |
YMBWIGXCZKHYQH
|
7.1 | Ki | 2 | — | |
FXOBRTHYLJLPSC
|
7.1 | IC50 | 3 | — | |
LFKDQCVODYHILG
|
7.1 | Ki | 2 | — | |
DPXITRVBJLQXDO
|
7.1 | IC50 | 2 | — | |
OKFXILKFTJTOKG
|
7.1 | Ki | 2 | — | |
QQFIDVOPZHXZPF
|
7.1 | IC50 | 3 | — | |
SKDVMPZQJMZEAC
|
7.1 | IC50 | 2 | — | |
TZSWJUXVIXDAFP
|
7.1 | IC50 | 2 | — | |
USUVLGWDWVYTDF
|
7.1 | IC50 | 2 | — |