Target Details
| UniProt AC | P06401 |
|---|---|
| Gene Symbol | PGR |
| Protein Name | Progesterone receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00104 (Hormone_recep) PF02161 (Prog_receptor) PF00105 (zf-C4) |
Summary
- Multi-target molecules 617
- Clinical molecules 33
- Avg pChEMBL 7.21
KEGG Pathways (5)
Associated Diseases (1)
Active Molecules (617)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
POQODJWQWWICOY
|
7.5 | IC50 | 2 | — | |
VKUBXLNVYQUCFV
|
7.5 | IC50 | 2 | — | |
RKZJWUOBFCJJTR
|
7.5 | Ki | 2 | — | |
ZTKAFVSUBJCXFM
|
7.5 | Ki | 3 | — | |
BNFIULLBFOWELZ
|
7.5 | IC50 | 2 | — | |
DFZYMRBKXQWSTE
|
7.5 | IC50 | 2 | — | |
GIBXFMCQBQGCKE
|
7.5 | IC50 | 2 | — | |
MHWZNBBELRMCAO
|
7.5 | IC50 | 3 | — | |
QIJJYGUDEMYDMJ
|
7.5 | IC50 | 2 | — | |
ZYOLWNDWLWOCNQ
|
7.5 | IC50 | 2 | — | |
DZIWDYAOHLYJGW
|
7.5 | IC50 | 2 | — | |
OCKLEWKOKFDMHP
|
7.5 | IC50 | 2 | — | |
KNTPSJWEFWVLCP
|
7.5 | Ki | 2 | — | |
MIPUTBSSNQTOCB
|
7.5 | Ki | 2 | — | |
MOMZVCIJGACLFL
|
7.5 | IC50 | 2 | — | |
UYBJISPAOAQTKQ
|
7.5 | IC50 | 2 | — | |
XXWVLLGWBXOMHQ
|
7.5 | IC50 | 2 | — | |
GGQRUDKBZGUEAN
|
7.5 | IC50 | 2 | — | |
HQCVWNZJFCYZOD
|
7.5 | Ki | 2 | — | |
ICFLHQGITDWVMH
|
7.5 | Ki | 2 | — | |
KDVSANSBFHATHQ
|
7.5 | IC50 | 2 | — | |
KGFMFEQQZNKWLP
|
7.5 | IC50 | 3 | — | |
LVZOQUMLGOHFGL
|
7.5 | IC50 | 3 | — | |
WWSDKIIWGPNMOK
|
7.5 | Ki | 2 | — | |
YXBSHEFOZZFYPO
|
7.5 | IC50 | 2 | — | |
JRIIXIXSRVUNTB
|
7.4 | IC50 | 2 | — | |
RMSGLBWSFHPNIN
|
7.4 | Ki | 2 | — | |
WJEDKJKCQOZDNI
|
7.4 | IC50 | 3 | — | |
ZXXGFBBNJBARSN
|
7.4 | IC50 | 2 | — | |
WHDYNTOHHUJBCQ
|
7.4 | IC50 | 2 | — | |
XTLUPLYDVHOHSW
|
7.4 | Ki | 4 | — | |
ZZZQZZTYLVXHSC
|
7.4 | IC50 | 2 | — | |
WYMZJAXBOGNVIB
|
7.4 | Ki | 2 | — | |
GDXYIWWYZWDRDL
|
7.4 | IC50 | 2 | — | |
GIRSNKRRSYXJKZ
|
7.4 | IC50 | 2 | — | |
KUWKSBLXZVHOLM
|
7.4 | IC50 | 2 | — | |
UCLMIPKAOVLOQS
|
7.4 | IC50 | 2 | — | |
IUZRAMZCEBNUIK
|
7.4 | IC50 | 2 | — | |
IXMWYDAQMMZUOZ
|
7.4 | IC50 | 2 | — | |
ZZWNDPPQMABJJG
|
7.4 | IC50 | 3 | — | |
MBZGPEHCTCTXRE
|
7.4 | Ki | 2 | — | |
IHUHWAUMFFURSJ
|
7.4 | IC50 | 2 | — | |
METQSPRSQINEEU
|
7.4 | IC50 | 3 | — | |
METQSPRSQINEEU
|
7.4 | IC50 | 3 | — | |
RZLNRXBPGQEHEO
|
7.4 | IC50 | 2 | — | |
VBGYFNUDIFNZRO
|
7.4 | Ki | 3 | — | |
ZOQCHOPYQLCJAE
|
7.4 | IC50 | 2 | — | |
DYJSODVHTVCXIA
|
7.3 | Ki | 4 | — | |
INHWHLPFIVXVHK
|
7.3 | IC50 | 2 | — | |
CXVVRTQQTVLRBH
|
7.3 | Ki | 2 | — |