Target Details
| UniProt AC | P06401 |
|---|---|
| Gene Symbol | PGR |
| Protein Name | Progesterone receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00104 (Hormone_recep) PF02161 (Prog_receptor) PF00105 (zf-C4) |
Summary
- Multi-target molecules 617
- Clinical molecules 33
- Avg pChEMBL 7.21
KEGG Pathways (5)
Associated Diseases (1)
Active Molecules (617)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ONOSXGJCDWPVFI
|
7.8 | IC50 | 2 | — | |
DQCNRZPBBUYZOQ
|
7.8 | IC50 | 2 | — | |
GUVXCWSUCSDGOW
|
7.8 | IC50 | 2 | — | |
HJOUYAMEBCDGKK
|
7.8 | IC50 | 2 | — | |
HMOAZJHSXXENHE
|
7.8 | IC50 | 3 | — | |
UFZZMZCIWOEUKP
|
7.8 | Ki | 4 | — | |
WAORTEATHIIKSN
|
7.8 | IC50 | 2 | — | |
WUXTURZHMMFRPK
|
7.8 | IC50 | 3 | — | |
ZVCDNODZUJDLPU
|
7.8 | IC50 | 2 | — | |
FZORYLRILGENBG
|
7.8 | Ki | 2 | — | |
NNWXOVXANQHVST
|
7.8 | IC50 | 2 | — | |
IJSGDARRCNDONL
|
7.8 | IC50 | 2 | — | |
RZCOQAQHAZHWEB
|
7.8 | IC50 | 3 | — | |
JOCQGPAPUMPYTP
|
7.7 | Ki | 2 | — | |
VRZVKIJRJRBQJT
|
7.7 | IC50 | 4 | — | |
OUXFXJUDVPDIII
|
7.7 | IC50 | 2 | — | |
WCWNFANFHMNQEP
|
7.7 | IC50 | 7 | Yes | |
FOPLNUAISVOILB
|
7.7 | Ki | 3 | — | |
SAVAEFOXNWPFKB
|
7.7 | Ki | 3 | — | |
WMWTYOKRWGGJOA
|
7.7 | IC50 | 4 | — | |
XTULMSXFIHGYFS
|
7.7 | IC50 | 3 | — | |
GIBZLWRPPUSMTC
|
7.7 | IC50 | 4 | — | |
LMHUNJRFYIMKDB
|
7.7 | Ki | 2 | — | |
PCGWJSDLFYYVRR
|
7.7 | Ki | 2 | — | |
URYARKSTCIJGME
|
7.7 | Ki | 3 | — | |
VKYPRKNSJRILPH
|
7.7 | Ki | 2 | — | |
VWCZQZNHWPQZGT
|
7.7 | Ki | 3 | — | |
WFESRNFSHAPECN
|
7.7 | Ki | 4 | Yes | |
ZWTCGJWGJMGWIM
|
7.7 | Ki | 3 | — | |
YKFHUVOJZGWRDY
|
7.7 | IC50 | 2 | — | |
JBHNSKHKWQLGNV
|
7.6 | Ki | 2 | — | |
MDMKCVXYKPOLIM
|
7.6 | Ki | 2 | — | |
NTXRXSSTKKNELF
|
7.6 | IC50 | 5 | Yes | |
WAORTEATHIIKSN
|
7.6 | IC50 | 2 | — | |
QFXLFIGPPAXZQQ
|
7.6 | IC50 | 2 | — | |
HUPZROPFBRSFDW
|
7.6 | Ki | 2 | — | |
IMKBAQWLEDSCAP
|
7.6 | IC50 | 2 | — | |
OMIMAFBBRNJDDU
|
7.6 | IC50 | 3 | — | |
LHEMFJILFRTVQP
|
7.6 | IC50 | 2 | — | |
NMIXBOUDRDWICA
|
7.6 | Ki | 3 | — | |
PHIKAOOZNGLKDI
|
7.6 | Ki | 4 | — | |
FQYNXWLDJCLBQP
|
7.5 | Ki | 3 | — | |
VOVIALXJUBGFJZ
|
7.5 | IC50 | 4 | — | |
JXRAVTIDZDMHLO
|
7.5 | Ki | 4 | — | |
KSRJOQNNZWTUHC
|
7.5 | Ki | 2 | — | |
PRCXSDHAGJJCKC
|
7.5 | IC50 | 2 | — | |
QXSLSLICSJPAFZ
|
7.5 | Ki | 2 | — | |
CJZROCCAPJVVQO
|
7.5 | IC50 | 3 | — | |
DXVZGTRLQAZISS
|
7.5 | IC50 | 2 | — | |
OZBSREXZWADXQE
|
7.5 | IC50 | 3 | — |