Target Details
| UniProt AC | P06401 |
|---|---|
| Gene Symbol | PGR |
| Protein Name | Progesterone receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00104 (Hormone_recep) PF02161 (Prog_receptor) PF00105 (zf-C4) |
Summary
- Multi-target molecules 617
- Clinical molecules 33
- Avg pChEMBL 7.21
KEGG Pathways (5)
Associated Diseases (1)
Active Molecules (617)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DJRBZWVBECJRTM
|
8.2 | IC50 | 2 | — | |
MWKSRKSEWLRPBL
|
8.2 | Kd | 1075 | — | |
LCDCPIOGHJGDBP
|
8.1 | IC50 | 2 | — | |
LSQKEQHYMWDEPS
|
8.1 | IC50 | 2 | — | |
CYBZSWXWFMWSAP
|
8.1 | Ki | 2 | — | |
ANPFZNKOHNLVIS
|
8.1 | IC50 | 2 | — | |
WLEYQRHXERCYNY
|
8.1 | Ki | 3 | — | |
UDDUGXMYFCMHJO
|
8.1 | IC50 | 3 | — | |
RSVKCRGCARHPAC
|
8.1 | Ki | 4 | — | |
FFBFTWHDFGXBAD
|
8.1 | Ki | 2 | — | |
NEYLJRNOSBUARA
|
8.1 | IC50 | 2 | — | |
CLZXITGNUVWIEP
|
8.0 | Ki | 2 | — | |
QASVQWYKHBDCLY
|
8.0 | IC50 | 2 | — | |
HXJYKDIOBRNHTQ
|
8.0 | IC50 | 2 | — | |
NVKFRYWNCLQAGR
|
8.0 | IC50 | 2 | — | |
GHECULMSYYJOBB
|
8.0 | Ki | 2 | — | |
ZAINQQRFGATLID
|
8.0 | Ki | 4 | — | |
STJWTSUWXXKJNZ
|
8.0 | IC50 | 2 | — | |
FDNUEWAYXCBDDX
|
8.0 | Ki | 2 | — | |
OHDDNRZGDGYKBR
|
7.9 | IC50 | 2 | — | |
BXMUAQLRVCWTKG
|
7.9 | IC50 | 3 | — | |
BBPIYWKWDHEGML
|
7.9 | IC50 | 2 | — | |
JKKYDDVIHYJRRB
|
7.9 | IC50 | 2 | — | |
SCVIEONTACSLJA
|
7.9 | IC50 | 3 | — | |
VKUBXLNVYQUCFV
|
7.9 | IC50 | 2 | — | |
WIJJCLHTLMPDEH
|
7.9 | IC50 | 2 | — | |
YSIQBSLZQKNAIY
|
7.9 | IC50 | 2 | — | |
OFRWAMYYBARBJR
|
7.9 | Ki | 2 | — | |
ZWGPOLYPUOBDPY
|
7.9 | Ki | 2 | — | |
AWYOCGCIYQEWJB
|
7.9 | Ki | 2 | — | |
DJDDNTUYFUVZIC
|
7.9 | IC50 | 2 | — | |
DVUOOXZFSLIMAG
|
7.9 | IC50 | 2 | — | |
GZULQASDNRKTNT
|
7.9 | Ki | 2 | — | |
PONOGVXIIRSESP
|
7.9 | Ki | 2 | — | |
PSGAAPLEWMOORI
|
7.9 | Ki | 2 | — | |
SPSACPMSSOTZPR
|
7.9 | IC50 | 2 | — | |
YXFZNSZDZKRXGZ
|
7.9 | IC50 | 2 | — | |
BQFHIOXHOTZDCT
|
7.9 | Ki | 2 | — | |
LUMRHKVOXMIPGU
|
7.9 | IC50 | 2 | — | |
NLPNUYHHRWOSGM
|
7.9 | IC50 | 4 | — | |
WPGAOHWZNCMFLY
|
7.9 | IC50 | 2 | — | |
IBAKVWWTMBODDP
|
7.9 | IC50 | 2 | — | |
IXAZIQYAFRPNHY
|
7.9 | Ki | 2 | — | |
FAZOJHMTURPXLD
|
7.8 | Ki | 2 | — | |
ZOUVODOOOFQPOC
|
7.8 | IC50 | 2 | — | |
DSMDXILQYZQPHU
|
7.8 | Ki | 2 | — | |
FBRSRKWFLZVSLF
|
7.8 | IC50 | 2 | — | |
HMOAZJHSXXENHE
|
7.8 | IC50 | 3 | — | |
KAVBXXNJZQGZIT
|
7.8 | IC50 | 2 | — | |
KRGAYZJXZMMOOH
|
7.8 | Ki | 2 | — |