Target Details
UniProt ACP06401
Gene SymbolPGR
Protein NameProgesterone receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00104 (Hormone_recep) PF02161 (Prog_receptor) PF00105 (zf-C4)
Summary
  • Multi-target molecules 617
  • Clinical molecules 33
  • Avg pChEMBL 7.21
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (617)
InChIKey pChEMBL Type Targets Clinical
LWYLVQVGWUQBSI 8.8 IC50 2
DTIMQMAYRMJPRM 8.8 Ki 2
NVTFLQJKFXTAOZ 8.8 Ki 2
NTYALJAURYTROE 8.7 Ki 6 Yes
VIKNJXKGJWUCNN 8.7 IC50 6 Yes
NGNZPJWDMRRGGD 8.7 Ki 2
VQFLIHCSQSPSJT 8.6 Ki 3
DLXBCJBMEVKPIX 8.6 Ki 9 Yes
JTYKTQGMYNYWGT 8.6 Ki 2
VRWXHHASXOUVMH 8.6 Ki 2
CTCHAYJBEBAVDT 8.6 Ki 6 Yes
FQYNXWLDJCLBQP 8.6 Ki 3
HKKAPCOJXICOAX 8.5 Ki 2
QFRVNOIAPBNRJM 8.5 IC50 2
BNYATMGZJPIGMW 8.5 IC50 2
DOGQPEOXOGREDU 8.5 IC50 2
PIIBHVFIQOSICN 8.5 IC50 2
VXKBREQCYRAEHY 8.5 IC50 3
CUIMAZBZRVOSOP 8.5 IC50 3
RXVVCKDZPLPROM 8.5 IC50 2
OPPYDCXBDREGJT 8.5 IC50 4
NBYXOMZEWLMKJB 8.5 Ki 3
RJKFOVLPORLFTN 8.5 Ki 10 Yes
RUEYZSNXUIKMJQ 8.5 Ki 2
KGVGNTCIQIYLQU 8.4 Ki 9 Yes
XGBWGDGYTTWUIM 8.4 Ki 3
IAUDUYJHOKBQLW 8.4 Ki 6 Yes
MWIXIWILHMYRGD 8.4 Ki 3
IMTGEDOKMRCXLE 8.4 Ki 6 Yes
NNEGFNICKYKFDF 8.4 Ki 2
KIOOLNRTWPFVHX 8.3 IC50 2
OZGJGGGYYPKMDN 8.3 Ki 3
DVIBYGTZNAJRGB 8.3 IC50 2
DZATYSMEKYVDKI 8.3 Ki 6 Yes
OCLPHOSZZDWUFZ 8.3 Ki 2
ZEZOALAOUQCQQW 8.3 Ki 3
DAZGBWZWTXJDJO 8.3 IC50 2
OGUUDCBPGBXZHI 8.3 IC50 2
ACDLPCXLODOBHE 8.3 IC50 3
SXIDZLMPGLSSSR 8.3 Ki 4
JAPBAKGEKZXGRM 8.2 Ki 3
GOHKIDSTSAUHCB 8.2 IC50 2
LGTLOCBNEXITRB 8.2 Ki 4
ANIOYQXTAMMUKZ 8.2 Ki 2
NTCBYBDADUSXSB 8.2 Ki 9 Yes
WVCKFHDLPYAJOU 8.2 Ki 5
ZDCMJDVSSLHLLQ 8.2 Ki 9 Yes
QXSLSLICSJPAFZ 8.2 Ki 3
OTDVEVBRJYVJHY 8.2 IC50 2
WFOHHEVAQLCSFM 8.2 Ki 3
2D structure