Target Details
| UniProt AC | P06401 |
|---|---|
| Gene Symbol | PGR |
| Protein Name | Progesterone receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00104 (Hormone_recep) PF02161 (Prog_receptor) PF00105 (zf-C4) |
Summary
- Multi-target molecules 617
- Clinical molecules 33
- Avg pChEMBL 7.21
KEGG Pathways (5)
Associated Diseases (1)
Active Molecules (617)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RJAYIUMTPVLORX
|
6.4 | IC50 | 2 | — | |
WFSBONJXUAXVJH
|
6.4 | IC50 | 3 | — | |
AXLNGHICNRTHMP
|
6.4 | IC50 | 2 | — | |
FFFOIRSYFQWGQH
|
6.4 | Ki | 2 | — | |
APDOEOQZQMSOFL
|
6.4 | IC50 | 2 | — | |
NLDACKJWSTTYSC
|
6.4 | Ki | 2 | — | |
ZDRUXXZVOLZIBA
|
6.4 | IC50 | 2 | — | |
ALDWINSGSURGLP
|
6.4 | IC50 | 3 | — | |
IJUMJWCKSDCFGS
|
6.4 | IC50 | 2 | — | |
JGAKOXMSUKTZLQ
|
6.4 | IC50 | 2 | — | |
MMLSXRYBGYGQEP
|
6.4 | IC50 | 2 | — | |
QYGXPNCCWFGVRU
|
6.4 | Ki | 2 | — | |
DPPNIDONMQTQMK
|
6.4 | Ki | 3 | — | |
KJUOEYJRZUJJLM
|
6.4 | IC50 | 3 | — | |
OHUSXUGFNIRYCY
|
6.4 | IC50 | 2 | — | |
ORGKYZVJZBDUGT
|
6.4 | IC50 | 2 | — | |
OSHWKQSKIVSROR
|
6.4 | IC50 | 2 | — | |
OSRXVTVKOPCOGY
|
6.4 | Ki | 3 | — | |
RHQPXBHOFIZXKG
|
6.4 | IC50 | 2 | — | |
UMKDQHBGTUYJCV
|
6.4 | IC50 | 2 | — | |
AWBMTFDCCHSMQU
|
6.4 | Ki | 2 | — | |
FBHBBILQSLGKPC
|
6.4 | Ki | 2 | — | |
HFWXCPFGOCGJDK
|
6.4 | IC50 | 3 | — | |
WDXRGPWQVHZTQJ
|
6.4 | IC50 | 5 | — | |
WOYXGESYPYMTAQ
|
6.4 | Ki | 2 | — | |
YDRMSDHDYRAUBR
|
6.4 | IC50 | 2 | — | |
PKGWJFNRGGGBJB
|
6.4 | IC50 | 3 | — | |
VPGLREFJYMSJHR
|
6.4 | Ki | 2 | — | |
XNULRSOGWPFPBL
|
6.4 | IC50 | 2 | — | |
CMHJMUZTXMDMKL
|
6.4 | IC50 | 3 | — | |
CPUIRDMVUBPAPK
|
6.4 | Ki | 3 | — | |
GTZWEKOQKQIWQD
|
6.4 | IC50 | 2 | — | |
IMGXWRKTVOMDLZ
|
6.4 | IC50 | 3 | — | |
QSDGRHKNICEVHX
|
6.4 | IC50 | 3 | — | |
CXFSVKGROITHRY
|
6.3 | Ki | 3 | — | |
FBLDDBTTXDBIGE
|
6.3 | Ki | 2 | — | |
HAJBHFSMKOWEHU
|
6.3 | IC50 | 2 | — | |
NAKVZBYNDIOTLA
|
6.3 | IC50 | 3 | — | |
OTRYZVITNGFGQP
|
6.3 | IC50 | 2 | — | |
PFUXODWITQFWRK
|
6.3 | Ki | 2 | — | |
SSAMEZHVGWGDGH
|
6.3 | IC50 | 3 | — | |
XOSVCJKDUIUUIB
|
6.3 | Ki | 2 | — | |
YWPNXVQAAHGWCZ
|
6.3 | IC50 | 2 | — | |
YXQPDNYJXVGIES
|
6.3 | Ki | 2 | — | |
FLXKJKBDBACQDP
|
6.3 | IC50 | 2 | — | |
QEYIPZOJYLGUHY
|
6.3 | IC50 | 2 | — | |
NOUXCOKPRXVTDP
|
6.3 | Ki | 4 | — | |
PVYTWCNJUWKUOG
|
6.3 | IC50 | 3 | — | |
AHCZZOJYVQVLQG
|
6.3 | IC50 | 3 | — | |
BTEQZWJLBYEBLQ
|
6.3 | Ki | 4 | — |