Target Details
| UniProt AC | P06401 |
|---|---|
| Gene Symbol | PGR |
| Protein Name | Progesterone receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00104 (Hormone_recep) PF02161 (Prog_receptor) PF00105 (zf-C4) |
Summary
- Multi-target molecules 617
- Clinical molecules 33
- Avg pChEMBL 7.21
KEGG Pathways (5)
Associated Diseases (1)
Active Molecules (617)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VHZPUDNSVGRVMB
|
11.5 | IC50 | 2 | — | |
WOFMFGQZHJDGCX
|
10.1 | Kd | 3 | — | |
OAYLSAHITBROEB
|
10.0 | IC50 | 2 | — | |
PDEYZVGOCYDQJF
|
9.7 | IC50 | 3 | — | |
VWUXBMIQPBEWFH
|
9.7 | IC50 | 8 | Yes | |
DZKSHTKHHHLSGZ
|
9.5 | IC50 | 3 | — | |
GJMNAFGEUJBOCE
|
9.5 | IC50 | 5 | Yes | |
HDCJFWTUMAKTNA
|
9.5 | IC50 | 2 | — | |
OHLMRBMVXRKABN
|
9.5 | Ki | 2 | — | |
GKQWMOXIBZCMDJ
|
9.5 | Ki | 3 | — | |
PSGAAPLEWMOORI
|
9.5 | Ki | 11 | Yes | |
WIUDNDXMQHQJIL
|
9.5 | IC50 | 2 | — | |
RCZNQWQDJPJWMD
|
9.4 | IC50 | 3 | — | |
WNRXXFMGMKLIHP
|
9.4 | Ki | 5 | Yes | |
MEFYNCWNNHNHMN
|
9.4 | Ki | 3 | — | |
IDGIKWDCKXJAES
|
9.4 | Ki | 3 | — | |
YTMMXBWUMWUPPN
|
9.3 | Ki | 2 | — | |
CCCIJQPRIXGQOE
|
9.3 | Ki | 4 | — | |
NPDSJEIIHNPHHF
|
9.3 | Ki | 2 | — | |
SSFWXDSRZJERKU
|
9.3 | Ki | 2 | — | |
HMBNPWKLPBPJMY
|
9.3 | Ki | 3 | — | |
POYMYRFGHYKMSL
|
9.3 | Ki | 4 | — | |
ISFPMZBOTSJQDY
|
9.2 | Ki | 2 | — | |
YISCUJJPIJSXKK
|
9.2 | IC50 | 2 | — | |
QCRMHUMUIWUQMT
|
9.2 | Ki | 3 | — | |
RTLRJRHSVSOAFD
|
9.2 | Ki | 3 | — | |
YXKBVHXOKVRRKO
|
9.2 | Ki | 6 | Yes | |
JIKFLEZNTIZKCI
|
9.2 | IC50 | 4 | — | |
HTCMKQLSSZWFTP
|
9.2 | Ki | 5 | Yes | |
TXUZVZSFRXZGTL
|
9.1 | IC50 | 7 | Yes | |
TXUZVZSFRXZGTL
|
9.1 | IC50 | 6 | — | |
OVIZCQBEPZRBDB
|
9.1 | Ki | 3 | — | |
BDYFDDGUXXUNJN
|
9.1 | Ki | 5 | Yes | |
KJSHBZLXBZYVMR
|
9.1 | Ki | 3 | — | |
ACXANRVNFDEJLV
|
9.0 | Ki | 2 | — | |
CEDQCHHKNHJFKO
|
9.0 | IC50 | 2 | — | |
WIMXURNPWBOQET
|
9.0 | IC50 | 4 | — | |
UAXYYPCBGHLJKQ
|
9.0 | Ki | 3 | — | |
YPUGASLTKIAOPT
|
9.0 | Ki | 6 | Yes | |
QFRVNOIAPBNRJM
|
8.9 | IC50 | 2 | — | |
CWXNSHLNBNLSSS
|
8.9 | Ki | 3 | — | |
MMQYPFTZXJAWGY
|
8.9 | Ki | 5 | Yes | |
RFZAHUIHPLZLLA
|
8.9 | Ki | 9 | Yes | |
YKQNBGVCIMLMLA
|
8.9 | Ki | 3 | — | |
FOPLNUAISVOILB
|
8.9 | Ki | 2 | — | |
MYDJWFCWWHPKCH
|
8.9 | Ki | 6 | Yes | |
KCVAVMXQQQXOLI
|
8.8 | Ki | 6 | Yes | |
LVCVMYKRVFAVCM
|
8.8 | Ki | 6 | Yes | |
UDYVQHLPMVKSOP
|
8.8 | Ki | 3 | — | |
ZVALABNDJZPNNC
|
8.8 | Ki | 3 | — |