Target Details
| UniProt AC | P06239 |
|---|---|
| Gene Symbol | LCK |
| Protein Name | Tyrosine-protein kinase Lck |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 1,537
- Clinical molecules 323
- Avg pChEMBL 7.15
KEGG Pathways (11)
- Human T-cell leukemia virus 1 infection
- IgSF CAM signaling
- NF-kappa B signaling pathway
- Natural killer cell mediated cytotoxicity
- Osteoclast differentiation
- PD-L1 expression and PD-1 checkpoint pathway in cancer
- Primary immunodeficiency
- T cell receptor signaling pathway
- Th1 and Th2 cell differentiation
- Th17 cell differentiation
- Yersinia infection
Associated Diseases (1)
Active Molecules (1,537)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JHDISIQMSVRVDG
|
6.3 | IC50 | 2 | — | |
JKTCYIDJXKFDGR
|
6.3 | IC50 | 3 | — | |
JRKSMTJDASLJBM
|
6.3 | IC50 | 3 | — | |
JUQXOMJYFWIQTO
|
6.3 | IC50 | 2 | — | |
KAOQBTDPUNWJTJ
|
6.3 | IC50 | 2 | — | |
KIXARXKYLWVJKE
|
6.3 | IC50 | 2 | — | |
KMKHVCGUHDWGJX
|
6.3 | IC50 | 2 | — | |
KSUUWWFAWIJYCZ
|
6.3 | IC50 | 3 | — | |
KUCNBQPAJZRQMJ
|
6.3 | IC50 | 11 | — | |
KVUZGQPEVDLDTA
|
6.3 | IC50 | 3 | — | |
LNVFYQLXYPFVNQ
|
6.3 | IC50 | 2 | — | |
LTWKJBFCYCDGCV
|
6.3 | IC50 | 2 | — | |
LUCKLKMOCDVQCV
|
6.3 | IC50 | 2 | — | |
MDBVZQSAIDJNIM
|
6.3 | IC50 | 2 | — | |
MUEFXKOEGUVPMC
|
6.3 | IC50 | 2 | — | |
MZMWNDRVYSIOHF
|
6.3 | IC50 | 2 | — | |
NIZWHJVGPCZQDZ
|
6.3 | IC50 | 3 | — | |
NQHRIAKNZJDTIS
|
6.3 | IC50 | 2 | — | |
NQVBBSCHHCKTOV
|
6.3 | IC50 | 3 | — | |
NXORMUJXJIKJBQ
|
6.3 | IC50 | 3 | — | |
OIBIOFXJAJUALW
|
6.3 | IC50 | 3 | — | |
OJEIECWWENNREZ
|
6.3 | IC50 | 2 | — | |
OMYAWPJJRZDQRE
|
6.3 | IC50 | 3 | — | |
PGOUMVSFSMZEQT
|
6.3 | IC50 | 3 | — | |
PJYYQTWKVBLVSS
|
6.3 | IC50 | 3 | — | |
PLKXLSABUWNGOL
|
6.3 | IC50 | 2 | — | |
PTGDURRRTYAKSP
|
6.3 | IC50 | 2 | — | |
PUKGRYCUACBXDB
|
6.3 | IC50 | 2 | — | |
QILQLPCWLHMKEX
|
6.3 | IC50 | 2 | — | |
QINBBTYIMWCVSQ
|
6.3 | IC50 | 2 | — | |
QMPCZRYAQUSGAU
|
6.3 | IC50 | 2 | — | |
QOJBPFSVPCKOOF
|
6.3 | IC50 | 3 | — | |
QQCIEUDKVLVHCV
|
6.3 | IC50 | 2 | — | |
QZCWPDPWSBOTEU
|
6.3 | IC50 | 7 | — | |
QZTCIPMCYKMSIT
|
6.3 | IC50 | 2 | — | |
RDBFWDTVOKUUGE
|
6.3 | IC50 | 3 | — | |
RITKUWAOEQBXTJ
|
6.3 | IC50 | 2 | Yes | |
RPQORVRVHTUMJD
|
6.3 | IC50 | 2 | — | |
RPTKFSUYFFYRIA
|
6.3 | IC50 | 2 | — | |
RWCFKPKDVWBGSU
|
6.3 | IC50 | 2 | — | |
SDGOXLDKFDEURY
|
6.3 | IC50 | 3 | — | |
SFKPBKWXQBFJHD
|
6.3 | IC50 | 2 | — | |
SGOXRXKFGRPCNW
|
6.3 | IC50 | 3 | — | |
SILNPGWUEYVWOG
|
6.3 | IC50 | 3 | — | |
SNXSBHRORYNWID
|
6.3 | IC50 | 2 | — | |
SRXOUOLDYVNBOW
|
6.3 | IC50 | 3 | — | |
STCSTSSDRJJGME
|
6.3 | IC50 | 4 | — | |
SZCFGZXOLAMRLX
|
6.3 | IC50 | 2 | — | |
TUUBKLDDTMKOCQ
|
6.3 | IC50 | 2 | — | |
TYSQKGWYQQCUCN
|
6.3 | IC50 | 2 | — |