Target Details
| UniProt AC | P06239 |
|---|---|
| Gene Symbol | LCK |
| Protein Name | Tyrosine-protein kinase Lck |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 1,537
- Clinical molecules 323
- Avg pChEMBL 7.15
KEGG Pathways (11)
- Human T-cell leukemia virus 1 infection
- IgSF CAM signaling
- NF-kappa B signaling pathway
- Natural killer cell mediated cytotoxicity
- Osteoclast differentiation
- PD-L1 expression and PD-1 checkpoint pathway in cancer
- Primary immunodeficiency
- T cell receptor signaling pathway
- Th1 and Th2 cell differentiation
- Th17 cell differentiation
- Yersinia infection
Associated Diseases (1)
Active Molecules (1,537)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HPDAVKSNTNLCBE
|
6.3 | IC50 | 3 | — | |
OVDBDNFZYMESOZ
|
6.3 | IC50 | 7 | — | |
QBWKPGNFQQJGFY
|
6.3 | IC50 | 5 | Yes | |
SRHZWIQYIDTHNP
|
6.3 | IC50 | 2 | — | |
WRAKTDGEPIERFS
|
6.3 | IC50 | 3 | — | |
AHOHWELPUXLPOF
|
6.3 | IC50 | 3 | — | |
KFTIUYWZCYZUGD
|
6.3 | IC50 | 3 | — | |
NKHIQOIFPZJFIJ
|
6.3 | IC50 | 3 | — | |
QGKULZNNOSWVPX
|
6.3 | IC50 | 2 | — | |
TUKOILYAIRACKC
|
6.3 | IC50 | 7 | Yes | |
UQRCJCNVNUFYDX
|
6.3 | Kd | 27 | — | |
WAKUIUNRDNSMQR
|
6.3 | Kd | 4 | — | |
MREXTQDSRCXTPN
|
6.3 | IC50 | 2 | — | |
OIJOOTMJWCNRQR
|
6.3 | IC50 | 2 | — | |
AYPQJCUSHCNNTD
|
6.3 | IC50 | 2 | — | |
BAFUFCIHPPFMHP
|
6.3 | IC50 | 3 | — | |
BNRJMXPCHXXMHT
|
6.3 | IC50 | 2 | — | |
BVAAFYRYVXTSGN
|
6.3 | IC50 | 3 | — | |
CBVUEAAQUJJHEA
|
6.3 | IC50 | 2 | — | |
CEAVFNQUCMOSMX
|
6.3 | IC50 | 3 | — | |
CMJGHWQDYMQXML
|
6.3 | IC50 | 2 | — | |
DAILMCHHPABCQU
|
6.3 | IC50 | 2 | — | |
DJBQGUXCAGMWNN
|
6.3 | IC50 | 3 | — | |
DMKUUHTTZPWLKF
|
6.3 | IC50 | 3 | — | |
DUTDXWCWCUJBLI
|
6.3 | IC50 | 3 | — | |
FGVHSAZTCGXYQT
|
6.3 | IC50 | 4 | — | |
FQCRNGFAAPZXFR
|
6.3 | IC50 | 2 | — | |
FQUIFYYDFZJJPV
|
6.3 | IC50 | 3 | — | |
FYLYZGYKYWJXEB
|
6.3 | IC50 | 2 | — | |
GFOHVJWVMQVBAU
|
6.3 | IC50 | 3 | — | |
GIBGWAMSRVOAKH
|
6.3 | IC50 | 3 | — | |
GJVRHNMHPUDIPK
|
6.3 | IC50 | 2 | — | |
GNUGYSKRAVVTRC
|
6.3 | IC50 | 2 | — | |
GQWYJNLBYWGULF
|
6.3 | IC50 | 2 | — | |
GZAQYCKKZVFFBO
|
6.3 | IC50 | 2 | — | |
HCIKRLPTFHVQGO
|
6.3 | IC50 | 3 | — | |
HDCPYODOQCXBDF
|
6.3 | IC50 | 3 | — | |
HEJMJEVSIIMKLI
|
6.3 | IC50 | 3 | — | |
HQWCPDUIKCIHEE
|
6.3 | IC50 | 3 | — | |
HXYLOJPXLAXQBK
|
6.3 | IC50 | 2 | — | |
IACPUILVLDGVIT
|
6.3 | IC50 | 3 | — | |
IBBDJASTLYREBW
|
6.3 | IC50 | 2 | — | |
IGFDSAPXMROBGZ
|
6.3 | IC50 | 2 | — | |
ILNFQODSBZTDGY
|
6.3 | IC50 | 3 | — | |
IOJROWSVDGSWME
|
6.3 | IC50 | 2 | — | |
IQBNYZLVGAFZIF
|
6.3 | IC50 | 2 | — | |
IWSCCPLUWZOTIQ
|
6.3 | IC50 | 2 | — | |
JBSYSXFZYWYJEL
|
6.3 | IC50 | 2 | — | |
JDCXTBTYAGHEQT
|
6.3 | IC50 | 2 | — | |
JGDSBJDDFRVDDI
|
6.3 | IC50 | 3 | — |