Target Details
| UniProt AC | P06239 |
|---|---|
| Gene Symbol | LCK |
| Protein Name | Tyrosine-protein kinase Lck |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 1,537
- Clinical molecules 323
- Avg pChEMBL 7.15
KEGG Pathways (11)
- Human T-cell leukemia virus 1 infection
- IgSF CAM signaling
- NF-kappa B signaling pathway
- Natural killer cell mediated cytotoxicity
- Osteoclast differentiation
- PD-L1 expression and PD-1 checkpoint pathway in cancer
- Primary immunodeficiency
- T cell receptor signaling pathway
- Th1 and Th2 cell differentiation
- Th17 cell differentiation
- Yersinia infection
Associated Diseases (1)
Active Molecules (1,537)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZJYIHVVBPSRRSO
|
6.7 | IC50 | 2 | — | |
ZTSOUDMNSOYCTG
|
6.7 | IC50 | 10 | — | |
CNWIKXJNZAJWKF
|
6.7 | IC50 | 2 | — | |
FWRZHTGVAAQEJX
|
6.7 | IC50 | 3 | — | |
RPZBWDOAZIJTBM
|
6.7 | IC50 | 2 | — | |
ZEUMEZFBWOSCJL
|
6.7 | IC50 | 3 | — | |
JAZNXJCUDFXHRC
|
6.6 | IC50 | 3 | — | |
JZTVWMNQNFKFGJ
|
6.6 | IC50 | 3 | Yes | |
NQWJYXLLLYRYCZ
|
6.6 | IC50 | 2 | — | |
RGCNFAMRCLHNFW
|
6.6 | IC50 | 3 | — | |
WINHZLLDWRZWRT
|
6.6 | Kd | 201 | Yes | |
MADROAFGGPUYNI
|
6.6 | IC50 | 4 | — | |
WZUGJNYAYDDNBV
|
6.6 | IC50 | 3 | — | |
CXXTWUWDVIYTID
|
6.6 | IC50 | 2 | — | |
HWFCHCRFQWEFMU
|
6.6 | Kd | 2 | — | |
MDBBPOZQZACUGK
|
6.6 | IC50 | 6 | Yes | |
QXDWLMJUKFRTHN
|
6.6 | IC50 | 2 | — | |
UQDLRCLRFNHSAU
|
6.6 | IC50 | 3 | — | |
VQAXOIUGIWGEFE
|
6.6 | Ki | 2 | — | |
XBTDIGWGOZVBHQ
|
6.6 | IC50 | 4 | Yes | |
REAMBIDJUBDLKK
|
6.6 | IC50 | 2 | — | |
AAKJLRGGTJKAMG
|
6.6 | Kd | 50 | Yes | |
ADMFLILDQJSEIK
|
6.6 | Ki | 72 | — | |
GWMATETWMAQOFL
|
6.6 | Ki | 36 | — | |
ILUGAYBMBIJXHC
|
6.6 | Ki | 9 | — | |
KOHNRDPXFDZZJF
|
6.6 | Ki | 31 | — | |
NSYXCWYWACQNOH
|
6.6 | Ki | 10 | — | |
NWMPVMMGSHXANZ
|
6.6 | Ki | 58 | — | |
PDZAPYOZOLWESW
|
6.6 | IC50 | 4 | — | |
PIQCTGMSNWUMAF
|
6.6 | Kd | 137 | Yes | |
RJZDECGDCKOHBV
|
6.6 | Ki | 70 | — | |
SJMFZIGFOIPNPE
|
6.6 | Ki | 10 | — | |
TVUWQDLBEOZVOU
|
6.6 | Ki | 41 | — | |
VMOVZKURWYNTLN
|
6.6 | Ki | 7 | — | |
WFTZMAAMCVPJJT
|
6.6 | Ki | 26 | — | |
YNVBUFWEFFQVHM
|
6.6 | Ki | 3 | — | |
YSUBPTBQVXDZFZ
|
6.6 | Ki | 2 | — | |
ZXLFIHLBHMLHFJ
|
6.6 | Ki | 31 | — | |
HXENBONILQLPNV
|
6.6 | IC50 | 3 | — | |
ITCYMXGHPXIVGP
|
6.6 | IC50 | 2 | — | |
XYSMLTDOEYEKPK
|
6.6 | IC50 | 3 | — | |
DZIUPOCVDSYPSY
|
6.6 | IC50 | 8 | Yes | |
HYNCPFLCZJKDDV
|
6.6 | IC50 | 2 | — | |
LQQYARMJQBHKQQ
|
6.6 | IC50 | 2 | — | |
QDRHYWFULQVDMF
|
6.6 | IC50 | 2 | Yes | |
SAMCEVLBPWDZMX
|
6.6 | IC50 | 5 | Yes | |
SDZFNFGEAWBFTM
|
6.6 | Ki | 2 | — | |
SHPFDGWALWEPGS
|
6.6 | Kd | 35 | — | |
TWTKQXHGZXXULH
|
6.6 | IC50 | 2 | — | |
XZIADLYCTOCKRV
|
6.6 | IC50 | 5 | — |