Target Details
| UniProt AC | P06239 |
|---|---|
| Gene Symbol | LCK |
| Protein Name | Tyrosine-protein kinase Lck |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 1,537
- Clinical molecules 323
- Avg pChEMBL 7.15
KEGG Pathways (11)
- Human T-cell leukemia virus 1 infection
- IgSF CAM signaling
- NF-kappa B signaling pathway
- Natural killer cell mediated cytotoxicity
- Osteoclast differentiation
- PD-L1 expression and PD-1 checkpoint pathway in cancer
- Primary immunodeficiency
- T cell receptor signaling pathway
- Th1 and Th2 cell differentiation
- Th17 cell differentiation
- Yersinia infection
Associated Diseases (1)
Active Molecules (1,537)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LQNDDQQRHZEHDD
|
6.7 | IC50 | 6 | Yes | |
RNOAOAWBMHREKO
|
6.7 | IC50 | 15 | — | |
XBINIPRQWSOQIE
|
6.7 | IC50 | 4 | Yes | |
LWMPTEZPBQOOSS
|
6.7 | IC50 | 3 | — | |
CWDDXFOLUXZGBV
|
6.7 | IC50 | 3 | — | |
OSAWFUCUZJNEID
|
6.7 | IC50 | 20 | — | |
ACNCCUVYXQGPKZ
|
6.7 | Ki | 31 | — | |
CHWHVQUNCYDPDK
|
6.7 | IC50 | 6 | Yes | |
DMTDZFGYURLLKX
|
6.7 | Ki | 13 | Yes | |
FQYLJBVSYHZWLT
|
6.7 | Ki | 35 | Yes | |
GNLAGGCSJGJECE
|
6.7 | Ki | 19 | Yes | |
JAMDNXUAYUHJLJ
|
6.7 | Ki | 40 | — | |
LDACHLNBCOVNBL
|
6.7 | IC50 | 8 | — | |
LSFLAQVDISHMNB
|
6.7 | Ki | 13 | — | |
MFAQYJIYDMLAIM
|
6.7 | Kd | 130 | Yes | |
MVPRWLBKNHWFPM
|
6.7 | IC50 | 6 | — | |
PFDUFECOJKSDAT
|
6.7 | Ki | 2 | — | |
QONPPIZSNSSCSK
|
6.7 | Ki | 45 | Yes | |
RKLGMDOZEOTQEM
|
6.7 | Ki | 12 | — | |
RYYNGWLOYLRZLK
|
6.7 | Ki | 104 | — | |
TZPUNPWJLMOANL
|
6.7 | IC50 | 6 | — | |
UTQPKPHUIMHAAN
|
6.7 | Ki | 22 | — | |
VTMJLOMESRVYBL
|
6.7 | IC50 | 5 | Yes | |
XBAIEEJJCJHBDL
|
6.7 | Ki | 17 | — | |
XMGFTZYNTYNOOJ
|
6.7 | Ki | 10 | — | |
YACXOXQTGJXYNX
|
6.7 | Ki | 11 | — | |
YEHCNYAQEBQCCS
|
6.7 | Ki | 74 | — | |
BTVPMDAMCUGYJV
|
6.7 | IC50 | 4 | — | |
MPFMLTBUDZGFRW
|
6.7 | IC50 | 2 | — | |
YBKODNZGBUDZRA
|
6.7 | IC50 | 3 | — | |
AAAXBDFZRXKRPL
|
6.7 | IC50 | 6 | Yes | |
AVHVXKAONMHRSS
|
6.7 | IC50 | 2 | — | |
GQHAHPQLCBBLDS
|
6.7 | Ki | 2 | — | |
HVXKQKFEHMGHSL
|
6.7 | Kd | 21 | — | |
JWXOLXZYHPKDLX
|
6.7 | IC50 | 4 | Yes | |
LEODTNLMHLRQCI
|
6.7 | IC50 | 2 | — | |
OHVZGZMTULBSNX
|
6.7 | IC50 | 2 | — | |
QUIQCYFSBGOBKE
|
6.7 | IC50 | 4 | — | |
WWXRVDUEBRGDFI
|
6.7 | IC50 | 2 | — | |
XKFTZKGMDDZMJI
|
6.7 | IC50 | 64 | Yes | |
ZAZQUFKQXMNBTJ
|
6.7 | IC50 | 4 | — | |
BTULSRXNMQZJDX
|
6.7 | IC50 | 2 | — | |
HIHOEGPXVVKJPP
|
6.7 | IC50 | 10 | — | |
CARJPEPCULYFFP
|
6.7 | Kd | 2 | — | |
CYTZASCNUGMIJP
|
6.7 | IC50 | 3 | Yes | |
FLQOKVHRJKLLEM
|
6.7 | IC50 | 3 | — | |
KGOIBABWCFAULY
|
6.7 | IC50 | 2 | — | |
REDBMKRPRFVCHI
|
6.7 | IC50 | 4 | Yes | |
RQVWDOMMFOUDTO
|
6.7 | IC50 | 3 | — | |
WNPDKPSZWPJRTH
|
6.7 | IC50 | 2 | — |