Target Details
| UniProt AC | P06239 |
|---|---|
| Gene Symbol | LCK |
| Protein Name | Tyrosine-protein kinase Lck |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 1,537
- Clinical molecules 323
- Avg pChEMBL 7.15
KEGG Pathways (11)
- Human T-cell leukemia virus 1 infection
- IgSF CAM signaling
- NF-kappa B signaling pathway
- Natural killer cell mediated cytotoxicity
- Osteoclast differentiation
- PD-L1 expression and PD-1 checkpoint pathway in cancer
- Primary immunodeficiency
- T cell receptor signaling pathway
- Th1 and Th2 cell differentiation
- Th17 cell differentiation
- Yersinia infection
Associated Diseases (1)
Active Molecules (1,537)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UJWXPHLWGVGIBB
|
7.3 | IC50 | 4 | Yes | |
UMNQEFXKDFGFNN
|
7.3 | Ki | 3 | — | |
UORAPQCBWYIISR
|
7.3 | IC50 | 12 | — | |
ZBCMHWUFWQFPLV
|
7.3 | IC50 | 9 | — | |
JPVQIIJQJZQGID
|
7.3 | IC50 | 4 | — | |
NESWXWLBMJYMDN
|
7.3 | IC50 | 3 | — | |
WQGHFGVHDRESMV
|
7.3 | IC50 | 3 | — | |
YDEDKRCWCCZXBE
|
7.3 | IC50 | 2 | — | |
AHEHCOROUMSVIO
|
7.3 | IC50 | 3 | — | |
AIFHSMOHDXGQMU
|
7.3 | IC50 | 2 | — | |
ATUMYQDCTGAFQY
|
7.3 | IC50 | 3 | — | |
BILNBAJWFVQGPG
|
7.3 | IC50 | 3 | — | |
BWYRLNXYRATYLM
|
7.3 | IC50 | 3 | — | |
BXNLHIVDMFDPAE
|
7.3 | IC50 | 2 | — | |
CBOOJABGBDIPBW
|
7.3 | IC50 | 3 | — | |
CDOHBLOZNLWOGC
|
7.3 | IC50 | 3 | — | |
CLQARABFQAGBAO
|
7.3 | IC50 | 3 | — | |
CXHZBOWLLILCRJ
|
7.3 | IC50 | 3 | — | |
DETYKZQLJPWOEJ
|
7.3 | IC50 | 3 | — | |
DPZGKYJHTOSMIA
|
7.3 | IC50 | 8 | — | |
FSCGAETYKPUJTF
|
7.3 | IC50 | 3 | — | |
FXQFQTDJCPCULX
|
7.3 | IC50 | 3 | Yes | |
GBZJWIWJKOKRGY
|
7.3 | IC50 | 3 | — | |
GRDQZTOKRYJEOD
|
7.3 | IC50 | 2 | — | |
HAFULHYXIOMYIW
|
7.3 | IC50 | 2 | — | |
HPHASEBRPJNUNL
|
7.3 | IC50 | 4 | — | |
JAXHLQYMTYAKTB
|
7.3 | IC50 | 3 | — | |
JCGXVYWABUYORV
|
7.3 | IC50 | 3 | — | |
JTUXDMHTCPSLEV
|
7.3 | IC50 | 2 | — | |
KJNOYLPRXXIEBI
|
7.3 | IC50 | 3 | — | |
KRBQVVJHGYWGFT
|
7.3 | IC50 | 2 | — | |
KZRDVFBPXXGSPD
|
7.3 | IC50 | 9 | — | |
LISZDFNSVXOEPV
|
7.3 | IC50 | 3 | — | |
LLUKGAWEUSVECT
|
7.3 | IC50 | 3 | — | |
MFVBCGSKSUGDCV
|
7.3 | IC50 | 3 | — | |
MHHXPHQTWQDELX
|
7.3 | IC50 | 2 | — | |
MILFETYWHLVOSO
|
7.3 | IC50 | 3 | — | |
MJQGHLODJHABRA
|
7.3 | IC50 | 10 | — | |
MRLOXOXQQPFOTC
|
7.3 | IC50 | 3 | — | |
MSLPJPREOGINFQ
|
7.3 | IC50 | 3 | — | |
NDQDOSYMYFLJFT
|
7.3 | IC50 | 3 | — | |
NOGZQTIFJFLZQV
|
7.3 | IC50 | 2 | — | |
NQPDYSIWILAKNW
|
7.3 | IC50 | 2 | — | |
OHKHARJWBBQMQI
|
7.3 | IC50 | 3 | — | |
OKHDBWUWJJHQTM
|
7.3 | IC50 | 4 | — | |
OLAAZMUTOKWQQN
|
7.3 | IC50 | 3 | — | |
OMIPTFNPFSGFLX
|
7.3 | IC50 | 2 | — | |
OTPKESFCTVIJSI
|
7.3 | IC50 | 2 | — | |
OWSJCCYMPPTALW
|
7.3 | IC50 | 3 | — | |
PZUMBRCJMFLXDR
|
7.3 | IC50 | 2 | — |