Target Details
| UniProt AC | P06239 |
|---|---|
| Gene Symbol | LCK |
| Protein Name | Tyrosine-protein kinase Lck |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 1,537
- Clinical molecules 323
- Avg pChEMBL 7.15
KEGG Pathways (11)
- Human T-cell leukemia virus 1 infection
- IgSF CAM signaling
- NF-kappa B signaling pathway
- Natural killer cell mediated cytotoxicity
- Osteoclast differentiation
- PD-L1 expression and PD-1 checkpoint pathway in cancer
- Primary immunodeficiency
- T cell receptor signaling pathway
- Th1 and Th2 cell differentiation
- Th17 cell differentiation
- Yersinia infection
Associated Diseases (1)
Active Molecules (1,537)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DBRQJIDNJIDEEK
|
7.6 | IC50 | 3 | — | |
DZEXCTFXOCMPSR
|
7.6 | IC50 | 3 | — | |
HFYHVKQQIOBAEU
|
7.6 | IC50 | 3 | — | |
MQRYORPEARKGSY
|
7.6 | IC50 | 4 | Yes | |
OSSISQQUQBLCRH
|
7.6 | IC50 | 2 | Yes | |
YKMSWECJITXGJA
|
7.6 | IC50 | 2 | — | |
AIEXZXMQDAIFBL
|
7.6 | IC50 | 3 | — | |
DHNJHSZXQFFMAJ
|
7.6 | IC50 | 3 | — | |
HXENBONILQLPNV
|
7.6 | IC50 | 3 | — | |
ITJWOPPSOKMWCK
|
7.6 | IC50 | 3 | Yes | |
LATXWNUJNSSMHV
|
7.6 | IC50 | 3 | — | |
OHIWAMBAFXDJCL
|
7.6 | IC50 | 3 | — | |
CSCOHEYTBLBQMG
|
7.5 | IC50 | 7 | Yes | |
GLDQJVYQRVZJIH
|
7.5 | IC50 | 3 | — | |
LAUHLGUSVSJYCI
|
7.5 | IC50 | 16 | — | |
MRZJQHJHMLBKTE
|
7.5 | IC50 | 2 | Yes | |
SXGLKAJWKHWEPI
|
7.5 | IC50 | 3 | — | |
WGBGLPNMHGTLQS
|
7.5 | IC50 | 3 | Yes | |
WSTUJEXAPHIEIM
|
7.5 | Kd | 10 | — | |
FQXQXOYNTXHBKK
|
7.5 | IC50 | 7 | — | |
LIOQVOACFAJWND
|
7.5 | IC50 | 3 | — | |
ZEYDBVDHJVJKOI
|
7.5 | IC50 | 3 | — | |
ZMWKUKIYVSUWAS
|
7.5 | IC50 | 4 | — | |
BJFQIPBUHJGODW
|
7.5 | IC50 | 3 | — | |
ORCBPUXWRVQPOS
|
7.5 | IC50 | 3 | — | |
OTTCBLPTHPBEEX
|
7.5 | Ki | 11 | Yes | |
PFZMYXREESNCJF
|
7.5 | IC50 | 3 | — | |
BNHYZCBZOBOXAW
|
7.5 | IC50 | 3 | — | |
HKSZLNNOFSGOKW
|
7.5 | Kd | 213 | — | |
JNIIGOXKPNCTTH
|
7.5 | IC50 | 4 | Yes | |
KRYULLMPWHIEHI
|
7.5 | IC50 | 2 | — | |
KTEIFNKAUNYNJU
|
7.5 | Kd | 114 | — | |
NHHQJBCNYHBUSI
|
7.5 | Kd | 220 | — | |
WYNDNQIGGGWABE
|
7.5 | IC50 | 4 | — | |
YAXIXGGRDHAOJL
|
7.5 | IC50 | 3 | — | |
ZJABPXCKZJSAKI
|
7.5 | IC50 | 3 | — | |
CUIYKFICQYRIMQ
|
7.5 | IC50 | 3 | Yes | |
FNTHJTUPRVAXFZ
|
7.5 | IC50 | 17 | — | |
LXURGGKEOPHREO
|
7.5 | IC50 | 13 | — | |
NITOVUIHLVISSN
|
7.5 | IC50 | 5 | Yes | |
ULBYNJSRGACZJB
|
7.5 | IC50 | 3 | — | |
WJEOLQLKVOPQFV
|
7.5 | Kd | 24 | — | |
ZGNQSVGROPGZJH
|
7.5 | IC50 | 3 | — | |
BLQYVHBZHAISJM
|
7.5 | Ki | 54 | — | |
FFCFHBVSGILIJY
|
7.5 | Ki | 17 | — | |
GXSZEJJGRAAVEG
|
7.5 | IC50 | 3 | — | |
KUNZDWIFPOMUOX
|
7.5 | Ki | 36 | — | |
UGEJLCNSVIVALC
|
7.5 | Ki | 41 | — | |
UXQLMVSZSYZFID
|
7.5 | Ki | 12 | — | |
WINHZLLDWRZWRT
|
7.5 | Ki | 66 | — |