Target Details
| UniProt AC | P06213 |
|---|---|
| Gene Symbol | INSR |
| Protein Name | Insulin receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00757 (Furin-like) PF17870 (Insulin_TMD) PF07714 (PK_Tyr_Ser-Thr) PF01030 (Recep_L_domain) |
Summary
- Multi-target molecules 656
- Clinical molecules 33
- Avg pChEMBL 7.55
KEGG Pathways (23)
- AMPK signaling pathway
- Adherens junction
- Aldosterone-regulated sodium reabsorption
- Alzheimer disease
- Diabetic cardiomyopathy
- FoxO signaling pathway
- HIF-1 signaling pathway
- Hormone signaling
- Insulin resistance
- Insulin signaling pathway
- Longevity regulating pathway
- Longevity regulating pathway - multiple species
- MAPK signaling pathway
- Non-alcoholic fatty liver disease
- Ovarian steroidogenesis
- PI3K-Akt signaling pathway
- Phospholipase D signaling pathway
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of lipolysis in adipocytes
- Type II diabetes mellitus
- cGMP-PKG signaling pathway
- mTOR signaling pathway
Associated Diseases (4)
Active Molecules (656)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DPQSQXGBMAXUAP
|
6.7 | IC50 | 3 | — | |
RKWOVOVDWBRGQO
|
6.7 | Kd | 5 | — | |
YMVVZENKOZBFDW
|
6.7 | IC50 | 2 | — | |
AILRADAXUVEEIR
|
6.7 | IC50 | 75 | — | |
TYYJYNQSJRUHFJ
|
6.7 | IC50 | 3 | — | |
WTLGABJSLMBEHB
|
6.7 | IC50 | 2 | — | |
BIKYDWLMTPRSQL
|
6.7 | Ki | 50 | — | |
DJOJKIGNNDWGRS
|
6.7 | Ki | 13 | — | |
GZYCQQBRSRIFII
|
6.7 | IC50 | 7 | — | |
KNARVZUUCLIBGV
|
6.7 | Ki | 33 | — | |
QKKIWEILHCXECO
|
6.7 | IC50 | 24 | — | |
WINHZLLDWRZWRT
|
6.7 | Ki | 66 | — | |
XJSFDMGICAWQFS
|
6.7 | Ki | 60 | — | |
YRFQWNJZGSTUOR
|
6.7 | IC50 | 2 | — | |
ZVWRFVCNQOECJS
|
6.7 | Ki | 71 | — | |
FQUQLTHTCSOGBY
|
6.7 | IC50 | 3 | — | |
CXQHYVUVSFXTMY
|
6.7 | Kd | 154 | — | |
HAYYBYPASCDWEQ
|
6.7 | IC50 | 47 | — | |
KOZFSFOOLUUIGY
|
6.7 | IC50 | 26 | — | |
SEJGTFPOEJWEGG
|
6.7 | Kd | 149 | — | |
UNCWKKAXUDLWHL
|
6.7 | IC50 | 2 | — | |
TZQJLQWNUAZYJQ
|
6.7 | IC50 | 3 | — | |
WLTMYDRAYRGWMO
|
6.7 | IC50 | 5 | — | |
JUTMYSXKSLZJQM
|
6.6 | IC50 | 2 | — | |
KWVOXKDNAQPLPP
|
6.6 | IC50 | 2 | — | |
PRRFEHPXFCRKNK
|
6.6 | IC50 | 2 | — | |
WSTUJEXAPHIEIM
|
6.6 | IC50 | 10 | — | |
CPVCXTGQEFSNOQ
|
6.6 | IC50 | 2 | — | |
SISCSFVXUVITFJ
|
6.6 | IC50 | 2 | — | |
NEWALRCVHVFLBK
|
6.6 | IC50 | 2 | — | |
XFABGERDXKXSEQ
|
6.6 | IC50 | 2 | — | |
LVXQLMJEKSIZDV
|
6.6 | IC50 | 2 | — | |
FDVSOQRNTAPCHB
|
6.6 | Ki | 40 | — | |
GXJSLIOOPZRPEV
|
6.6 | Ki | 34 | — | |
NRZYTPAJGVTKIM
|
6.6 | Ki | 38 | — | |
ZLEPBLGJEZUDSL
|
6.6 | IC50 | 2 | — | |
DCQGBFHFVFACQU
|
6.6 | IC50 | 3 | — | |
KTEIFNKAUNYNJU
|
6.6 | IC50 | 114 | — | |
NWUSHDACDTZXCD
|
6.6 | IC50 | 2 | — | |
RDFZVFFSXWGAKR
|
6.6 | IC50 | 2 | — | |
UTNZTKXNTBTXTL
|
6.6 | IC50 | 2 | — | |
SWDUUFOEGXYQAO
|
6.6 | IC50 | 3 | — | |
UETYAVAIGWIDEO
|
6.6 | IC50 | 3 | — | |
XMKAFTZMVDNUII
|
6.6 | IC50 | 2 | — | |
RQDNRYSBNFWQCV
|
6.5 | IC50 | 3 | — | |
ZEURXJJLFFSRDT
|
6.5 | IC50 | 2 | — | |
QSLMZWGPJXKPBS
|
6.5 | IC50 | 3 | — | |
NRQSCGVAXSQZCR
|
6.5 | IC50 | 4 | — | |
GKQIKYWYJQQLLD
|
6.5 | IC50 | 3 | — | |
PLSQYACXDKUYFC
|
6.5 | IC50 | 3 | — |