Target Details
| UniProt AC | P06213 |
|---|---|
| Gene Symbol | INSR |
| Protein Name | Insulin receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00757 (Furin-like) PF17870 (Insulin_TMD) PF07714 (PK_Tyr_Ser-Thr) PF01030 (Recep_L_domain) |
Summary
- Multi-target molecules 656
- Clinical molecules 33
- Avg pChEMBL 7.55
KEGG Pathways (23)
- AMPK signaling pathway
- Adherens junction
- Aldosterone-regulated sodium reabsorption
- Alzheimer disease
- Diabetic cardiomyopathy
- FoxO signaling pathway
- HIF-1 signaling pathway
- Hormone signaling
- Insulin resistance
- Insulin signaling pathway
- Longevity regulating pathway
- Longevity regulating pathway - multiple species
- MAPK signaling pathway
- Non-alcoholic fatty liver disease
- Ovarian steroidogenesis
- PI3K-Akt signaling pathway
- Phospholipase D signaling pathway
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of lipolysis in adipocytes
- Type II diabetes mellitus
- cGMP-PKG signaling pathway
- mTOR signaling pathway
Associated Diseases (4)
Active Molecules (656)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MCCCQFAOMZMZKE
|
7.2 | Ki | 52 | — | |
OWRXHGAFWZFFCW
|
7.2 | Ki | 113 | — | |
BCSHRERPHLTPEE
|
7.2 | IC50 | 3 | — | |
ORFGUEWOGJKLFU
|
7.2 | IC50 | 2 | — | |
RTGPQVHYQAWJEV
|
7.2 | IC50 | 2 | — | |
RTQRIPALPGYRNN
|
7.2 | IC50 | 2 | — | |
HAFZQSVDZNBXHX
|
7.2 | IC50 | 2 | — | |
MNJPFSBAYJQZOE
|
7.2 | IC50 | 3 | — | |
NXKBBURYGABXCP
|
7.2 | IC50 | 2 | — | |
ZWVZORIKUNOTCS
|
7.1 | IC50 | 10 | Yes | |
FUGZYLOFWXVFQU
|
7.1 | IC50 | 3 | Yes | |
SCJMHNYQTKWNRD
|
7.1 | IC50 | 2 | — | |
YCGAVAFYTUFYPA
|
7.1 | IC50 | 6 | Yes | |
LBMWDLUJEOLXOE
|
7.1 | IC50 | 2 | — | |
CQFVDHNTTRWVQD
|
7.1 | Ki | 9 | — | |
QDCQSLLXPYSDTE
|
7.1 | IC50 | 2 | — | |
XKZQZMSAWVDRSP
|
7.1 | IC50 | 39 | Yes | |
BCSHRERPHLTPEE
|
7.1 | IC50 | 3 | — | |
DEBFWFAAIWZWSH
|
7.1 | IC50 | 3 | — | |
KJWZHCRQZUOQJR
|
7.1 | IC50 | 3 | — | |
IIFZHKOYTWEVOZ
|
7.0 | IC50 | 2 | — | |
RLDIJFHXXAQFAJ
|
7.0 | IC50 | 2 | — | |
AHLIOYKRAKANRB
|
7.0 | IC50 | 2 | — | |
GCDSDVNITVBCDW
|
7.0 | IC50 | 17 | — | |
YHWJHUBPWLCING
|
7.0 | IC50 | 3 | — | |
KJDKBIYPTUYYHT
|
7.0 | IC50 | 2 | — | |
MUAICZWSFWUFNA
|
7.0 | IC50 | 2 | — | |
VERWOWGGCGHDQE
|
7.0 | IC50 | 23 | — | |
JCTYSOVQZGLZOP
|
7.0 | IC50 | 2 | — | |
ASBGJVNBZBSENK
|
7.0 | IC50 | 2 | — | |
BCTIPSBBPQBXAG
|
7.0 | IC50 | 4 | — | |
BMTLGYPQYJNECV
|
7.0 | IC50 | 3 | — | |
BOJLJYRVWHJBLQ
|
7.0 | IC50 | 2 | — | |
CFIBXVQLBVNOHW
|
7.0 | Ki | 64 | — | |
GCACQFKGBBFZLV
|
7.0 | IC50 | 3 | — | |
GRXLBTDEMQIUOG
|
7.0 | IC50 | 3 | — | |
JGMJCQJURLCLJC
|
7.0 | IC50 | 2 | — | |
KUYIQVZTFYAICK
|
7.0 | IC50 | 2 | — | |
KYVIQYWGGPLPCH
|
7.0 | IC50 | 3 | — | |
LAVUQVGESJYCJA
|
7.0 | IC50 | 2 | — | |
NFKMFNBKEOQNPZ
|
7.0 | Ki | 43 | — | |
NQBOWNPIRYVPJI
|
7.0 | IC50 | 2 | — | |
OVDSPTSBIQCAIN
|
7.0 | IC50 | 7 | — | |
QRCUKJSISICWNH
|
7.0 | IC50 | 2 | — | |
QSNLBMCGRQUEPH
|
7.0 | IC50 | 2 | — | |
RNICSIBFPJOYHB
|
7.0 | IC50 | 2 | — | |
UOUIRSAMKHDQKN
|
7.0 | IC50 | 2 | — | |
WPHKIQPVPYJNAX
|
7.0 | Ki | 81 | — | |
XRMQCRQMFWASRC
|
7.0 | IC50 | 2 | — | |
YMIJUBCSOKSFRU
|
7.0 | Ki | 87 | — |