Target Details
| UniProt AC | P06213 |
|---|---|
| Gene Symbol | INSR |
| Protein Name | Insulin receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00757 (Furin-like) PF17870 (Insulin_TMD) PF07714 (PK_Tyr_Ser-Thr) PF01030 (Recep_L_domain) |
Summary
- Multi-target molecules 656
- Clinical molecules 33
- Avg pChEMBL 7.55
KEGG Pathways (23)
- AMPK signaling pathway
- Adherens junction
- Aldosterone-regulated sodium reabsorption
- Alzheimer disease
- Diabetic cardiomyopathy
- FoxO signaling pathway
- HIF-1 signaling pathway
- Hormone signaling
- Insulin resistance
- Insulin signaling pathway
- Longevity regulating pathway
- Longevity regulating pathway - multiple species
- MAPK signaling pathway
- Non-alcoholic fatty liver disease
- Ovarian steroidogenesis
- PI3K-Akt signaling pathway
- Phospholipase D signaling pathway
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of lipolysis in adipocytes
- Type II diabetes mellitus
- cGMP-PKG signaling pathway
- mTOR signaling pathway
Associated Diseases (4)
Active Molecules (656)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RNIDGDNODCTPSJ
|
8.3 | IC50 | 2 | — | |
CENVUXSKJJMKIU
|
8.3 | IC50 | 2 | — | |
ZCTVEBRXLFXVIK
|
8.3 | IC50 | 3 | — | |
MMJWRPJCZSSSNA
|
8.3 | IC50 | 2 | — | |
TWJHARJINSWCDD
|
8.2 | IC50 | 2 | — | |
CKZWESXBMQBAAD
|
8.2 | IC50 | 2 | — | |
IHRFTDHYCNWNFR
|
8.2 | IC50 | 3 | — | |
JKEFKVZKYKUDGL
|
8.2 | IC50 | 2 | — | |
RWASATDZTQIHPA
|
8.2 | IC50 | 2 | — | |
UZPCCONBZIFGNY
|
8.2 | IC50 | 2 | — | |
FLEAYYMORDPWAJ
|
8.2 | Ki | 90 | — | |
MCHOTIIDAJHLED
|
8.2 | IC50 | 5 | Yes | |
PKCDDUHJAFVJJB
|
8.2 | Ki | 13 | — | |
MWKSRKSEWLRPBL
|
8.2 | Kd | 1075 | — | |
SKFDSQFYKXYVPS
|
8.2 | IC50 | 9 | Yes | |
XMJRRSFVUFDVMT
|
8.2 | IC50 | 2 | — | |
HSCSBODZXPHWFM
|
8.1 | IC50 | 2 | — | |
AWKVKBJHESFTRA
|
8.1 | IC50 | 2 | — | |
GDRLJBDXWDATLA
|
8.1 | IC50 | 13 | — | |
WDUXPXHDIYWLHP
|
8.1 | IC50 | 3 | — | |
IEPKZTQXMCCRFJ
|
8.1 | IC50 | 4 | — | |
BHLTVGNUTOSHBD
|
8.0 | IC50 | 3 | — | |
GANNLFTUWFAJIC
|
8.0 | IC50 | 2 | — | |
KYTDVMCLOSUQEH
|
8.0 | IC50 | 2 | — | |
LTIMJKHVDDEVSP
|
8.0 | IC50 | 2 | — | |
SBLMCLDRWJNEJK
|
8.0 | IC50 | 17 | — | |
SFPSNTOXJBCKGE
|
8.0 | IC50 | 2 | — | |
TWFGYFUYNRUBKC
|
8.0 | IC50 | 2 | — | |
XZAWNQULYQTFPH
|
8.0 | IC50 | 2 | — | |
ZGFXRISUXOJOLE
|
8.0 | IC50 | 2 | — | |
ZNLCRBCFRLCIFE
|
8.0 | IC50 | 4 | Yes | |
HAPYOEZQKCQEPE
|
8.0 | IC50 | 2 | — | |
OIPVNLQCUGTYJW
|
8.0 | IC50 | 2 | — | |
QVMUQQQYQHYSBY
|
8.0 | IC50 | 2 | — | |
QDJZMRPVQLAGDJ
|
7.9 | IC50 | 2 | — | |
ZNWUBQNDIPEESB
|
7.9 | IC50 | 2 | — | |
XGZORHKVFKUMAV
|
7.9 | IC50 | 4 | — | |
IDRQGRCXNROMMS
|
7.9 | IC50 | 3 | — | |
COMVVKFCZPWGAV
|
7.8 | IC50 | 2 | — | |
XRVFEWYOEIYZGB
|
7.8 | IC50 | 3 | — | |
SIVMXJQFCAHOMI
|
7.8 | IC50 | 2 | — | |
GQGMUKOYILWOIQ
|
7.8 | Ki | 25 | — | |
WXMYXQYBHNGGNH
|
7.8 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
7.8 | IC50 | 408 | — | |
YQXBTLYMIWQFAN
|
7.7 | IC50 | 2 | — | |
LUZLOIYOYLEIRH
|
7.7 | IC50 | 2 | — | |
AEFLOLLJJAKGQJ
|
7.7 | IC50 | 2 | — | |
AKHXBNQXYOJHSZ
|
7.7 | IC50 | 2 | — | |
HAGKVAUHAUZMBY
|
7.7 | IC50 | 2 | — | |
LLYDHPYAMNHNIM
|
7.7 | IC50 | 2 | — |