Target Details
| UniProt AC | P06213 |
|---|---|
| Gene Symbol | INSR |
| Protein Name | Insulin receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00757 (Furin-like) PF17870 (Insulin_TMD) PF07714 (PK_Tyr_Ser-Thr) PF01030 (Recep_L_domain) |
Summary
- Multi-target molecules 656
- Clinical molecules 33
- Avg pChEMBL 7.55
KEGG Pathways (23)
- AMPK signaling pathway
- Adherens junction
- Aldosterone-regulated sodium reabsorption
- Alzheimer disease
- Diabetic cardiomyopathy
- FoxO signaling pathway
- HIF-1 signaling pathway
- Hormone signaling
- Insulin resistance
- Insulin signaling pathway
- Longevity regulating pathway
- Longevity regulating pathway - multiple species
- MAPK signaling pathway
- Non-alcoholic fatty liver disease
- Ovarian steroidogenesis
- PI3K-Akt signaling pathway
- Phospholipase D signaling pathway
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of lipolysis in adipocytes
- Type II diabetes mellitus
- cGMP-PKG signaling pathway
- mTOR signaling pathway
Associated Diseases (4)
Active Molecules (656)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LWVQAFSEKOOOAI
|
9.4 | IC50 | 2 | — | |
OPSIJGYSVYFFGS
|
9.4 | IC50 | 2 | — | |
OYQMWWVIYBSJLB
|
9.4 | IC50 | 2 | — | |
UVJDZKBPVPTIRA
|
9.4 | IC50 | 2 | — | |
YRLINYQMYNEFJG
|
9.4 | IC50 | 2 | — | |
GLSBPQXKUMSIMB
|
9.4 | IC50 | 2 | — | |
HUHCYTMKDOFWSG
|
9.4 | IC50 | 2 | — | |
LDYDMNAZFRCWNR
|
9.4 | IC50 | 2 | — | |
RKWGNTHTPQXXQN
|
9.4 | IC50 | 2 | — | |
RZLRBIAISAXDHA
|
9.4 | IC50 | 2 | — | |
FLTJPMCKNUNPRH
|
9.4 | IC50 | 3 | — | |
QJWZXYIVWQUAAO
|
9.4 | IC50 | 2 | — | |
KVFQSNCDMQJZPD
|
9.4 | IC50 | 2 | — | |
IQLMHUMYHUUAQQ
|
9.4 | IC50 | 2 | — | |
JGLSPBGRSLPKAQ
|
9.3 | IC50 | 2 | — | |
QJSZKBYCIGDBBS
|
9.3 | IC50 | 2 | — | |
FHMWNSNIIZHZPJ
|
9.3 | IC50 | 2 | — | |
PTPQXKBVULYOLN
|
9.3 | IC50 | 2 | — | |
IAIFZADOAVHXEL
|
9.3 | IC50 | 2 | — | |
MUAJURKWULOSJG
|
9.3 | IC50 | 2 | — | |
ZZJJJCFYECEHNN
|
9.3 | IC50 | 2 | — | |
CWSQJENYIZLGER
|
9.3 | IC50 | 2 | — | |
YDCSUBLUYMXIOG
|
9.2 | IC50 | 2 | — | |
NXJDOMZWUPMZFE
|
9.2 | IC50 | 2 | — | |
RVIMGPNKJMIZJW
|
9.2 | IC50 | 2 | — | |
RNRVBUQQZHOCBU
|
9.2 | IC50 | 2 | — | |
BHOLGBKCKRPFPA
|
9.2 | IC50 | 2 | — | |
GWVCRFPHEQXQJR
|
9.2 | IC50 | 2 | — | |
DMQJVMSMJXCZOS
|
9.2 | IC50 | 2 | — | |
ALHWHMNSEAIFMC
|
9.2 | IC50 | 2 | — | |
YEPYKAAAXUCSMP
|
9.1 | IC50 | 2 | — | |
QWPNPMFVZNBPEA
|
9.1 | IC50 | 2 | — | |
VVXWJQWOEIYIHP
|
9.1 | IC50 | 2 | — | |
VZVLZJITGHRMBT
|
9.1 | IC50 | 2 | — | |
BAIRSNTWXBQKHG
|
9.1 | IC50 | 2 | — | |
CPFRXSGEPFEUFG
|
9.1 | IC50 | 2 | — | |
PCUMDMKSEZJNLA
|
9.1 | IC50 | 2 | — | |
ZSIGECCEZMACTJ
|
9.1 | IC50 | 2 | — | |
YQWFNFUEJRELJX
|
9.1 | IC50 | 2 | — | |
CZHQIACJGGUSQU
|
9.1 | IC50 | 2 | — | |
DLKUDUSWHQNMDW
|
9.1 | IC50 | 2 | — | |
LEVAPGLCIYCDDH
|
9.1 | IC50 | 3 | — | |
SBDSSXKUILJHSM
|
9.1 | IC50 | 2 | — | |
LGLJGJQDMXPFHU
|
9.0 | IC50 | 2 | — | |
SFBCVPDTLHGKAL
|
9.0 | IC50 | 2 | — | |
FENCVPRSVOEMHI
|
9.0 | IC50 | 2 | — | |
IILFQZAVZNEIKL
|
9.0 | IC50 | 2 | — | |
JKGUWRSWKIHSTP
|
9.0 | IC50 | 2 | — | |
KCFKHBXTNWBJGZ
|
9.0 | IC50 | 2 | — | |
KCZLTVJTTQQVRB
|
9.0 | IC50 | 2 | — |