Target Details
| UniProt AC | P06213 |
|---|---|
| Gene Symbol | INSR |
| Protein Name | Insulin receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00757 (Furin-like) PF17870 (Insulin_TMD) PF07714 (PK_Tyr_Ser-Thr) PF01030 (Recep_L_domain) |
Summary
- Multi-target molecules 656
- Clinical molecules 33
- Avg pChEMBL 7.55
KEGG Pathways (23)
- AMPK signaling pathway
- Adherens junction
- Aldosterone-regulated sodium reabsorption
- Alzheimer disease
- Diabetic cardiomyopathy
- FoxO signaling pathway
- HIF-1 signaling pathway
- Hormone signaling
- Insulin resistance
- Insulin signaling pathway
- Longevity regulating pathway
- Longevity regulating pathway - multiple species
- MAPK signaling pathway
- Non-alcoholic fatty liver disease
- Ovarian steroidogenesis
- PI3K-Akt signaling pathway
- Phospholipase D signaling pathway
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of lipolysis in adipocytes
- Type II diabetes mellitus
- cGMP-PKG signaling pathway
- mTOR signaling pathway
Associated Diseases (4)
Active Molecules (656)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ACRVYPAOYVTCDU
|
9.7 | IC50 | 2 | — | |
JBTWMLFMVHUXEX
|
9.7 | IC50 | 2 | — | |
JHRKWSGMWPZSKV
|
9.7 | IC50 | 2 | — | |
UCLVRCLUQFRAIO
|
9.7 | IC50 | 2 | — | |
VHIBZYACLHIGAD
|
9.7 | IC50 | 2 | — | |
KVKJFFOOZLJLIE
|
9.7 | IC50 | 2 | — | |
RPGJMEAIZVOJBL
|
9.7 | IC50 | 2 | — | |
SXIJONAFQCNJBP
|
9.7 | IC50 | 2 | — | |
XMFQIFQGGPJVOC
|
9.7 | IC50 | 2 | — | |
KPIGJFWGDBIKGO
|
9.6 | IC50 | 2 | — | |
KUHKYMBXFNXFAZ
|
9.6 | IC50 | 2 | — | |
LNCMGLWONSBOCY
|
9.6 | IC50 | 2 | — | |
XYXCIYOUOPDGOR
|
9.6 | IC50 | 2 | — | |
YQJRFYXDFBSSKL
|
9.6 | IC50 | 2 | — | |
DLPSKFBVVGFFPU
|
9.6 | IC50 | 2 | — | |
DUJYZAINCFXLIR
|
9.6 | IC50 | 2 | — | |
PTCFPPCYMCVXEU
|
9.6 | IC50 | 2 | — | |
BOHBMNHGQQYWHB
|
9.6 | IC50 | 2 | — | |
GOFWFAUOCPWWFW
|
9.6 | IC50 | 2 | — | |
QSPDKYVHOBOPDX
|
9.6 | IC50 | 2 | — | |
PVNIKRFRAZTHDL
|
9.6 | IC50 | 2 | — | |
RXAVSKHCIFNSSC
|
9.6 | IC50 | 2 | — | |
UGRLUSFRPRDZAG
|
9.6 | IC50 | 2 | — | |
YOOMZWXNMOLJNG
|
9.6 | IC50 | 2 | — | |
GEGBULDNFJOMON
|
9.6 | IC50 | 2 | — | |
UORNJEUJPWRNCR
|
9.6 | IC50 | 2 | — | |
FFVJVKCJYRSTDW
|
9.6 | IC50 | 2 | — | |
HPUNVQVUHWPBNZ
|
9.6 | IC50 | 2 | — | |
OBYITYSRDPDKFQ
|
9.6 | IC50 | 2 | — | |
JTKKDJAXGOCIOK
|
9.5 | IC50 | 2 | — | |
CGKVOZLVEYQYNI
|
9.5 | IC50 | 2 | — | |
DEOQOEQPXFZCOT
|
9.5 | IC50 | 2 | — | |
PRSCIAZLYQXCHO
|
9.5 | IC50 | 2 | — | |
QGYNHTKWDSQMIE
|
9.5 | IC50 | 2 | — | |
VEYYJQOJUNVXRV
|
9.5 | IC50 | 2 | — | |
VKXWYVXZTMFYQA
|
9.5 | IC50 | 2 | — | |
AZXRBWUQPGETKR
|
9.5 | IC50 | 2 | — | |
FCAIWXLANPUWBS
|
9.5 | IC50 | 2 | — | |
SKGYZKPSLOLJCF
|
9.5 | IC50 | 2 | — | |
ARCZPWVFAOSJRU
|
9.5 | IC50 | 2 | — | |
RHENXWJKGMRHEV
|
9.5 | IC50 | 2 | — | |
WIGMQNAICQDORZ
|
9.5 | IC50 | 2 | — | |
XKOGTAJAHIXUKP
|
9.5 | IC50 | 2 | — | |
FNNJMLPKSOMUFS
|
9.4 | IC50 | 2 | — | |
ISJBELANSICSFT
|
9.4 | IC50 | 2 | — | |
DXWPAGJGSYGDPW
|
9.4 | IC50 | 2 | — | |
RIVKOYDUUSWKNV
|
9.4 | IC50 | 2 | — | |
YPFRABRKNDFAON
|
9.4 | IC50 | 2 | — | |
ZPBKIKCGBBLRFM
|
9.4 | IC50 | 2 | — | |
JCAOTPBZOINVCN
|
9.4 | IC50 | 2 | — |