Target Details
| UniProt AC | P06213 |
|---|---|
| Gene Symbol | INSR |
| Protein Name | Insulin receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00757 (Furin-like) PF17870 (Insulin_TMD) PF07714 (PK_Tyr_Ser-Thr) PF01030 (Recep_L_domain) |
Summary
- Multi-target molecules 656
- Clinical molecules 33
- Avg pChEMBL 7.55
KEGG Pathways (23)
- AMPK signaling pathway
- Adherens junction
- Aldosterone-regulated sodium reabsorption
- Alzheimer disease
- Diabetic cardiomyopathy
- FoxO signaling pathway
- HIF-1 signaling pathway
- Hormone signaling
- Insulin resistance
- Insulin signaling pathway
- Longevity regulating pathway
- Longevity regulating pathway - multiple species
- MAPK signaling pathway
- Non-alcoholic fatty liver disease
- Ovarian steroidogenesis
- PI3K-Akt signaling pathway
- Phospholipase D signaling pathway
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of lipolysis in adipocytes
- Type II diabetes mellitus
- cGMP-PKG signaling pathway
- mTOR signaling pathway
Associated Diseases (4)
Active Molecules (656)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XIQAFZIFYBEQQW
|
6.4 | IC50 | 3 | — | |
XQCYJMDRMXBJIP
|
6.4 | IC50 | 2 | — | |
YJRZCHGBUZZOPZ
|
6.4 | IC50 | 2 | — | |
YRUIXESBPXQWOD
|
6.4 | IC50 | 3 | — | |
YYLKKYCXAOBSRM
|
6.4 | Kd | 191 | — | |
ACYSIZUFQATBIE
|
6.4 | IC50 | 2 | — | |
FUGPVNRCNPSEKE
|
6.4 | IC50 | 2 | — | |
UIFHDCIICKTEAL
|
6.4 | IC50 | 3 | — | |
YQPHBBQBBMIYLO
|
6.4 | IC50 | 6 | Yes | |
ADAQBVKANMBBGO
|
6.4 | IC50 | 2 | — | |
DOXJXXFTEWRETQ
|
6.4 | IC50 | 4 | Yes | |
LSEPNYIMWPZFLK
|
6.4 | IC50 | 2 | — | |
PIBITIKJRIGPID
|
6.4 | IC50 | 3 | — | |
QXIOZIFTPMAING
|
6.4 | IC50 | 17 | — | |
UYBILPBKQDAXTL
|
6.4 | IC50 | 2 | — | |
AFTBNZZMNUUEFO
|
6.4 | IC50 | 7 | — | |
GMAZSCDBFSDVRI
|
6.4 | IC50 | 3 | — | |
LIWMTOPLJLFZKX
|
6.4 | IC50 | 2 | — | |
UMBIRSZUCJNBHB
|
6.4 | IC50 | 18 | — | |
ACYSIZUFQATBIE
|
6.4 | IC50 | 2 | — | |
CDTMQKLFPXZZMW
|
6.3 | IC50 | 2 | — | |
HXYIPFOMCPLBAX
|
6.3 | IC50 | 3 | — | |
SAHMNRNXZPYQHB
|
6.3 | IC50 | 3 | — | |
VJWLMBVALMQEMA
|
6.3 | IC50 | 3 | — | |
XDTMZEAHVJVNJG
|
6.3 | IC50 | 2 | — | |
ZIPMVFDKNBGKAT
|
6.3 | IC50 | 3 | — | |
GGJPKPHOWZDYAP
|
6.3 | IC50 | 2 | — | |
LYOCYPVMXHFJAK
|
6.3 | IC50 | 2 | — | |
NBMMGFKSCSDKBQ
|
6.3 | IC50 | 2 | — | |
NMJMRSQTDLRCRQ
|
6.3 | IC50 | 7 | — | |
IXXBKMMVWWTOCC
|
6.3 | IC50 | 2 | — | |
NBGLUPSFCNIDOO
|
6.3 | IC50 | 2 | — | |
WJBWDHCGIKSMMX
|
6.3 | IC50 | 2 | — | |
ZTKZGNHMDMISHE
|
6.3 | IC50 | 3 | — | |
QMDSNSHMWIVCND
|
6.3 | IC50 | 2 | — | |
ZKSMNJVVPOADIE
|
6.3 | IC50 | 3 | — | |
ADMFLILDQJSEIK
|
6.3 | Ki | 72 | — | |
CQBBMNXXVMOFCA
|
6.3 | Ki | 39 | — | |
CZQVOIDVDAVDFW
|
6.3 | Ki | 18 | — | |
FXQWJULRETZHHW
|
6.3 | Ki | 14 | — | |
GDYZFFBMSBDTAA
|
6.3 | Ki | 60 | — | |
HKZKELVPGXJIMW
|
6.3 | Ki | 41 | — | |
KRIUNPBAQZGFQA
|
6.3 | Ki | 76 | — | |
MQRDVGBWWVWMEN
|
6.3 | Ki | 47 | — | |
MZDKLVOWGIOKTN
|
6.3 | Ki | 80 | — | |
NRSGWEVTVGZDFC
|
6.3 | Ki | 50 | — | |
PGXXNNIGDDGRPV
|
6.3 | IC50 | 2 | — | |
RTDSHUGNRVXRHN
|
6.3 | Ki | 51 | — | |
UJBJWYNPUOLFIZ
|
6.3 | IC50 | 49 | — | |
UOVCGJXDGOGOCZ
|
6.3 | Ki | 59 | — |