Target Details
| UniProt AC | P06213 |
|---|---|
| Gene Symbol | INSR |
| Protein Name | Insulin receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00757 (Furin-like) PF17870 (Insulin_TMD) PF07714 (PK_Tyr_Ser-Thr) PF01030 (Recep_L_domain) |
Summary
- Multi-target molecules 656
- Clinical molecules 33
- Avg pChEMBL 7.55
KEGG Pathways (23)
- AMPK signaling pathway
- Adherens junction
- Aldosterone-regulated sodium reabsorption
- Alzheimer disease
- Diabetic cardiomyopathy
- FoxO signaling pathway
- HIF-1 signaling pathway
- Hormone signaling
- Insulin resistance
- Insulin signaling pathway
- Longevity regulating pathway
- Longevity regulating pathway - multiple species
- MAPK signaling pathway
- Non-alcoholic fatty liver disease
- Ovarian steroidogenesis
- PI3K-Akt signaling pathway
- Phospholipase D signaling pathway
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of lipolysis in adipocytes
- Type II diabetes mellitus
- cGMP-PKG signaling pathway
- mTOR signaling pathway
Associated Diseases (4)
Active Molecules (656)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DWLZYJOAPBAXQM
|
10.3 | IC50 | 2 | — | |
FLBQTCODPBJFTD
|
10.3 | IC50 | 2 | — | |
DANRHRCSZZGXLP
|
10.1 | IC50 | 2 | — | |
KUXYUFHYERAGDG
|
10.1 | IC50 | 2 | — | |
WFXSEBKHQBTMMS
|
10.1 | IC50 | 2 | — | |
ZEPVDOIWFVBKOM
|
10.1 | IC50 | 2 | — | |
GBTTYDWBVFNAEA
|
10.1 | IC50 | 2 | — | |
MRNCAMTZMKCLDO
|
10.1 | IC50 | 2 | — | |
NWCSJPOCTCBOEW
|
10.1 | IC50 | 2 | — | |
DKWOGWIUVLBDHC
|
10.0 | IC50 | 2 | — | |
DRYYTRLZCKWIGZ
|
10.0 | IC50 | 2 | — | |
KZXBXGNMGTZACU
|
10.0 | IC50 | 2 | — | |
URABRDOUNMLPLA
|
10.0 | IC50 | 2 | — | |
KXDLJCXLOFTQOJ
|
10.0 | IC50 | 2 | — | |
SOUDXNZKWYTFFW
|
10.0 | IC50 | 2 | — | |
PAEPNROAXKXFOQ
|
9.9 | IC50 | 2 | — | |
JRKWDAZGBOBRPT
|
9.9 | IC50 | 2 | — | |
MRTQXPYBEKCXAN
|
9.9 | IC50 | 2 | — | |
MZRCFUHXHKAGCK
|
9.9 | IC50 | 2 | — | |
NJBNQVCQKINYLS
|
9.9 | IC50 | 2 | — | |
OWPFZNYKPFPFIT
|
9.9 | IC50 | 2 | — | |
YOFGUEQIPVDBEL
|
9.9 | IC50 | 2 | — | |
GLLLAYKUVMFJER
|
9.8 | IC50 | 2 | — | |
GMHBLFNISBWXBO
|
9.8 | IC50 | 2 | — | |
SDTDXGMQPJHODR
|
9.8 | IC50 | 2 | — | |
WSEOWNBBPGNYRJ
|
9.8 | IC50 | 2 | — | |
XYBRNZWRDMIYFT
|
9.8 | IC50 | 2 | — | |
BKYSHTIOCHNDDH
|
9.8 | IC50 | 2 | — | |
CNBMRJSFULHWLZ
|
9.8 | IC50 | 2 | — | |
FCGZIEABISYQOO
|
9.8 | IC50 | 2 | — | |
CLXCUJAIQNKPCW
|
9.8 | IC50 | 2 | — | |
DEUXRKZJLFSYAO
|
9.8 | IC50 | 2 | — | |
IYYUJNJRKWXTJJ
|
9.8 | IC50 | 2 | — | |
NDVDUHONBQZAGA
|
9.8 | IC50 | 2 | — | |
OSGQGIINHNRMCL
|
9.8 | IC50 | 2 | — | |
RXLGVLBKICWANA
|
9.8 | IC50 | 2 | — | |
SAJTWQRLZVYSCP
|
9.8 | IC50 | 2 | — | |
UHHADNYIBMJTNI
|
9.8 | IC50 | 2 | — | |
VJSMYRLRQBWBQP
|
9.8 | IC50 | 2 | — | |
HCMFOVBYPFSDST
|
9.8 | IC50 | 2 | — | |
IEFXGIIDRDRIGF
|
9.8 | IC50 | 2 | — | |
IEMCBHBTNFUENC
|
9.8 | IC50 | 2 | — | |
OPYZOEXGCQPJNO
|
9.8 | IC50 | 2 | — | |
RWSCTJGHFHKJNJ
|
9.8 | IC50 | 2 | — | |
IBFTXGLRFZFDGT
|
9.7 | IC50 | 2 | — | |
IDUFXVFDCDFZDE
|
9.7 | IC50 | 2 | — | |
QSOSQIVFCJZEIL
|
9.7 | IC50 | 2 | — | |
UBDSRPCDONKGEF
|
9.7 | IC50 | 2 | — | |
DXLDXBDJHXQCCM
|
9.7 | IC50 | 2 | — | |
UKOMEKAHPLDSQG
|
9.7 | IC50 | 2 | — |