Target Details
UniProt ACP05981
Gene SymbolHPN
Protein NameSerine protease hepsin
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF09272 (Hepsin-SRCR) PF00089 (Trypsin)
Summary
  • Multi-target molecules 113
  • Clinical molecules 1
  • Avg pChEMBL 7.91
KEGG Pathways (1)
Top Co-occurrence Targets
Active Molecules (113)
InChIKey pChEMBL Type Targets Clinical
LNIRCTXHOVOSQG 8.2 IC50 3
PLLBBBICXMICNE 8.1 IC50 4
WKJNTWXQNNBXRN 8.1 IC50 2
ULIOUSXOKNOZQV 8.1 IC50 2
GWIRLHLNQLEUAV 8.1 Ki 3
ZQAJCRKPCMIAGU 8.1 IC50 2
NQUYPPYJOZKUFP 8.0 IC50 2
TVPUCYVDZLCUFP 8.0 IC50 2
IWSNQHXPYYMOLJ 8.0 IC50 2
MZLDHCSWGXPGJS 7.9 IC50 2
DQKGGUJIFZQGEB 7.8 IC50 3
RFDXBWAKPXTPCV 7.8 IC50 3
GEHOIKOYROYGLS 7.8 IC50 2
CMECINVDWRULPU 7.7 IC50 3
QGHPTZNADRNLAZ 7.7 IC50 2
ZOXIMPKMBVMIOP 7.7 IC50 2
NDQHQXALHKXAMC 7.7 IC50 2
GIZRMCORNKTMDA 7.6 IC50 2
FRENLDXJNSJMFU 7.5 IC50 3
WQDFAUJSOUQVHN 7.4 IC50 3
UPDFOAXKIVEQLH 7.4 IC50 2
GDBQQVLCIARPGH 7.2 Ki 10
OLNJKAXRBXUBTB 7.2 Ki 10 Yes
MBBPFTAWIJCEBL 7.2 Ki 3
GAVRMVQHHVMXFD 7.1 Ki 11
VDHFUZQXRACOII 7.0 Ki 2
CMQOQSPVFQTXTQ 7.0 Ki 4
VXVYXKAPTSJLCT 7.0 Ki 4
SKCJIIRKAVOSJL 7.0 Ki 2
GYXAJVPFFILTAV 7.0 Ki 2
WRVPVQAIXXARDJ 6.9 Ki 2
BVJKSLJMTUHQJM 6.9 Ki 2
MQTZNXMJQAAJDM 6.9 IC50 2
NNOFPIZGQIFDSZ 6.9 IC50 3
YHSFSXZVHUXTQX 6.7 Ki 2
HINXTEQWTTZJOH 6.7 Ki 7
VIPGDRKEADGMFI 6.7 Ki 2
NUZWLKWWNNJHPT 6.6 IC50 2
SIHSWLYSGZGJPP 6.6 Ki 2
VUNXKPNZAAYJKP 6.6 Ki 2
GFZNRMYFECIHSP 6.6 Ki 2
YVXIHFMTTRAGON 6.6 Ki 2
WPXVPKNQHQDFKA 6.5 Ki 2
JHARRMAYSVPENO 6.5 Ki 4
XBTBFQPWQHBKEV 6.4 Ki 2
YKGYIDJEEQRWQH 6.4 IC50 6
DDDBXZXECGEQRK 6.4 Ki 2
PHVFHKZPZJRDRJ 6.4 Ki 5
PIFQUSTVOQWPJQ 6.3 IC50 2
GBFNBYMSXRCRBZ 6.3 Ki 7
2D structure