Target Details
UniProt ACP05981
Gene SymbolHPN
Protein NameSerine protease hepsin
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF09272 (Hepsin-SRCR) PF00089 (Trypsin)
Summary
  • Multi-target molecules 113
  • Clinical molecules 1
  • Avg pChEMBL 7.91
KEGG Pathways (1)
Top Co-occurrence Targets
Active Molecules (113)
InChIKey pChEMBL Type Targets Clinical
ZHIKDBGWXAAPBG 10.1 IC50 3
WQISNVQCRKRHME 10.1 Ki 4
BLOFNYQHKSGSGE 9.8 Ki 3
NEQGCINBAXAQKD 9.8 IC50 5
GBWLZSRRLJETHI 9.7 IC50 5
BSCYVKJQDUSMFJ 9.7 Ki 3
WKFXBFMYZUNDEO 9.7 Ki 3
MMCZPBUBUPXIQM 9.6 Ki 4
RETMNWIAJUVWLF 9.6 Ki 3
RJBLHAMXODQZMM 9.5 IC50 4
LNFLFMVSXZPRHU 9.5 Ki 3
MDTKEYLCTKYBSK 9.4 IC50 4
QNGSZDJLWYVTQN 9.4 Ki 3
CNVNITMLGKDQQY 9.3 Ki 3
RIMDWLGGSDTBKR 9.3 IC50 2
MQQNFDZXWVTQEH 9.3 Ki 11
QQRQFIXRVWJLNT 9.3 Ki 10
AIAPZNJOJFJSQR 9.3 IC50 4
UNOVDKDICJRWRT 9.3 Ki 3
PFSNIQDNVQKULM 9.2 Ki 3
CFSDWWHMXFUPKB 9.2 Ki 3
DIOWGKUHSWDAQR 9.2 Ki 3
QCZLVVCFUACPGA 9.2 Ki 3
QHJAGEUQNNACSP 9.2 IC50 2
VFNBZASFQVJNJZ 9.2 Ki 3
DVZQOTUGXDAQNJ 9.2 Ki 3
SVOXYTTZYOSESO 9.2 Ki 4
ZLIIZOMJAUACIT 9.2 IC50 4
ZTZVSJUJOHEBFJ 9.0 IC50 4
PIYDBRKFQAMHCU 9.0 IC50 3
JRNGHBUUFQDBPT 9.0 Ki 8
RTSUFXOZXIDYFZ 9.0 Ki 5
AGLYIVQPVAYVMN 8.9 Ki 3
PHPJWSFXNNRMES 8.9 Ki 3
ZRJSFZXXCBTZHR 8.8 Ki 3
LOJOAZJDEFCKLF 8.8 IC50 3
ZWJVSNFLVMBMRD 8.7 IC50 2
KJLKBVQGEXTILS 8.7 Ki 3
WWUOOSJKTRFWDJ 8.6 Ki 3
AIAPZNJOJFJSQR 8.6 IC50 4
YXFPBFNFMATBRQ 8.5 Ki 4
VAHZBDOLKHNQEE 8.5 Ki 4
JTHVOFMYRRNGPA 8.4 Ki 3
HENHNGFKMLDXRP 8.4 Ki 3
CWPABYGTEGMLDD 8.3 IC50 3
BVIZJIXKCBABFU 8.3 IC50 4
QKWNZGZXTOQLON 8.2 IC50 2
XASIMHXSUQUHLV 8.2 Ki 7
KULBLQGJDWZVDS 8.2 IC50 2
NEDJZMSZNJMQAV 8.2 IC50 2
2D structure