Target Details
| UniProt AC | P05771 |
|---|---|
| Gene Symbol | PRKCB |
| Protein Name | Protein kinase C beta type |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF00168 (C2) PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 457
- Clinical molecules 133
- Avg pChEMBL 7.4
KEGG Pathways (73)
- AGE-RAGE signaling pathway in diabetic complications
- African trypanosomiasis
- Aldosterone synthesis and secretion
- Aldosterone-regulated sodium reabsorption
- Amoebiasis
- Amphetamine addiction
- B cell receptor signaling pathway
- Calcium signaling pathway
- Carbohydrate digestion and absorption
- Chemical carcinogenesis - receptor activation
- Chemokine signaling pathway
- Choline metabolism in cancer
- Cholinergic synapse
- Circadian entrainment
- Coronavirus disease - COVID-19
- Diabetic cardiomyopathy
- Dopaminergic synapse
- EGFR tyrosine kinase inhibitor resistance
- Endocrine and other factor-regulated calcium reabsorption
- ErbB signaling pathway
- Fc gamma R-mediated phagocytosis
- Focal adhesion
- GABAergic synapse
- Gap junction
- Gastric acid secretion
- Glioma
- Glutamatergic synapse
- GnRH secretion
- GnRH signaling pathway
- Growth hormone synthesis, secretion and action
- HIF-1 signaling pathway
- Hepatitis B
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- IgSF CAM signaling
- Inflammatory mediator regulation of TRP channels
- Influenza A
- Insulin resistance
- Insulin secretion
- Leishmaniasis
- Leukocyte transendothelial migration
- Long-term depression
- Long-term potentiation
- MAPK signaling pathway
- Melanogenesis
- MicroRNAs in cancer
- Morphine addiction
- NF-kappa B signaling pathway
- Natural killer cell mediated cytotoxicity
- Neuroactive ligand signaling
- Neutrophil extracellular trap formation
- Non-small cell lung cancer
- Oxytocin signaling pathway
- Pancreatic secretion
- Parathyroid hormone synthesis, secretion and action
- Pathways in cancer
- Pathways of neurodegeneration - multiple diseases
- Phosphatidylinositol signaling system
- Proteoglycans in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Retrograde endocannabinoid signaling
- Salivary secretion
- Serotonergic synapse
- Sphingolipid signaling pathway
- Spinocerebellar ataxia
- Thyroid hormone signaling pathway
- Thyroid hormone synthesis
- VEGF signaling pathway
- Vascular smooth muscle contraction
- Wnt signaling pathway
- mTOR signaling pathway
Active Molecules (457)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BMBIKZHGTPMMMM
|
6.3 | IC50 | 14 | — | |
CPRVBHBRBVVLHL
|
6.3 | IC50 | 11 | — | |
ATBAETXFFCOZOY
|
6.3 | IC50 | 39 | — | |
CCRCRSXDKXZDGK
|
6.3 | IC50 | 12 | Yes | |
JSPAUBUYPPZXSG
|
6.3 | Ki | 17 | Yes | |
ORNADCNXUPZOQN
|
6.3 | IC50 | 15 | — | |
OYPYXQXNEBSSGB
|
6.3 | Ki | 8 | Yes | |
NEGCBIBMPAHBIM
|
6.3 | IC50 | 12 | Yes | |
BAQFZMFDZMQJAM
|
6.2 | IC50 | 12 | Yes | |
HHSIUHRARDLCPM
|
6.2 | IC50 | 5 | Yes | |
TXBFOGDMTCNBBT
|
6.2 | IC50 | 12 | Yes | |
PEHFMYWGWHPKOC
|
6.2 | IC50 | 3 | — | |
PXONMVAMARNSJO
|
6.2 | Ki | 4 | — | |
ORVUCMUEXPKXML
|
6.2 | IC50 | 3 | — | |
QQKKPWJFHBFCTH
|
6.2 | IC50 | 10 | Yes | |
TWUWFRLZDWDJLT
|
6.2 | Ki | 10 | Yes | |
ZUKHVOLIPVGCHQ
|
6.2 | Ki | 10 | Yes | |
MVQGUYKZTHVOEH
|
6.2 | Ki | 8 | Yes | |
HLXIFVDYTGEUJV
|
6.2 | IC50 | 15 | Yes | |
QRBLWZIADYBYNA
|
6.2 | IC50 | 5 | — | |
KPJDEGAKXAUVAC
|
6.2 | Ki | 15 | Yes | |
VLUGUCDUHZVABE
|
6.2 | IC50 | 6 | — | |
WQSCDMQTCWOCID
|
6.2 | IC50 | 2 | — | |
XYUFCXJZFZPEJD
|
6.2 | IC50 | 5 | — | |
XYUFCXJZFZPEJD
|
6.2 | IC50 | 4 | — | |
JMJSTGZRLYHCCI
|
6.2 | IC50 | 5 | — | |
SIXGXRZCYDCNFL
|
6.2 | IC50 | 4 | — | |
CWFIQHQECWPWQG
|
6.2 | IC50 | 16 | Yes | |
MWKSRKSEWLRPBL
|
6.2 | Kd | 1075 | — | |
ORNADCNXUPZOQN
|
6.2 | IC50 | 15 | — | |
RDFXBYJUHGEYHA
|
6.2 | IC50 | 9 | Yes | |
KLYPYTHLYUUKMT
|
6.2 | Ki | 4 | — | |
CAGLPTUMBKISRZ
|
6.1 | IC50 | 2 | — | |
AXTAPYRUEKNRBA
|
6.1 | IC50 | 24 | — | |
CEMBEUHBOHDWPN
|
6.1 | IC50 | 4 | — | |
QYTBMLLWBZLPMF
|
6.1 | IC50 | 6 | — | |
DZIUPOCVDSYPSY
|
6.1 | IC50 | 8 | Yes | |
GCNSUXMONRYRHL
|
6.1 | IC50 | 4 | Yes | |
WSXYBDKZFNJOTP
|
6.1 | IC50 | 12 | Yes | |
MRBNLCLXWRXFJX
|
6.1 | IC50 | 15 | — | |
RZHAEOSLBJVDFX
|
6.1 | IC50 | 5 | — | |
GVSRILDMSGVJTR
|
6.1 | IC50 | 7 | — | |
ZMNWXCJLFBVMEJ
|
6.1 | IC50 | 3 | — | |
OBRQLJITIRIMLQ
|
6.1 | IC50 | 11 | — | |
KHGDEZDNICAMOO
|
6.1 | IC50 | 6 | — | |
GHRBXKFGXPOEGA
|
6.0 | IC50 | 12 | Yes | |
IBTJHABKSWXSHB
|
6.0 | IC50 | 2 | — | |
WNDOFCPEDZYDPL
|
6.0 | IC50 | 10 | — | |
DVMQYKHCZLPSAP
|
6.0 | IC50 | 5 | — | |
BMXGRFBSHSEZOP
|
6.0 | IC50 | 5 | Yes |