Target Details
| UniProt AC | P05556 |
|---|---|
| Gene Symbol | ITGB1 |
| Protein Name | Integrin beta-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07974 (EGF_2) PF23105 (EGF_integrin) PF18372 (I-EGF_1) PF08725 (Integrin_b_cyt) PF07965 (Integrin_B_tail) PF00362 (Integrin_beta) PF17205 (PSI_integrin) |
Summary
- Multi-target molecules 1,572
- Clinical molecules 0
- Avg pChEMBL 7.77
KEGG Pathways (29)
- Arrhythmogenic right ventricular cardiomyopathy
- Axon guidance
- Bacterial invasion of epithelial cells
- Cell adhesion molecule (CAM) interaction
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Focal adhesion
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- IgSF CAM signaling
- Integrin signaling
- Leishmaniasis
- Leukocyte transendothelial migration
- PI3K-Akt signaling pathway
- Pathogenic Escherichia coli infection
- Pathways in cancer
- Pertussis
- Phagosome
- Platelet activation
- Proteoglycans in cancer
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Shigellosis
- Small cell lung cancer
- Tight junction
- Toxoplasmosis
- Virion - Rotavirus
- Yersinia infection
Active Molecules (1,572)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WQKGOLGYPXZSSX
|
8.5 | IC50 | 2 | — | |
XWFOQFNTOYPKSS
|
8.5 | IC50 | 2 | — | |
YXFDUNGSOONFHY
|
8.5 | IC50 | 2 | — | |
ZWYAVCQGXAHVLZ
|
8.5 | IC50 | 2 | — | |
CPBOFXSFJQORHL
|
8.5 | IC50 | 2 | — | |
DBRVODXNNJOQHW
|
8.5 | IC50 | 2 | — | |
FXNGYKSGVMSVJB
|
8.5 | IC50 | 2 | — | |
JTHRYJJUORFXHX
|
8.5 | IC50 | 2 | — | |
USYYNLPEWBGIMJ
|
8.5 | IC50 | 2 | — | |
BADDGEGOMPMKGI
|
8.5 | IC50 | 2 | — | |
CPADDNAHPXAQNL
|
8.5 | IC50 | 2 | — | |
LPTLKRBMBJHFHY
|
8.5 | IC50 | 3 | — | |
ONTULEYBHLEJBB
|
8.5 | IC50 | 2 | — | |
QVXKEVCSWQRIDQ
|
8.5 | IC50 | 2 | — | |
UMIUGDHVXREPOA
|
8.5 | IC50 | 2 | — | |
ADRBWUVQHKFVMS
|
8.5 | IC50 | 3 | — | |
BESXQTSZSXTMFO
|
8.5 | IC50 | 2 | — | |
RQFGLPBPADHEDL
|
8.5 | IC50 | 2 | — | |
ZMSHCQNPVJGYNG
|
8.5 | IC50 | 2 | — | |
QQSLHONKFQQQNS
|
8.5 | IC50 | 2 | — | |
YOCCTHZQHRBDCH
|
8.5 | IC50 | 3 | — | |
DWDDWGYZNYHOGW
|
8.4 | IC50 | 2 | — | |
LKUHHZPYAGRQJR
|
8.4 | IC50 | 2 | — | |
LYBFJWLDWYPLFI
|
8.4 | IC50 | 2 | — | |
PRAQNLQOJOFZRC
|
8.4 | IC50 | 2 | — | |
MZPKCSOECXTYLC
|
8.4 | IC50 | 2 | — | |
OURYZIAAXSSBIO
|
8.4 | IC50 | 5 | — | |
BRPCXPCQFDLQMG
|
8.4 | IC50 | 2 | — | |
DGTPDOWNYVTTSD
|
8.4 | IC50 | 2 | — | |
KDBWXBVKPMEHLY
|
8.4 | IC50 | 2 | — | |
VHVHUZLIYQWAJK
|
8.4 | IC50 | 2 | — | |
AHCTUJXINUDHPY
|
8.4 | IC50 | 2 | — | |
BYRKTALPFLWGRH
|
8.4 | IC50 | 2 | — | |
UQZSJSAYODPZDI
|
8.4 | IC50 | 2 | — | |
VWGXMPUNQZIEBK
|
8.4 | IC50 | 2 | — | |
WEVSHWPVGKQWOF
|
8.4 | IC50 | 2 | — | |
XWZXOSXSUDVTSY
|
8.4 | IC50 | 3 | — | |
BWEJBCQAWORYOW
|
8.4 | IC50 | 2 | — | |
IUFCIFVCEOUHLU
|
8.4 | IC50 | 2 | — | |
NSGJGOWVFDUULW
|
8.4 | Ki | 2 | — | |
QTTOUXZPHJSBFZ
|
8.4 | IC50 | 2 | — | |
ROXYEKDRUFPSTJ
|
8.4 | IC50 | 2 | — | |
SGNBDDWCPLULSJ
|
8.4 | Ki | 2 | — | |
ZMHRAQMRFBHOKH
|
8.4 | IC50 | 2 | — | |
ZZQVVTQOTXKPIG
|
8.4 | IC50 | 2 | — | |
IDUDYLQZZVVIFO
|
8.4 | IC50 | 3 | — | |
UHGBRBWWHMGFEZ
|
8.4 | IC50 | 2 | — | |
VARBGWCQRGTWAS
|
8.4 | IC50 | 2 | — | |
LWCMKXYMIBQWPV
|
8.4 | IC50 | 2 | — | |
CPBOFXSFJQORHL
|
8.4 | IC50 | 2 | — |