Target Details
| UniProt AC | P05556 |
|---|---|
| Gene Symbol | ITGB1 |
| Protein Name | Integrin beta-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07974 (EGF_2) PF23105 (EGF_integrin) PF18372 (I-EGF_1) PF08725 (Integrin_b_cyt) PF07965 (Integrin_B_tail) PF00362 (Integrin_beta) PF17205 (PSI_integrin) |
Summary
- Multi-target molecules 1,572
- Clinical molecules 0
- Avg pChEMBL 7.77
KEGG Pathways (29)
- Arrhythmogenic right ventricular cardiomyopathy
- Axon guidance
- Bacterial invasion of epithelial cells
- Cell adhesion molecule (CAM) interaction
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Focal adhesion
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- IgSF CAM signaling
- Integrin signaling
- Leishmaniasis
- Leukocyte transendothelial migration
- PI3K-Akt signaling pathway
- Pathogenic Escherichia coli infection
- Pathways in cancer
- Pertussis
- Phagosome
- Platelet activation
- Proteoglycans in cancer
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Shigellosis
- Small cell lung cancer
- Tight junction
- Toxoplasmosis
- Virion - Rotavirus
- Yersinia infection
Active Molecules (1,572)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VPJJESVGYJPWNF
|
8.7 | IC50 | 2 | — | |
DZZGWIOPCRAELG
|
8.7 | IC50 | 2 | — | |
RYYQCANRHNEFSA
|
8.7 | Ki | 2 | — | |
HISUKZFCUMSJFG
|
8.6 | IC50 | 3 | — | |
HJBLGUARYIQSOP
|
8.6 | IC50 | 2 | — | |
SSYLLNMYBQFPCH
|
8.6 | IC50 | 3 | — | |
ULYHJYGNJKWWDI
|
8.6 | IC50 | 2 | — | |
QARMMTGRKYICJC
|
8.6 | IC50 | 2 | — | |
AESXNYDCOYLGAH
|
8.6 | IC50 | 2 | — | |
GJFNKTYJRCAGCV
|
8.6 | IC50 | 3 | — | |
LETDUXBWZBQZEK
|
8.6 | IC50 | 2 | — | |
QLSFJHYLUVSHEA
|
8.6 | IC50 | 2 | — | |
BQGQVBGSESRXLR
|
8.6 | Ki | 2 | — | |
BTYSVIBSJVRJTA
|
8.6 | Ki | 2 | — | |
LKEWELOHCDVPMS
|
8.6 | IC50 | 4 | — | |
YDWZFLXHAFVVPG
|
8.6 | Ki | 2 | — | |
MUMCFXBPBDMRQQ
|
8.6 | IC50 | 2 | — | |
PRTDUHZCDXSBIZ
|
8.6 | IC50 | 5 | — | |
VXONPVFJSPELTA
|
8.6 | IC50 | 2 | — | |
YUOMCSBLOMSMSI
|
8.6 | IC50 | 3 | — | |
ZMXBIIQMSGOIRZ
|
8.6 | Kd | 7 | — | |
BYRKTALPFLWGRH
|
8.6 | IC50 | 2 | — | |
JOZJWMSTRAKGKY
|
8.6 | IC50 | 2 | — | |
KFKKFCVUQZXZEI
|
8.6 | IC50 | 2 | — | |
KZYWKHUJTXLNJM
|
8.6 | IC50 | 5 | — | |
LKNNQWMGOZFFKT
|
8.6 | IC50 | 3 | — | |
OCIRIHRFAHXBIT
|
8.6 | IC50 | 3 | — | |
SAYYIMRPRXVLIL
|
8.6 | IC50 | 3 | — | |
ILIJAAWQIUXHNY
|
8.6 | IC50 | 2 | — | |
LTQGACDEOSCTBA
|
8.6 | IC50 | 3 | — | |
YKDBMBISKSKBIS
|
8.6 | IC50 | 2 | — | |
ZLNBTVYNXDCEPU
|
8.6 | IC50 | 2 | — | |
AZIOXOMBBGKKBJ
|
8.5 | IC50 | 3 | — | |
FZMHKLISSNPJKF
|
8.5 | IC50 | 2 | — | |
KHZVLOYNGSJKBU
|
8.5 | IC50 | 2 | — | |
LYIQTSRHBZHIPH
|
8.5 | IC50 | 2 | — | |
XAVTVDBSJQZNHA
|
8.5 | IC50 | 2 | — | |
ZVYKWIXTSCOLQS
|
8.5 | IC50 | 2 | — | |
AEAYDNFPSLYSOA
|
8.5 | IC50 | 2 | — | |
BNMACLPLFKEEMT
|
8.5 | IC50 | 2 | — | |
FOABJUOBCGOTCS
|
8.5 | IC50 | 2 | — | |
IBXMYCNAAVLIET
|
8.5 | IC50 | 4 | — | |
ILKTTWKSRXZSRE
|
8.5 | IC50 | 2 | — | |
IXDDZIVBYAEUTN
|
8.5 | IC50 | 3 | — | |
JIYOXFLRVUFAQT
|
8.5 | IC50 | 2 | — | |
MKCISCXMJCFWLW
|
8.5 | IC50 | 2 | — | |
MONYNIRDTFXWKB
|
8.5 | IC50 | 2 | — | |
QMHTXRUDZGHUND
|
8.5 | IC50 | 2 | — | |
WEBZMJPCAJJKTN
|
8.5 | IC50 | 2 | — | |
WEXUEGAYHTYTGF
|
8.5 | IC50 | 2 | — |