Target Details
| UniProt AC | P05556 |
|---|---|
| Gene Symbol | ITGB1 |
| Protein Name | Integrin beta-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07974 (EGF_2) PF23105 (EGF_integrin) PF18372 (I-EGF_1) PF08725 (Integrin_b_cyt) PF07965 (Integrin_B_tail) PF00362 (Integrin_beta) PF17205 (PSI_integrin) |
Summary
- Multi-target molecules 1,572
- Clinical molecules 0
- Avg pChEMBL 7.77
KEGG Pathways (29)
- Arrhythmogenic right ventricular cardiomyopathy
- Axon guidance
- Bacterial invasion of epithelial cells
- Cell adhesion molecule (CAM) interaction
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Focal adhesion
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- IgSF CAM signaling
- Integrin signaling
- Leishmaniasis
- Leukocyte transendothelial migration
- PI3K-Akt signaling pathway
- Pathogenic Escherichia coli infection
- Pathways in cancer
- Pertussis
- Phagosome
- Platelet activation
- Proteoglycans in cancer
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Shigellosis
- Small cell lung cancer
- Tight junction
- Toxoplasmosis
- Virion - Rotavirus
- Yersinia infection
Active Molecules (1,572)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OSNQUPAEVQKVCT
|
8.8 | IC50 | 2 | — | |
UEBUMZGZKUPTHB
|
8.8 | IC50 | 4 | — | |
GNBZNYOXBLSXKD
|
8.8 | IC50 | 3 | — | |
UZDJXPGRSXEUQF
|
8.8 | IC50 | 2 | — | |
YTYJFLBPXSXTSC
|
8.8 | IC50 | 2 | — | |
JREFABWTIILFKQ
|
8.8 | IC50 | 2 | — | |
NVSCTWCNVXBLQP
|
8.8 | IC50 | 3 | — | |
OHGDWXKKIOEWBM
|
8.8 | IC50 | 2 | — | |
QCSCWVKEGWWYHS
|
8.8 | IC50 | 2 | — | |
UZVROHMMUDQAOJ
|
8.8 | IC50 | 5 | — | |
YZZMJHSHQYXEFZ
|
8.8 | IC50 | 2 | — | |
ZPYVSGYLDUOOIZ
|
8.8 | IC50 | 2 | — | |
LYEWIWRMQRJNFS
|
8.8 | IC50 | 2 | — | |
UDEOSPCGCDINCC
|
8.8 | IC50 | 2 | — | |
HJWCBRDYEUTPNN
|
8.8 | IC50 | 2 | — | |
RYQVJWYRMJZFAD
|
8.8 | IC50 | 2 | — | |
WUAFZBANWSFBSP
|
8.8 | IC50 | 2 | — | |
CWIZGCPRLPKGAW
|
8.7 | IC50 | 2 | — | |
KCHWAIVFBMDFOL
|
8.7 | IC50 | 2 | — | |
KGDZUGSBEBVXKQ
|
8.7 | IC50 | 3 | — | |
YDHAGPCZRFQPOI
|
8.7 | IC50 | 6 | — | |
ZSLLAAOZAJPOMZ
|
8.7 | IC50 | 2 | — | |
FSIOKPLPDOYRFJ
|
8.7 | IC50 | 2 | — | |
BRXOSTDCWWZMCS
|
8.7 | IC50 | 2 | — | |
NAGIMKJAUDLRFH
|
8.7 | IC50 | 4 | — | |
SCAJVSZKETYPPT
|
8.7 | IC50 | 3 | — | |
QBLBCXCNIKAKNO
|
8.7 | IC50 | 3 | — | |
BYORRPJZRWMSCK
|
8.7 | IC50 | 2 | — | |
CKPFLCVDCRYWAY
|
8.7 | IC50 | 3 | — | |
IHZDVSSJVCEYBR
|
8.7 | Ki | 2 | — | |
JEBRWBXEAHSNTF
|
8.7 | Ki | 2 | — | |
JHBJKRQQEIQKHE
|
8.7 | IC50 | 2 | — | |
JMRHAIGRROKJRA
|
8.7 | IC50 | 2 | — | |
QTTOUXZPHJSBFZ
|
8.7 | IC50 | 2 | — | |
SJHWRZBMMCDJDX
|
8.7 | IC50 | 2 | — | |
UCBYYQWMMNUSGH
|
8.7 | IC50 | 8 | — | |
UHXBOYLWYUPYDA
|
8.7 | IC50 | 3 | — | |
UOCOERCBTSGDPC
|
8.7 | IC50 | 2 | — | |
UOQRUCISSASGLE
|
8.7 | IC50 | 2 | — | |
VVZGYMGXVWZKDS
|
8.7 | IC50 | 2 | — | |
XFHCUQCLLGVBIK
|
8.7 | IC50 | 3 | — | |
ZSKXPSIETQZQJF
|
8.7 | Ki | 2 | — | |
MZVLJIIBEREKBQ
|
8.7 | IC50 | 2 | — | |
UMSYINVARMBJFW
|
8.7 | IC50 | 2 | — | |
WRHKZVFBIZOZCV
|
8.7 | IC50 | 2 | — | |
WRHKZVFBIZOZCV
|
8.7 | IC50 | 2 | — | |
WGSFNDOOBOZLMA
|
8.7 | IC50 | 3 | — | |
CBLWZZPATNWACH
|
8.7 | IC50 | 2 | — | |
GRSVHAPJHOVVNB
|
8.7 | IC50 | 2 | — | |
GSCXEBUWSNKNJK
|
8.7 | IC50 | 3 | — |