Target Details
| UniProt AC | P05556 |
|---|---|
| Gene Symbol | ITGB1 |
| Protein Name | Integrin beta-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07974 (EGF_2) PF23105 (EGF_integrin) PF18372 (I-EGF_1) PF08725 (Integrin_b_cyt) PF07965 (Integrin_B_tail) PF00362 (Integrin_beta) PF17205 (PSI_integrin) |
Summary
- Multi-target molecules 1,572
- Clinical molecules 0
- Avg pChEMBL 7.77
KEGG Pathways (29)
- Arrhythmogenic right ventricular cardiomyopathy
- Axon guidance
- Bacterial invasion of epithelial cells
- Cell adhesion molecule (CAM) interaction
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Focal adhesion
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- IgSF CAM signaling
- Integrin signaling
- Leishmaniasis
- Leukocyte transendothelial migration
- PI3K-Akt signaling pathway
- Pathogenic Escherichia coli infection
- Pathways in cancer
- Pertussis
- Phagosome
- Platelet activation
- Proteoglycans in cancer
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Shigellosis
- Small cell lung cancer
- Tight junction
- Toxoplasmosis
- Virion - Rotavirus
- Yersinia infection
Active Molecules (1,572)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NJWAMCOTWKQQQO
|
9.0 | IC50 | 2 | — | |
OPKAUQAIFQSBOZ
|
9.0 | IC50 | 2 | — | |
SMMNOJYHMMCWQP
|
9.0 | IC50 | 5 | — | |
VVWWYYCPGHVEKY
|
9.0 | IC50 | 3 | — | |
WPKLWLSFNMQEKC
|
9.0 | IC50 | 3 | — | |
XFEBZCPSSQZCEA
|
9.0 | IC50 | 3 | — | |
ZAMKDPACDNUZPJ
|
9.0 | IC50 | 8 | — | |
XXMAAHCJSQLUJD
|
8.9 | IC50 | 2 | — | |
BWAUVRFZNDRMLY
|
8.9 | IC50 | 8 | — | |
DQNZNDKDCJZRKQ
|
8.9 | IC50 | 2 | — | |
MWICRKHXHXGESF
|
8.9 | IC50 | 3 | — | |
CAXSRPBPCGUCIY
|
8.9 | IC50 | 3 | — | |
JQZNUGKWTQHGEY
|
8.9 | IC50 | 2 | — | |
OUOYSXSWASMDOM
|
8.9 | IC50 | 2 | — | |
POLDUUDTCKSSFP
|
8.9 | IC50 | 3 | — | |
ZWTNWDWPPZZGCJ
|
8.9 | IC50 | 2 | — | |
FPKILHQBPJHCHS
|
8.9 | IC50 | 2 | — | |
ATIKCNMCFMFEID
|
8.9 | IC50 | 2 | — | |
CQECYVMYMPYNBF
|
8.9 | IC50 | 2 | — | |
CXHCNOMGODVIKB
|
8.9 | IC50 | 7 | — | |
HTKRKKLTEHJRRC
|
8.9 | IC50 | 2 | — | |
SQQCECFUGOZGKP
|
8.9 | IC50 | 3 | — | |
ULSOWJGEUXLWAX
|
8.9 | IC50 | 2 | — | |
YKTFSYAGPCXYHA
|
8.9 | IC50 | 2 | — | |
DLBHIUWUQMPJLY
|
8.9 | IC50 | 2 | — | |
NEHVNFYXIGYVRB
|
8.9 | IC50 | 2 | — | |
CBKWFBALGVYSLI
|
8.8 | IC50 | 2 | — | |
DBUZBTZXIHIIOJ
|
8.8 | IC50 | 2 | — | |
GKBOWSGQVIXZHX
|
8.8 | IC50 | 2 | — | |
MMLPNYXAJOWDEN
|
8.8 | IC50 | 2 | — | |
SMNXQFKEUFRQPU
|
8.8 | IC50 | 2 | — | |
ZOESWPXJPYGCKJ
|
8.8 | IC50 | 2 | — | |
XGNHXBRBECYIIH
|
8.8 | IC50 | 2 | — | |
GNNSUMADLWATJP
|
8.8 | IC50 | 5 | — | |
NDTSMDJDMBJXNX
|
8.8 | IC50 | 2 | — | |
PLQYIPNBZHAKRA
|
8.8 | IC50 | 3 | — | |
PWARPDYCBZDQLI
|
8.8 | IC50 | 2 | — | |
QGKYFEGJAYKPGL
|
8.8 | IC50 | 2 | — | |
UNKOTAZGQDRZGB
|
8.8 | IC50 | 2 | — | |
VZARBYRZKJWXIK
|
8.8 | IC50 | 2 | — | |
ASBZESJHVHSKOI
|
8.8 | IC50 | 2 | — | |
AZJYXUVHLYXCJY
|
8.8 | IC50 | 2 | — | |
AZJYXUVHLYXCJY
|
8.8 | IC50 | 2 | — | |
BSNWAPOUYOPCPS
|
8.8 | IC50 | 6 | — | |
GCTCMPMLQFPTJM
|
8.8 | IC50 | 2 | — | |
HIUGMXDAZTUBDD
|
8.8 | Ki | 2 | — | |
HUPHLMZTLJGDRG
|
8.8 | IC50 | 3 | — | |
JTUKSGXZGMYCDU
|
8.8 | IC50 | 2 | — | |
LXOSRVCKEOYAQT
|
8.8 | IC50 | 2 | — | |
OJYKDVHESROECH
|
8.8 | IC50 | 2 | — |