Target Details
| UniProt AC | P05556 |
|---|---|
| Gene Symbol | ITGB1 |
| Protein Name | Integrin beta-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07974 (EGF_2) PF23105 (EGF_integrin) PF18372 (I-EGF_1) PF08725 (Integrin_b_cyt) PF07965 (Integrin_B_tail) PF00362 (Integrin_beta) PF17205 (PSI_integrin) |
Summary
- Multi-target molecules 1,572
- Clinical molecules 0
- Avg pChEMBL 7.77
KEGG Pathways (29)
- Arrhythmogenic right ventricular cardiomyopathy
- Axon guidance
- Bacterial invasion of epithelial cells
- Cell adhesion molecule (CAM) interaction
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Focal adhesion
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- IgSF CAM signaling
- Integrin signaling
- Leishmaniasis
- Leukocyte transendothelial migration
- PI3K-Akt signaling pathway
- Pathogenic Escherichia coli infection
- Pathways in cancer
- Pertussis
- Phagosome
- Platelet activation
- Proteoglycans in cancer
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Shigellosis
- Small cell lung cancer
- Tight junction
- Toxoplasmosis
- Virion - Rotavirus
- Yersinia infection
Active Molecules (1,572)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZEDVVTNZWFMRKR
|
9.1 | IC50 | 3 | — | |
GYNQANKDGGTNRK
|
9.1 | IC50 | 3 | — | |
CRLOUCQPUXMUCD
|
9.1 | IC50 | 2 | — | |
GYRBFYNAOXAEPO
|
9.1 | IC50 | 2 | — | |
HIKDGFUZLZJZCB
|
9.1 | IC50 | 8 | — | |
RTQDJONLCOQVMI
|
9.1 | IC50 | 2 | — | |
UUXTZGJGBUBTBQ
|
9.1 | IC50 | 2 | — | |
WHAMHFBSIWLDIJ
|
9.1 | IC50 | 2 | — | |
FPKILHQBPJHCHS
|
9.1 | IC50 | 3 | — | |
OVAMYRDVZGRBCF
|
9.1 | IC50 | 2 | — | |
JPDURLRTQZCKKD
|
9.1 | IC50 | 2 | — | |
LPPNDFOQUKQERO
|
9.1 | IC50 | 3 | — | |
VTZMVMKHYIBVPC
|
9.1 | IC50 | 3 | — | |
XHCXORPSNPUSKF
|
9.1 | IC50 | 2 | — | |
XLANGJRVQABTFO
|
9.1 | IC50 | 5 | — | |
KFMZAEHOOJXIHH
|
9.0 | IC50 | 3 | — | |
NXAVFGCSONIIII
|
9.0 | IC50 | 2 | — | |
PUGXPRVUVZGAHB
|
9.0 | IC50 | 2 | — | |
FQKAGOPIYIPBGP
|
9.0 | IC50 | 2 | — | |
KSRNGDACGBIPKZ
|
9.0 | IC50 | 3 | — | |
ZLSOUAKIYFWGAA
|
9.0 | IC50 | 2 | — | |
LWMXBHHAGNVCLL
|
9.0 | IC50 | 3 | — | |
BQGQVBGSESRXLR
|
9.0 | Ki | 2 | — | |
BQYBIJDRTDZCAJ
|
9.0 | IC50 | 8 | — | |
BTYSVIBSJVRJTA
|
9.0 | Ki | 2 | — | |
FZHRZAHVVNSORE
|
9.0 | IC50 | 2 | — | |
GFTVRPWYQDITLC
|
9.0 | IC50 | 5 | — | |
LXYBJVGMCKOMFL
|
9.0 | IC50 | 2 | — | |
POFWSMHHXSOAAJ
|
9.0 | Ki | 2 | — | |
PQNWKBRBHJLNTG
|
9.0 | IC50 | 2 | — | |
SFAOKQAQLNGQIZ
|
9.0 | IC50 | 3 | — | |
USEDUTJSKDZBGX
|
9.0 | IC50 | 2 | — | |
UTLDJUNUIMQLSJ
|
9.0 | IC50 | 3 | — | |
VOKWLPMZPWNTFX
|
9.0 | IC50 | 2 | — | |
XRXSSPOFDFFALK
|
9.0 | IC50 | 8 | — | |
YVTBYYRAVCBZCJ
|
9.0 | IC50 | 2 | — | |
ZIPHKIDWZBDOSS
|
9.0 | IC50 | 3 | — | |
ZSKXPSIETQZQJF
|
9.0 | Ki | 2 | — | |
PWMAEWNRSJGUGQ
|
9.0 | IC50 | 2 | — | |
NFMHJWOVOIOOTE
|
9.0 | IC50 | 3 | — | |
OFKDMFLFKUWHRQ
|
9.0 | IC50 | 2 | — | |
QLBXWVBTUGYSGI
|
9.0 | IC50 | 8 | — | |
AAQGLFLATBVJPM
|
9.0 | IC50 | 3 | — | |
AEMBNJITTWJYBV
|
9.0 | IC50 | 3 | — | |
BLKCXKZUJXHCGP
|
9.0 | IC50 | 4 | — | |
CGSLGBRMSMBNMX
|
9.0 | IC50 | 6 | — | |
CJRDXSVCUSRJDR
|
9.0 | IC50 | 8 | — | |
GRKQLMXUWWDASB
|
9.0 | IC50 | 2 | — | |
JNMQDVKBQWASOW
|
9.0 | IC50 | 3 | — | |
KKZBAYODMNBMQJ
|
9.0 | IC50 | 3 | — |