Target Details
| UniProt AC | P05556 |
|---|---|
| Gene Symbol | ITGB1 |
| Protein Name | Integrin beta-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07974 (EGF_2) PF23105 (EGF_integrin) PF18372 (I-EGF_1) PF08725 (Integrin_b_cyt) PF07965 (Integrin_B_tail) PF00362 (Integrin_beta) PF17205 (PSI_integrin) |
Summary
- Multi-target molecules 1,572
- Clinical molecules 0
- Avg pChEMBL 7.77
KEGG Pathways (29)
- Arrhythmogenic right ventricular cardiomyopathy
- Axon guidance
- Bacterial invasion of epithelial cells
- Cell adhesion molecule (CAM) interaction
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Focal adhesion
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- IgSF CAM signaling
- Integrin signaling
- Leishmaniasis
- Leukocyte transendothelial migration
- PI3K-Akt signaling pathway
- Pathogenic Escherichia coli infection
- Pathways in cancer
- Pertussis
- Phagosome
- Platelet activation
- Proteoglycans in cancer
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Shigellosis
- Small cell lung cancer
- Tight junction
- Toxoplasmosis
- Virion - Rotavirus
- Yersinia infection
Active Molecules (1,572)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HWTDZVDHOSKTML
|
9.3 | IC50 | 3 | — | |
RNWJDKPVADJMJR
|
9.3 | IC50 | 3 | — | |
YXPCBCHWUVICEH
|
9.3 | IC50 | 2 | — | |
KAGRGOJSNNEPTP
|
9.3 | IC50 | 2 | — | |
LMTFGZLYPXNJRU
|
9.3 | IC50 | 2 | — | |
QPBVMPSYTAHRNI
|
9.3 | IC50 | 2 | — | |
BXXARJACSOMMKX
|
9.3 | IC50 | 2 | — | |
DAEIMVCXNQVMSM
|
9.3 | IC50 | 3 | — | |
LTEAZKWKEALJQD
|
9.3 | IC50 | 4 | — | |
WFNCDDGCGNUXLG
|
9.3 | IC50 | 2 | — | |
SITGJFUZUFHSHU
|
9.2 | IC50 | 3 | — | |
RXOAYEHOAAHUMM
|
9.2 | IC50 | 2 | — | |
MFCABRSSOZYCRL
|
9.2 | IC50 | 8 | — | |
NWQAJABKOGMVNQ
|
9.2 | IC50 | 2 | — | |
PEFBVOAICYLSAF
|
9.2 | IC50 | 8 | — | |
QTBFGJFGHGTDRF
|
9.2 | IC50 | 8 | — | |
SHRSEUHJTZQLRO
|
9.2 | IC50 | 8 | — | |
CRLQMBSOODURJR
|
9.2 | IC50 | 3 | — | |
BLLLAUHTNAVSQR
|
9.2 | IC50 | 5 | — | |
BRZKFEHVZLVFIJ
|
9.2 | IC50 | 2 | — | |
FSJCFVNPVGEGOY
|
9.2 | IC50 | 2 | — | |
NOWFLJYSWCXTKI
|
9.2 | IC50 | 2 | — | |
IYTTUCDELWMTPJ
|
9.2 | IC50 | 2 | — | |
SATRONDTGPPWOY
|
9.2 | IC50 | 3 | — | |
GDEQKRGKHZOXGD
|
9.2 | IC50 | 8 | — | |
XQYVKXLNFSIYBI
|
9.2 | IC50 | 2 | — | |
AKXPOHLUWJPKQY
|
9.2 | IC50 | 2 | — | |
BKYBRLBEBOMPJQ
|
9.2 | IC50 | 3 | — | |
OSOUXNDWVSWDJT
|
9.2 | IC50 | 2 | — | |
QPZOEIQRDYCGMD
|
9.2 | IC50 | 5 | — | |
RLDCURKHNWEZOG
|
9.2 | IC50 | 3 | — | |
RTYLRDWEJUNBLU
|
9.2 | IC50 | 8 | — | |
UDGWKAUBGPXUNT
|
9.2 | IC50 | 2 | — | |
YPAMHQMVIMQKOR
|
9.2 | IC50 | 8 | — | |
RJALSTOENHOZQV
|
9.1 | IC50 | 3 | — | |
SALKSINYSDSNQB
|
9.1 | IC50 | 2 | — | |
VVKWSNOGZODKEQ
|
9.1 | IC50 | 3 | — | |
XTGPAZFJJAYMMR
|
9.1 | IC50 | 2 | — | |
QPBGCQHXTQTQCH
|
9.1 | IC50 | 2 | — | |
NVHYHKRZUDLBBQ
|
9.1 | IC50 | 3 | — | |
QSVHEGNXLMFWSO
|
9.1 | IC50 | 3 | — | |
GSCDUHGSEPUEQF
|
9.1 | IC50 | 3 | — | |
SMZRAZWAVQZBEC
|
9.1 | IC50 | 3 | — | |
XINCANZSFCTALF
|
9.1 | IC50 | 2 | — | |
CCBJMQPSBBHXRQ
|
9.1 | IC50 | 2 | — | |
IPSRDFZOWABPRU
|
9.1 | IC50 | 4 | — | |
POFWSMHHXSOAAJ
|
9.1 | Ki | 2 | — | |
PTCMVGOQRMWOTP
|
9.1 | IC50 | 4 | — | |
PUJRKGKDIKCRSV
|
9.1 | Ki | 2 | — | |
VOCBDNRGLAJDJJ
|
9.1 | Ki | 2 | — |