Target Details
| UniProt AC | P05556 |
|---|---|
| Gene Symbol | ITGB1 |
| Protein Name | Integrin beta-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07974 (EGF_2) PF23105 (EGF_integrin) PF18372 (I-EGF_1) PF08725 (Integrin_b_cyt) PF07965 (Integrin_B_tail) PF00362 (Integrin_beta) PF17205 (PSI_integrin) |
Summary
- Multi-target molecules 1,572
- Clinical molecules 0
- Avg pChEMBL 7.77
KEGG Pathways (29)
- Arrhythmogenic right ventricular cardiomyopathy
- Axon guidance
- Bacterial invasion of epithelial cells
- Cell adhesion molecule (CAM) interaction
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Focal adhesion
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- IgSF CAM signaling
- Integrin signaling
- Leishmaniasis
- Leukocyte transendothelial migration
- PI3K-Akt signaling pathway
- Pathogenic Escherichia coli infection
- Pathways in cancer
- Pertussis
- Phagosome
- Platelet activation
- Proteoglycans in cancer
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Shigellosis
- Small cell lung cancer
- Tight junction
- Toxoplasmosis
- Virion - Rotavirus
- Yersinia infection
Active Molecules (1,572)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NBFYQDLZBZGXPB
|
9.5 | IC50 | 4 | — | |
NICNHDFNJXGGJV
|
9.5 | IC50 | 2 | — | |
PXIBPFAADDDFDQ
|
9.5 | IC50 | 3 | — | |
GMZQXSJOGNIVAK
|
9.5 | IC50 | 3 | — | |
SPYRCTMYBNFJRX
|
9.5 | IC50 | 3 | — | |
WKEYMRCHVPVMOY
|
9.5 | IC50 | 3 | — | |
GDSMXSYVAAVCRV
|
9.5 | IC50 | 3 | — | |
APJVOWJJCXAZNW
|
9.4 | IC50 | 3 | — | |
FILAPYMFTPTZNJ
|
9.4 | IC50 | 2 | — | |
CJASQSIGTKSMFJ
|
9.4 | IC50 | 3 | — | |
UTRBTIFHRKMFMU
|
9.4 | IC50 | 3 | — | |
XVFGXBXVSHPQNQ
|
9.4 | IC50 | 3 | — | |
GRIXHDLHYDUGHP
|
9.4 | IC50 | 2 | — | |
MMIPQFQYOLUDRE
|
9.4 | IC50 | 3 | — | |
FAQBNGGMUXLXSQ
|
9.4 | IC50 | 3 | — | |
JXVVEFIKDDVLOS
|
9.4 | IC50 | 8 | — | |
LBTMUQGNXSWGSG
|
9.4 | IC50 | 3 | — | |
MMKDEARGHIPLGR
|
9.4 | IC50 | 2 | — | |
QPZMNXQBHCXEKU
|
9.4 | IC50 | 2 | — | |
YQOFOSAJQMWIAT
|
9.4 | IC50 | 4 | — | |
AHUFAXIJOQGUOY
|
9.4 | IC50 | 2 | — | |
HLDVFPCKENBYRZ
|
9.4 | IC50 | 2 | — | |
GMXTVNCMABOSEI
|
9.4 | IC50 | 3 | — | |
RUTGLWCLWPBBMZ
|
9.4 | IC50 | 2 | — | |
LBTMUQGNXSWGSG
|
9.4 | IC50 | 3 | — | |
JSMSAVCWGLIOCE
|
9.4 | IC50 | 2 | — | |
TZHPMUDTJGJDTC
|
9.4 | IC50 | 2 | — | |
ZFEZMZIUQXOHHJ
|
9.4 | IC50 | 2 | — | |
IAXOAOUFMTWSPG
|
9.3 | IC50 | 3 | — | |
KLRZAJNROFRNBT
|
9.3 | IC50 | 2 | — | |
DDXWRMMINAREGF
|
9.3 | IC50 | 3 | — | |
FJTPRDFOASDXPB
|
9.3 | IC50 | 3 | — | |
NSAOFDPAHXXLPO
|
9.3 | IC50 | 3 | — | |
IRVJBUBWERQASS
|
9.3 | IC50 | 3 | — | |
VFYLHJRNSIZWQQ
|
9.3 | IC50 | 3 | — | |
XNBNFFZMGGWODG
|
9.3 | IC50 | 4 | — | |
XOCAITJQZBYGFQ
|
9.3 | IC50 | 5 | — | |
ACPZTVFLIFYRRX
|
9.3 | IC50 | 3 | — | |
GYUQWZWCORBSLX
|
9.3 | IC50 | 2 | — | |
HLUUKMWLLADVRH
|
9.3 | IC50 | 2 | — | |
CQLHRAHQMMCYBN
|
9.3 | IC50 | 2 | — | |
JUBGULNNHUDWAO
|
9.3 | IC50 | 3 | — | |
JZHPHPOLAVKTRC
|
9.3 | IC50 | 2 | — | |
JZHPHPOLAVKTRC
|
9.3 | IC50 | 2 | — | |
MOQBCMVOFUTVHS
|
9.3 | Ki | 2 | — | |
OBOJFQICXTYCRY
|
9.3 | IC50 | 8 | — | |
OYRUZFJXLJQJNA
|
9.3 | IC50 | 3 | — | |
YHFWYPZHVJZULG
|
9.3 | IC50 | 2 | — | |
WIBDJDYXWICGSX
|
9.3 | IC50 | 2 | — | |
CELGRUOLPJJNJO
|
9.3 | IC50 | 3 | — |