Target Details
| UniProt AC | P05556 |
|---|---|
| Gene Symbol | ITGB1 |
| Protein Name | Integrin beta-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07974 (EGF_2) PF23105 (EGF_integrin) PF18372 (I-EGF_1) PF08725 (Integrin_b_cyt) PF07965 (Integrin_B_tail) PF00362 (Integrin_beta) PF17205 (PSI_integrin) |
Summary
- Multi-target molecules 1,572
- Clinical molecules 0
- Avg pChEMBL 7.77
KEGG Pathways (29)
- Arrhythmogenic right ventricular cardiomyopathy
- Axon guidance
- Bacterial invasion of epithelial cells
- Cell adhesion molecule (CAM) interaction
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Focal adhesion
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- IgSF CAM signaling
- Integrin signaling
- Leishmaniasis
- Leukocyte transendothelial migration
- PI3K-Akt signaling pathway
- Pathogenic Escherichia coli infection
- Pathways in cancer
- Pertussis
- Phagosome
- Platelet activation
- Proteoglycans in cancer
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Shigellosis
- Small cell lung cancer
- Tight junction
- Toxoplasmosis
- Virion - Rotavirus
- Yersinia infection
Active Molecules (1,572)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JMYVXFQHQUNKFF
|
9.8 | IC50 | 2 | — | |
LUQNTQZWQQXMQY
|
9.8 | IC50 | 3 | — | |
ZNLSNWBYZFYQKK
|
9.8 | IC50 | 3 | — | |
ZUYLZBWPGTXZOO
|
9.8 | IC50 | 3 | — | |
OXNNEMDLTGEMOR
|
9.8 | Ki | 2 | — | |
DXZXXIJEZVYUJW
|
9.8 | IC50 | 3 | — | |
MGAGDDCVRPUJAS
|
9.8 | IC50 | 3 | — | |
UZEJXLHLCJUOKN
|
9.8 | IC50 | 3 | — | |
NOEWSRIYUKZVEG
|
9.7 | IC50 | 3 | — | |
AQGOTKCWRZAUIP
|
9.7 | IC50 | 3 | — | |
HGEHCBNZQHVLJS
|
9.7 | IC50 | 3 | — | |
QSPRBGPZFIOHRF
|
9.7 | IC50 | 3 | — | |
VBHVOJJDISNENC
|
9.7 | IC50 | 3 | — | |
YECQPPDRORMNRX
|
9.7 | IC50 | 3 | — | |
KNSPFVAZTITFFW
|
9.7 | IC50 | 3 | — | |
LPPNDFOQUKQERO
|
9.7 | IC50 | 3 | — | |
QGOXLUXYLLZODC
|
9.7 | IC50 | 3 | — | |
RDYYKKRRLZVNCE
|
9.7 | IC50 | 2 | — | |
DVLBSXLUGBCBRC
|
9.7 | IC50 | 3 | — | |
IGRGIQWZKAUHDT
|
9.7 | IC50 | 3 | — | |
IWJUFTWRMKICLP
|
9.7 | IC50 | 2 | — | |
VEAVPXNJUXKCMP
|
9.7 | IC50 | 3 | — | |
HAFRWCGZNZNVIH
|
9.7 | IC50 | 3 | — | |
MMYBBVWYPAIKBK
|
9.7 | IC50 | 2 | — | |
MXTOSAOISBOVCI
|
9.7 | IC50 | 3 | — | |
PRUPKWNQAVQPOI
|
9.7 | IC50 | 3 | — | |
WTUXQGQYRAGZCP
|
9.7 | IC50 | 3 | — | |
XMJDMDBLEIGQSK
|
9.7 | IC50 | 3 | — | |
HPTAYLDQFBSRPO
|
9.6 | IC50 | 2 | — | |
BNIJMUVCQMIEQC
|
9.6 | IC50 | 3 | — | |
LAVKEKZSIBZMRJ
|
9.6 | IC50 | 3 | — | |
MTTOAAIJCSWQGQ
|
9.6 | IC50 | 2 | — | |
QDGGQCVCHRACBF
|
9.6 | IC50 | 2 | — | |
TXDUNPFVQQSUTP
|
9.6 | IC50 | 3 | — | |
OEJOIHNKFVHVEB
|
9.6 | IC50 | 3 | — | |
UAWIVFLVAQKETC
|
9.6 | IC50 | 3 | — | |
CSMQOKNTHTXJFG
|
9.6 | IC50 | 3 | — | |
MLGBLCHXNBTYRD
|
9.6 | IC50 | 2 | — | |
YGJLELVDLMNGTP
|
9.6 | IC50 | 3 | — | |
DLLGQRYZARKEBS
|
9.6 | IC50 | 3 | — | |
UKDPVOZZLJCIKT
|
9.6 | IC50 | 3 | — | |
VPIVICLWCZPBIT
|
9.5 | IC50 | 3 | — | |
CJSJCPSXRGQDKE
|
9.5 | IC50 | 2 | — | |
CJSJCPSXRGQDKE
|
9.5 | IC50 | 2 | — | |
HXCIDANYYUBZDI
|
9.5 | IC50 | 2 | — | |
JHRWRZACLCUNPT
|
9.5 | IC50 | 3 | — | |
ZNTZLEVMFVHFEN
|
9.5 | IC50 | 2 | — | |
CXSIVJHZBHTFAQ
|
9.5 | IC50 | 3 | — | |
QHVMOHLLRYTFPS
|
9.5 | IC50 | 2 | — | |
YDWCAPCMYPCFNI
|
9.5 | IC50 | 2 | — |