Target Details
| UniProt AC | P05556 |
|---|---|
| Gene Symbol | ITGB1 |
| Protein Name | Integrin beta-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07974 (EGF_2) PF23105 (EGF_integrin) PF18372 (I-EGF_1) PF08725 (Integrin_b_cyt) PF07965 (Integrin_B_tail) PF00362 (Integrin_beta) PF17205 (PSI_integrin) |
Summary
- Multi-target molecules 1,572
- Clinical molecules 0
- Avg pChEMBL 7.77
KEGG Pathways (29)
- Arrhythmogenic right ventricular cardiomyopathy
- Axon guidance
- Bacterial invasion of epithelial cells
- Cell adhesion molecule (CAM) interaction
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Focal adhesion
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- IgSF CAM signaling
- Integrin signaling
- Leishmaniasis
- Leukocyte transendothelial migration
- PI3K-Akt signaling pathway
- Pathogenic Escherichia coli infection
- Pathways in cancer
- Pertussis
- Phagosome
- Platelet activation
- Proteoglycans in cancer
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Shigellosis
- Small cell lung cancer
- Tight junction
- Toxoplasmosis
- Virion - Rotavirus
- Yersinia infection
Active Molecules (1,572)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NVVGCQABIHSJSQ
|
8.4 | IC50 | 2 | — | |
GCESVLHCMHNRBV
|
8.4 | IC50 | 2 | — | |
ITXAAOWFOURIHK
|
8.4 | IC50 | 2 | — | |
ITXAAOWFOURIHK
|
8.4 | IC50 | 2 | — | |
SUPGBSSFNJDXNH
|
8.4 | IC50 | 2 | — | |
TXGCBKLXHVSCNM
|
8.4 | IC50 | 2 | — | |
TXTKZSBIOMEMHC
|
8.4 | IC50 | 3 | — | |
GGRFOSOSNAVBNN
|
8.3 | IC50 | 2 | — | |
IUEVXNMBIIQKAS
|
8.3 | IC50 | 2 | — | |
ZRKHLKCFHURIEZ
|
8.3 | IC50 | 2 | — | |
ZYGZRMMSJAKXOS
|
8.3 | IC50 | 2 | — | |
ZYGZRMMSJAKXOS
|
8.3 | IC50 | 2 | — | |
HPOGEWKAYYHIGE
|
8.3 | IC50 | 3 | — | |
RBTXBEVPBKTAJE
|
8.3 | IC50 | 2 | — | |
NVVGCQABIHSJSQ
|
8.3 | IC50 | 6 | — | |
RJGXUVWHSRSSMR
|
8.3 | IC50 | 2 | — | |
UFHRTJXQBDQBIP
|
8.3 | IC50 | 2 | — | |
WTQCOABHBBAPPQ
|
8.3 | IC50 | 2 | — | |
ZEAGMKZBQHJQAR
|
8.3 | IC50 | 2 | — | |
ADUOFHJYAVYDCK
|
8.3 | IC50 | 2 | — | |
MAUMVJHUMXPCFT
|
8.3 | IC50 | 2 | — | |
MWLPKZBBCRIXMO
|
8.3 | IC50 | 4 | — | |
NNTGHJBTOUDOGY
|
8.3 | IC50 | 2 | — | |
NYIZCWIYRUTEKV
|
8.3 | IC50 | 5 | — | |
GERYTDGNULKRJC
|
8.3 | IC50 | 2 | — | |
GLAVTOUIMCZWGE
|
8.3 | IC50 | 2 | — | |
PMVDOKGCDYKXLD
|
8.3 | IC50 | 2 | — | |
CVBUCTGSDPYFLF
|
8.3 | IC50 | 2 | — | |
FHNQKWOESOPUGN
|
8.3 | IC50 | 2 | — | |
JEBRWBXEAHSNTF
|
8.3 | Ki | 2 | — | |
MREBBDFKXMXJBV
|
8.3 | IC50 | 2 | — | |
OHOJPZUGJPTYSY
|
8.3 | Ki | 2 | — | |
SIXJMSJQDGDEAK
|
8.3 | IC50 | 2 | — | |
VVRIPMSPBSGFPZ
|
8.3 | IC50 | 3 | — | |
NCNWVDNQQKXAAM
|
8.3 | IC50 | 2 | — | |
NIBDXGIMKZXWGB
|
8.3 | IC50 | 2 | — | |
XHZIKHVYHSVYCX
|
8.3 | IC50 | 2 | — | |
ZWFUXTUZVCZUMC
|
8.3 | IC50 | 2 | — | |
HNZUOEFJYXSXOO
|
8.3 | IC50 | 2 | — | |
UPEGZTKVOGNGIP
|
8.3 | IC50 | 2 | — | |
FETXIQQMXPIQAE
|
8.3 | IC50 | 2 | — | |
IWUIDYZQPXSVJK
|
8.3 | IC50 | 2 | — | |
UIQZHYNNPYXEGY
|
8.3 | IC50 | 2 | — | |
UNDDSOFKUNBHJW
|
8.3 | IC50 | 2 | — | |
UXIFXRPPOKZVPG
|
8.3 | IC50 | 4 | — | |
WIADTCNCIOEKBT
|
8.3 | IC50 | 2 | — | |
WMAYUSHYHMSHFY
|
8.3 | IC50 | 6 | — | |
RBEBHTTXTRLDHD
|
8.2 | IC50 | 2 | — | |
ACYKBAYFNYDVSD
|
8.2 | IC50 | 2 | — | |
KTSCJCLXFWHLBQ
|
8.2 | IC50 | 4 | — |