Target Details
| UniProt AC | P05556 |
|---|---|
| Gene Symbol | ITGB1 |
| Protein Name | Integrin beta-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07974 (EGF_2) PF23105 (EGF_integrin) PF18372 (I-EGF_1) PF08725 (Integrin_b_cyt) PF07965 (Integrin_B_tail) PF00362 (Integrin_beta) PF17205 (PSI_integrin) |
Summary
- Multi-target molecules 1,572
- Clinical molecules 0
- Avg pChEMBL 7.77
KEGG Pathways (29)
- Arrhythmogenic right ventricular cardiomyopathy
- Axon guidance
- Bacterial invasion of epithelial cells
- Cell adhesion molecule (CAM) interaction
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Focal adhesion
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- IgSF CAM signaling
- Integrin signaling
- Leishmaniasis
- Leukocyte transendothelial migration
- PI3K-Akt signaling pathway
- Pathogenic Escherichia coli infection
- Pathways in cancer
- Pertussis
- Phagosome
- Platelet activation
- Proteoglycans in cancer
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Shigellosis
- Small cell lung cancer
- Tight junction
- Toxoplasmosis
- Virion - Rotavirus
- Yersinia infection
Active Molecules (1,572)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CUGPAWBXPURXLJ
|
10.7 | IC50 | 2 | — | |
DIZKXBOQGMAUNQ
|
10.7 | IC50 | 2 | — | |
FLCABSOQRLNJOS
|
10.4 | IC50 | 2 | — | |
OOYFOUHICCOHRQ
|
10.4 | IC50 | 2 | — | |
QPHITNQZXAUFEI
|
10.3 | IC50 | 2 | — | |
UWDSAWYVWRSKPP
|
10.3 | IC50 | 3 | — | |
OIMQYWATTYNADK
|
10.3 | IC50 | 2 | — | |
KXYAXQVLPNBUFO
|
10.2 | IC50 | 5 | — | |
GLJNHEQKGADNBQ
|
10.2 | IC50 | 2 | — | |
PRQQKDSSBGZCOL
|
10.2 | IC50 | 2 | — | |
QYLJBVNSXNPXCO
|
10.2 | IC50 | 3 | — | |
QYLJBVNSXNPXCO
|
10.2 | IC50 | 2 | — | |
WNKRETACHGJVKC
|
10.2 | IC50 | 3 | — | |
KANJDBFQNBEJPS
|
10.1 | IC50 | 2 | — | |
PALKXFSSVDMBNG
|
10.1 | IC50 | 3 | — | |
WIGSTHDXCOUXAO
|
10.1 | IC50 | 2 | — | |
QODRKUNYZZPWLY
|
10.1 | IC50 | 3 | — | |
GBQPAVGINXEHKX
|
10.1 | IC50 | 2 | — | |
JFSVPFIOVGIBHH
|
10.1 | IC50 | 2 | — | |
NYEPXWPYFSDIDX
|
10.1 | IC50 | 2 | — | |
RBYPTCVDQLQTJV
|
10.1 | IC50 | 3 | — | |
HBHMXAWUVLNJOM
|
10.0 | IC50 | 2 | — | |
IILNCTZMDUGCHL
|
10.0 | IC50 | 3 | — | |
JGCUUCXMZKFRKP
|
10.0 | IC50 | 3 | — | |
JUYLDRDBPRKGGI
|
10.0 | IC50 | 2 | — | |
LRJXQAWFNQBGLZ
|
10.0 | IC50 | 5 | — | |
LTMQOAYQBDWTIQ
|
10.0 | IC50 | 3 | — | |
NFLKOACGNNGCMZ
|
10.0 | IC50 | 2 | — | |
OPJBDVVJACDHPY
|
10.0 | IC50 | 3 | — | |
QLEPVYXTIMUWHF
|
10.0 | IC50 | 2 | — | |
RMGCKDRVLUITMO
|
10.0 | IC50 | 2 | — | |
RZDYGMVWRQQDRU
|
10.0 | IC50 | 2 | — | |
ASYDYYRPDBLCFU
|
10.0 | IC50 | 3 | — | |
ASYDYYRPDBLCFU
|
10.0 | IC50 | 3 | — | |
KFNKHVGWGQDFPY
|
10.0 | IC50 | 3 | — | |
MFMLIJVXQARVAA
|
10.0 | IC50 | 2 | — | |
AIALEJRVPVZVLO
|
9.9 | IC50 | 2 | — | |
AJZHUKFTTKIGAR
|
9.9 | IC50 | 3 | — | |
BBLPBZKWFCDYOO
|
9.9 | IC50 | 2 | — | |
CYRASILRFNUMJX
|
9.9 | IC50 | 3 | — | |
DHLWZPYEINGBFR
|
9.9 | IC50 | 3 | — | |
LDWAIULYHJTVQT
|
9.9 | IC50 | 3 | — | |
UERMUNMPBXMBHT
|
9.9 | IC50 | 3 | — | |
XDGSCLZNDKEXAE
|
9.9 | IC50 | 3 | — | |
BFLDDNSQCPEXPM
|
9.8 | IC50 | 2 | — | |
MCAIXYIMLUUTHW
|
9.8 | IC50 | 3 | — | |
MGKZYWCSUHALDJ
|
9.8 | IC50 | 3 | — | |
WOZSUXNJFSSYJW
|
9.8 | IC50 | 3 | — | |
HQJUSSKANCDJDV
|
9.8 | IC50 | 2 | — | |
HXCSQLRXMBOJCE
|
9.8 | IC50 | 3 | — |