Target Details
| UniProt AC | P05198 |
|---|---|
| Gene Symbol | EIF2S1 |
| Protein Name | Eukaryotic translation initiation factor 2 subunit 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07541 (EIF_2_alpha) PF00575 (S1) |
Summary
- Multi-target molecules 22
- Clinical molecules 0
- Avg pChEMBL 7.13
KEGG Pathways (15)
- Alzheimer disease
- Amyotrophic lateral sclerosis
- Apoptosis
- Autophagy - animal
- Hepatitis C
- Herpes simplex virus 1 infection
- Influenza A
- Lipid and atherosclerosis
- Measles
- Mitophagy - animal
- Non-alcoholic fatty liver disease
- Parkinson disease
- Pathways of neurodegeneration - multiple diseases
- Prion disease
- Protein processing in endoplasmic reticulum
Active Molecules (22)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YNDQMKBAYRFBMW
|
8.1 | IC50 | 2 | — | |
XHUVPVATWTZPPU
|
7.7 | IC50 | 2 | — | |
JSHFTMAPLMJGCF
|
7.6 | IC50 | 2 | — | |
ZAEWPVUVQVUGEE
|
7.6 | IC50 | 2 | — | |
BRIWRAFDHZTJPE
|
7.5 | IC50 | 2 | — | |
CVTISFUIJNOONP
|
7.4 | IC50 | 2 | — | |
WFLLOUGNTSBEON
|
7.4 | IC50 | 2 | — | |
VJSNNBDPTLXPPT
|
7.4 | IC50 | 2 | — | |
XMXNMDQZYHHSSJ
|
7.3 | IC50 | 2 | — | |
YXMQYIZUPKQHRP
|
7.3 | IC50 | 2 | — | |
GZISLAWEFNWGCT
|
7.3 | IC50 | 2 | — | |
XMJPZNCMRRFABT
|
7.2 | IC50 | 2 | — | |
LBLBTNIBKKNQAH
|
7.1 | IC50 | 2 | — | |
MWKSRKSEWLRPBL
|
7.1 | Kd | 1075 | — | |
XFMJNFJUBNDIMV
|
6.9 | IC50 | 2 | — | |
RPSNLKRQONAZHZ
|
6.7 | IC50 | 2 | — | |
BRIWRAFDHZTJPE
|
6.7 | IC50 | 2 | — | |
FYRWUAWBPDXQPZ
|
6.7 | IC50 | 2 | — | |
QXFDNMNTISNJLZ
|
6.5 | IC50 | 2 | — | |
PNRYWGAXPBKWAG
|
6.5 | IC50 | 2 | — | |
AZVXWPCFOZFXMJ
|
6.4 | IC50 | 2 | — | |
HZQGFXQCDQMBMH
|
6.2 | IC50 | 2 | — |