Target Details
| UniProt AC | P05129 |
|---|---|
| Gene Symbol | PRKCG |
| Protein Name | Protein kinase C gamma type |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF00168 (C2) PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 311
- Clinical molecules 119
- Avg pChEMBL 7.06
KEGG Pathways (64)
- African trypanosomiasis
- Aldosterone synthesis and secretion
- Aldosterone-regulated sodium reabsorption
- Amoebiasis
- Amphetamine addiction
- Calcium signaling pathway
- Chemical carcinogenesis - receptor activation
- Choline metabolism in cancer
- Cholinergic synapse
- Circadian entrainment
- Coronavirus disease - COVID-19
- Diabetic cardiomyopathy
- Dopaminergic synapse
- EGFR tyrosine kinase inhibitor resistance
- Endocrine and other factor-regulated calcium reabsorption
- ErbB signaling pathway
- Fc gamma R-mediated phagocytosis
- Focal adhesion
- GABAergic synapse
- Gap junction
- Gastric acid secretion
- Glioma
- Glutamatergic synapse
- GnRH secretion
- Growth hormone synthesis, secretion and action
- HIF-1 signaling pathway
- Hepatitis B
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- IgSF CAM signaling
- Inflammatory mediator regulation of TRP channels
- Insulin secretion
- Leukocyte transendothelial migration
- Long-term depression
- Long-term potentiation
- MAPK signaling pathway
- Melanogenesis
- MicroRNAs in cancer
- Morphine addiction
- Natural killer cell mediated cytotoxicity
- Neuroactive ligand signaling
- Neutrophil extracellular trap formation
- Non-small cell lung cancer
- Oxytocin signaling pathway
- Pancreatic secretion
- Parathyroid hormone synthesis, secretion and action
- Pathways in cancer
- Pathways of neurodegeneration - multiple diseases
- Phosphatidylinositol signaling system
- Proteoglycans in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Retrograde endocannabinoid signaling
- Salivary secretion
- Serotonergic synapse
- Sphingolipid signaling pathway
- Spinocerebellar ataxia
- Thyroid hormone signaling pathway
- Thyroid hormone synthesis
- VEGF signaling pathway
- Vascular smooth muscle contraction
- Wnt signaling pathway
- mTOR signaling pathway
Associated Diseases (1)
Active Molecules (311)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KLTAXINXABHYMC
|
6.6 | IC50 | 5 | — | |
KYCYRGUYNYCBAH
|
6.6 | IC50 | 7 | — | |
LAOIBIIMKUINJL
|
6.6 | IC50 | 12 | Yes | |
IXOVKVHWGKDXKQ
|
6.6 | IC50 | 12 | Yes | |
LHQWPYOYDRVMFI
|
6.6 | IC50 | 10 | Yes | |
ZEYTZKVCOZMUKL
|
6.6 | IC50 | 5 | — | |
BRZYOTMFHLERHD
|
6.5 | Ki | 17 | Yes | |
KLYPYTHLYUUKMT
|
6.5 | Ki | 4 | — | |
WPSBCJTXGDVGAZ
|
6.5 | IC50 | 5 | — | |
RVIJQMOQZFCSHL
|
6.5 | Ki | 8 | Yes | |
ARKNUCQRPYIUMU
|
6.5 | IC50 | 6 | — | |
SFDFKLDQKSPRHB
|
6.5 | IC50 | 15 | Yes | |
XNKIVXYFRPYKHO
|
6.5 | IC50 | 12 | Yes | |
ZCBUQCWBWNUWSU
|
6.5 | IC50 | 59 | — | |
ZOGSVRRXRLSQNC
|
6.5 | IC50 | 6 | — | |
FLEAYYMORDPWAJ
|
6.5 | Ki | 90 | — | |
IIMMUGRHSXMDBU
|
6.5 | IC50 | 4 | — | |
KRIUNPBAQZGFQA
|
6.5 | Ki | 76 | — | |
SBFPHSVZEXSHTL
|
6.5 | Ki | 62 | — | |
TVIALAOHRQNPOI
|
6.5 | IC50 | 12 | Yes | |
YEHCNYAQEBQCCS
|
6.5 | Ki | 74 | — | |
PXONMVAMARNSJO
|
6.5 | Ki | 4 | — | |
STEGBXHZVWLLAP
|
6.5 | IC50 | 6 | — | |
KOVNFJBXMBASSU
|
6.5 | IC50 | 4 | — | |
HPCPUHOULFPBCQ
|
6.5 | IC50 | 12 | Yes | |
JDZXLEPJWLCESI
|
6.5 | IC50 | 12 | Yes | |
RHBWAFDCVFMIFK
|
6.5 | IC50 | 12 | Yes | |
RPLXVENRWORMRX
|
6.4 | IC50 | 12 | Yes | |
JXDMRMYIFDKNHE
|
6.4 | IC50 | 4 | — | |
PEZLAFKDOMGSEL
|
6.4 | IC50 | 4 | — | |
PEZLAFKDOMGSEL
|
6.4 | IC50 | 4 | — | |
BMGQWWVMWDBQGC
|
6.4 | IC50 | 147 | Yes | |
CEMBEUHBOHDWPN
|
6.4 | IC50 | 4 | — | |
MQFYZWYYZGTHAN
|
6.4 | IC50 | 14 | — | |
UXKZMYMPEYJJKA
|
6.4 | IC50 | 5 | — | |
DKOCZDDCSUQYTF
|
6.4 | IC50 | 5 | — | |
GWJHMRBQEUHFOC
|
6.4 | Ki | 42 | — | |
HHLKZSJXDAZIGG
|
6.4 | IC50 | 10 | Yes | |
IJMSAWGGWOGISJ
|
6.4 | IC50 | 3 | — | |
VYXIZKJRRNWQAK
|
6.4 | IC50 | 6 | — | |
XFWUTMHVDGPWLH
|
6.4 | Ki | 75 | — | |
XYUFCXJZFZPEJD
|
6.4 | IC50 | 5 | — | |
XYUFCXJZFZPEJD
|
6.4 | IC50 | 4 | — | |
SIXGXRZCYDCNFL
|
6.4 | IC50 | 4 | — | |
KAJXOWFGKYKMMZ
|
6.4 | IC50 | 26 | Yes | |
MVPSDKPPZLPMBB
|
6.4 | Ki | 7 | Yes | |
QRBLWZIADYBYNA
|
6.4 | IC50 | 5 | — | |
ZFNQOYBHHLGQDV
|
6.3 | IC50 | 12 | Yes | |
BMBIKZHGTPMMMM
|
6.3 | IC50 | 14 | — | |
PQWWKDOKHDWZBH
|
6.3 | IC50 | 6 | — |