Target Details
| UniProt AC | P05129 |
|---|---|
| Gene Symbol | PRKCG |
| Protein Name | Protein kinase C gamma type |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF00168 (C2) PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 311
- Clinical molecules 119
- Avg pChEMBL 7.06
KEGG Pathways (64)
- African trypanosomiasis
- Aldosterone synthesis and secretion
- Aldosterone-regulated sodium reabsorption
- Amoebiasis
- Amphetamine addiction
- Calcium signaling pathway
- Chemical carcinogenesis - receptor activation
- Choline metabolism in cancer
- Cholinergic synapse
- Circadian entrainment
- Coronavirus disease - COVID-19
- Diabetic cardiomyopathy
- Dopaminergic synapse
- EGFR tyrosine kinase inhibitor resistance
- Endocrine and other factor-regulated calcium reabsorption
- ErbB signaling pathway
- Fc gamma R-mediated phagocytosis
- Focal adhesion
- GABAergic synapse
- Gap junction
- Gastric acid secretion
- Glioma
- Glutamatergic synapse
- GnRH secretion
- Growth hormone synthesis, secretion and action
- HIF-1 signaling pathway
- Hepatitis B
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- IgSF CAM signaling
- Inflammatory mediator regulation of TRP channels
- Insulin secretion
- Leukocyte transendothelial migration
- Long-term depression
- Long-term potentiation
- MAPK signaling pathway
- Melanogenesis
- MicroRNAs in cancer
- Morphine addiction
- Natural killer cell mediated cytotoxicity
- Neuroactive ligand signaling
- Neutrophil extracellular trap formation
- Non-small cell lung cancer
- Oxytocin signaling pathway
- Pancreatic secretion
- Parathyroid hormone synthesis, secretion and action
- Pathways in cancer
- Pathways of neurodegeneration - multiple diseases
- Phosphatidylinositol signaling system
- Proteoglycans in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Retrograde endocannabinoid signaling
- Salivary secretion
- Serotonergic synapse
- Sphingolipid signaling pathway
- Spinocerebellar ataxia
- Thyroid hormone signaling pathway
- Thyroid hormone synthesis
- VEGF signaling pathway
- Vascular smooth muscle contraction
- Wnt signaling pathway
- mTOR signaling pathway
Associated Diseases (1)
Active Molecules (311)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LUZOFMGZMUZSSK
|
6.9 | Ki | 8 | Yes | |
DRCBMJUPXHWGMN
|
6.8 | IC50 | 15 | Yes | |
MGQDMSJZRRHMFT
|
6.8 | IC50 | 6 | — | |
VEMLCWMDXJGJLI
|
6.8 | Ki | 8 | Yes | |
JWVXPOMGWPAEAJ
|
6.8 | IC50 | 10 | Yes | |
QNULKTUETCUJKC
|
6.8 | IC50 | 14 | Yes | |
CZIVUSJISIAXJB
|
6.8 | IC50 | 18 | — | |
ADMFLILDQJSEIK
|
6.8 | Ki | 72 | — | |
NNVINYYJNCKGRA
|
6.8 | IC50 | 5 | — | |
OOPMDKIRVTXOPT
|
6.8 | IC50 | 11 | — | |
JCHWETQOLSPUBV
|
6.8 | IC50 | 14 | — | |
MGQDMSJZRRHMFT
|
6.8 | IC50 | 6 | — | |
MGQDMSJZRRHMFT
|
6.8 | IC50 | 6 | — | |
JHKZENPNLYAVCT
|
6.8 | IC50 | 15 | Yes | |
OQSTWXKHTZWKLD
|
6.8 | IC50 | 15 | Yes | |
DQYBRTASHMYDJG
|
6.7 | IC50 | 13 | Yes | |
LGSHHKIOBFPSEK
|
6.7 | IC50 | 12 | Yes | |
QMGUOJYZJKLOLH
|
6.7 | IC50 | 21 | Yes | |
FUMCKNCUEAQHCV
|
6.7 | Ki | 103 | — | |
LRZYYIZFBXFSJB
|
6.7 | Ki | 69 | — | |
OWRXHGAFWZFFCW
|
6.7 | Ki | 113 | — | |
TWUWFRLZDWDJLT
|
6.7 | Ki | 10 | Yes | |
UAQJVFADAYIBGC
|
6.7 | Ki | 23 | — | |
NTXWXFSAJRMWNA
|
6.7 | IC50 | 15 | — | |
RAOJISQDGOOXTK
|
6.7 | IC50 | 14 | Yes | |
DNPFEENAAKLCMC
|
6.7 | IC50 | 6 | — | |
HCDKPFLBNVCSDB
|
6.7 | IC50 | 5 | — | |
HCDKPFLBNVCSDB
|
6.7 | IC50 | 5 | — | |
HIUHVDROHDSKTC
|
6.7 | Ki | 20 | — | |
PXONMVAMARNSJO
|
6.7 | Ki | 4 | — | |
MEXUTNIFSHFQRG
|
6.7 | IC50 | 21 | Yes | |
GZJKVFKNTQXSQM
|
6.7 | IC50 | 12 | Yes | |
PQWWKDOKHDWZBH
|
6.7 | IC50 | 6 | — | |
MZNUNTIEUOYNNT
|
6.6 | IC50 | 12 | Yes | |
OXEOHAXVZADDOC
|
6.6 | IC50 | 12 | Yes | |
CYRPAUWSHGGREB
|
6.6 | Ki | 8 | Yes | |
YSVVBGPTTSJYPA
|
6.6 | IC50 | 12 | Yes | |
BPNUQXPIQBZCMR
|
6.6 | Ki | 60 | — | |
KOZFSFOOLUUIGY
|
6.6 | IC50 | 26 | — | |
LMIPLKOPDQGFNB
|
6.6 | IC50 | 4 | — | |
NHHQJBCNYHBUSI
|
6.6 | Ki | 220 | — | |
NIUBYBAPAVVDMG
|
6.6 | IC50 | 6 | — | |
NIUBYBAPAVVDMG
|
6.6 | IC50 | 6 | — | |
OUJZYQBEFNDJQN
|
6.6 | Ki | 71 | — | |
RKUKAACYUCUJEE
|
6.6 | Ki | 58 | — | |
SSZFVGXDYBMVDD
|
6.6 | IC50 | 12 | Yes | |
TXVBBLNFLUZGIT
|
6.6 | IC50 | 6 | — | |
XPHWIERLJBFPFV
|
6.6 | Ki | 69 | — | |
YOVNFNXUCOWYSG
|
6.6 | Ki | 33 | Yes | |
PBCZSGKMGDDXIJ
|
6.6 | IC50 | 12 | Yes |