Target Details
| UniProt AC | P05129 |
|---|---|
| Gene Symbol | PRKCG |
| Protein Name | Protein kinase C gamma type |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF00168 (C2) PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 311
- Clinical molecules 119
- Avg pChEMBL 7.06
KEGG Pathways (64)
- African trypanosomiasis
- Aldosterone synthesis and secretion
- Aldosterone-regulated sodium reabsorption
- Amoebiasis
- Amphetamine addiction
- Calcium signaling pathway
- Chemical carcinogenesis - receptor activation
- Choline metabolism in cancer
- Cholinergic synapse
- Circadian entrainment
- Coronavirus disease - COVID-19
- Diabetic cardiomyopathy
- Dopaminergic synapse
- EGFR tyrosine kinase inhibitor resistance
- Endocrine and other factor-regulated calcium reabsorption
- ErbB signaling pathway
- Fc gamma R-mediated phagocytosis
- Focal adhesion
- GABAergic synapse
- Gap junction
- Gastric acid secretion
- Glioma
- Glutamatergic synapse
- GnRH secretion
- Growth hormone synthesis, secretion and action
- HIF-1 signaling pathway
- Hepatitis B
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- IgSF CAM signaling
- Inflammatory mediator regulation of TRP channels
- Insulin secretion
- Leukocyte transendothelial migration
- Long-term depression
- Long-term potentiation
- MAPK signaling pathway
- Melanogenesis
- MicroRNAs in cancer
- Morphine addiction
- Natural killer cell mediated cytotoxicity
- Neuroactive ligand signaling
- Neutrophil extracellular trap formation
- Non-small cell lung cancer
- Oxytocin signaling pathway
- Pancreatic secretion
- Parathyroid hormone synthesis, secretion and action
- Pathways in cancer
- Pathways of neurodegeneration - multiple diseases
- Phosphatidylinositol signaling system
- Proteoglycans in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Retrograde endocannabinoid signaling
- Salivary secretion
- Serotonergic synapse
- Sphingolipid signaling pathway
- Spinocerebellar ataxia
- Thyroid hormone signaling pathway
- Thyroid hormone synthesis
- VEGF signaling pathway
- Vascular smooth muscle contraction
- Wnt signaling pathway
- mTOR signaling pathway
Associated Diseases (1)
Active Molecules (311)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GPGZMTPPOHCJRE
|
7.8 | IC50 | 16 | Yes | |
MKPSMRQVGPTYRL
|
7.8 | IC50 | 6 | — | |
SMZYTCQRZVNFFJ
|
7.8 | IC50 | 16 | Yes | |
YIZRPXUMLQCIMQ
|
7.8 | IC50 | 9 | — | |
CHTMRWQLNNRRFJ
|
7.8 | Ki | 70 | — | |
CXSQMXRQOZZFLD
|
7.8 | IC50 | 18 | — | |
PBCZSGKMGDDXIJ
|
7.8 | IC50 | 68 | Yes | |
FXGHOAZJQNLNFD
|
7.8 | IC50 | 13 | Yes | |
HKSZLNNOFSGOKW
|
7.7 | IC50 | 49 | Yes | |
XYUFCXJZFZPEJD
|
7.7 | IC50 | 9 | — | |
AZIMEXGKUWHPQV
|
7.7 | IC50 | 12 | Yes | |
FSBMWCWKNXQVMP
|
7.7 | IC50 | 12 | Yes | |
HSZCSAUAGLABDS
|
7.7 | Ki | 5 | — | |
OWJIKBAZUBPKGN
|
7.7 | IC50 | 6 | — | |
OWJIKBAZUBPKGN
|
7.7 | IC50 | 7 | — | |
VXYDJXMHISGSDA
|
7.7 | Ki | 59 | — | |
XUTMONHBGYHWES
|
7.7 | Ki | 5 | — | |
YUKJJLKBBAFYNN
|
7.7 | IC50 | 12 | Yes | |
KPCVAMMFCPIUIU
|
7.5 | IC50 | 12 | Yes | |
OAVGBZOFDPFGPJ
|
7.5 | IC50 | 42 | Yes | |
OWJIKBAZUBPKGN
|
7.5 | IC50 | 6 | — | |
OWJIKBAZUBPKGN
|
7.5 | IC50 | 7 | — | |
XXDWSQPJTJZKSJ
|
7.5 | IC50 | 12 | Yes | |
XYUFCXJZFZPEJD
|
7.5 | IC50 | 9 | — | |
XYUFCXJZFZPEJD
|
7.5 | IC50 | 23 | Yes | |
ZZSBPGIGIUFJRA
|
7.5 | IC50 | 15 | Yes | |
FELQRVDTGNDOSI
|
7.5 | IC50 | 15 | Yes | |
OARXLGLBMAHALM
|
7.5 | IC50 | 12 | Yes | |
BSFNGHCTZDCQBF
|
7.5 | Ki | 93 | — | |
MYOUXQLHWTWXON
|
7.5 | IC50 | 16 | Yes | |
ZKHDDJKHTPLPOQ
|
7.5 | Ki | 62 | — | |
YDZJEODKNRAYMA
|
7.5 | IC50 | 12 | Yes | |
XYUFCXJZFZPEJD
|
7.5 | IC50 | 6 | — | |
GQCWIZZVARXZGR
|
7.5 | IC50 | 6 | — | |
ZYUGNHPOVKADFZ
|
7.5 | IC50 | 11 | — | |
HPBJQOWLAKYNDM
|
7.4 | IC50 | 15 | Yes | |
AMSOPBXQXSAAAC
|
7.4 | IC50 | 12 | Yes | |
DASVAQCTVIQROX
|
7.4 | Ki | 8 | Yes | |
WQEXBJWFPAMSGJ
|
7.4 | Ki | 8 | Yes | |
GQCWIZZVARXZGR
|
7.4 | IC50 | 6 | — | |
KJGUOQMSLKZPAT
|
7.4 | IC50 | 17 | Yes | |
MKPSMRQVGPTYRL
|
7.4 | IC50 | 5 | — | |
USEYXZSHZLLAJS
|
7.4 | IC50 | 6 | — | |
VWVYILCFSYNJHF
|
7.4 | IC50 | 49 | — | |
WOFBHAKTZOZODW
|
7.4 | IC50 | 6 | — | |
XSRHBCYNCKAFKS
|
7.4 | Ki | 45 | — | |
NTUVEMUMVHHACY
|
7.4 | IC50 | 12 | Yes | |
KDIRIFZBLUSLJU
|
7.4 | Ki | 5 | — | |
CKJRKRPDNLRZPQ
|
7.3 | IC50 | 6 | — | |
KOZFSFOOLUUIGY
|
7.3 | IC50 | 88 | Yes |