Target Details
| UniProt AC | P05107 |
|---|---|
| Gene Symbol | ITGB2 |
| Protein Name | Integrin beta-2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF23105 (EGF_integrin) PF08725 (Integrin_b_cyt) PF07965 (Integrin_B_tail) PF00362 (Integrin_beta) PF17205 (PSI_integrin) |
Summary
- Multi-target molecules 373
- Clinical molecules 0
- Avg pChEMBL 7.14
KEGG Pathways (21)
- Amoebiasis
- Cell adhesion molecule (CAM) interaction
- Complement and coagulation cascades
- Hippo signaling pathway
- Human T-cell leukemia virus 1 infection
- IgSF CAM signaling
- Integrin signaling
- Legionellosis
- Leishmaniasis
- Leukocyte transendothelial migration
- Malaria
- Natural killer cell mediated cytotoxicity
- Neutrophil extracellular trap formation
- Pertussis
- Phagosome
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Rheumatoid arthritis
- Staphylococcus aureus infection
- Tuberculosis
- Viral myocarditis
Associated Diseases (1)
Active Molecules (373)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IVETWPTYQWRCOV
|
6.4 | Kd | 3 | — | |
FLEDTAVZFHUYSW
|
6.4 | IC50 | 3 | — | |
GKTUFNINEUKFJG
|
6.4 | IC50 | 3 | — | |
JPIBRKWWCXXBBJ
|
6.4 | IC50 | 3 | — | |
DDJGJQWKZJMZCL
|
6.4 | IC50 | 3 | — | |
GMDRWNJYSVNFBO
|
6.4 | IC50 | 3 | — | |
RCJLHHUGMJBOQG
|
6.3 | IC50 | 3 | — | |
FAEVSCKIBUDMQJ
|
6.3 | IC50 | 3 | — | |
GUXYQKMGUHCFDG
|
6.3 | IC50 | 3 | — | |
XIVLZMACKMSZRH
|
6.3 | IC50 | 3 | — | |
FRTCDBYRRZDOQQ
|
6.3 | IC50 | 3 | — | |
QUFQVFKQRMTIMD
|
6.3 | IC50 | 3 | — | |
XXLJXHUHENVDCY
|
6.3 | IC50 | 3 | — | |
BYQWOSKTUPJKFV
|
6.3 | IC50 | 3 | — | |
COVPLULNDBDXTN
|
6.3 | IC50 | 3 | — | |
YZCNYQLRQDZAIE
|
6.3 | IC50 | 3 | — | |
JLPFLAVJCXFYQO
|
6.3 | IC50 | 3 | — | |
MTAOLVAODYGSDX
|
6.3 | IC50 | 3 | — | |
PAOXPBIXQUNYMI
|
6.3 | IC50 | 3 | — | |
KHWFLVYYKGXMPW
|
6.3 | IC50 | 3 | — | |
OLMNMKWZYAOBIK
|
6.3 | IC50 | 3 | — | |
HOJGBSXDHZVYRK
|
6.2 | IC50 | 3 | — | |
AVYYYDWRPGSZGL
|
6.2 | IC50 | 3 | — | |
GZUBGTRIHHDYOX
|
6.2 | IC50 | 3 | — | |
MOPRGMKHXDVBQR
|
6.2 | IC50 | 3 | — | |
AQVUSOQZBUOAJM
|
6.2 | IC50 | 3 | — | |
AYINYYMJNHOUSM
|
6.2 | IC50 | 3 | — | |
BDMKWKGKWYADLX
|
6.2 | IC50 | 3 | — | |
JFWCMDPBPZTELG
|
6.2 | IC50 | 3 | — | |
KEQWSKKEOZLWRV
|
6.2 | IC50 | 3 | — | |
LFNWSXGKAAHEMT
|
6.2 | IC50 | 3 | — | |
NTQOVYVRCPMWAF
|
6.2 | IC50 | 3 | — | |
SLYGCFGQHBIXPM
|
6.2 | IC50 | 3 | — | |
LXBNAFUQTGPRDK
|
6.2 | Kd | 3 | — | |
NZDSKVKNJZPPBI
|
6.2 | IC50 | 3 | — | |
PMUGSFJFKNRORH
|
6.2 | IC50 | 3 | — | |
RKPWNENDRHTTBF
|
6.2 | IC50 | 3 | — | |
CWERXZGWAYOKSY
|
6.2 | IC50 | 3 | — | |
FXYDXLJEJBXFBD
|
6.2 | IC50 | 7 | — | |
PUAUSJUWVGDGCP
|
6.2 | IC50 | 3 | — | |
VDCWKOMRFTYIHX
|
6.2 | IC50 | 3 | — | |
XZXXUNSFXFQLLU
|
6.2 | IC50 | 3 | — | |
JXXZCGNZJULUEM
|
6.1 | IC50 | 3 | — | |
TXMYNHMEJQOXEL
|
6.1 | IC50 | 3 | — | |
YYCCOHSORPUJOI
|
6.1 | IC50 | 3 | — | |
DEQNAOBMFIOGRH
|
6.1 | IC50 | 3 | — | |
GKARTWDJGSTNQC
|
6.1 | IC50 | 3 | — | |
MDRVMCFSALAITN
|
6.1 | IC50 | 3 | — | |
MTCSXDMZKVZCAO
|
6.1 | Kd | 3 | — | |
WBTAHXUCBNIOHJ
|
6.1 | IC50 | 3 | — |